RU92016490A - Новые 2-сахаринилметил(арил и арокси)ацетаты, применимые в качестве ингибиторов протеолитических ферментов, их композиции и способ их применения - Google Patents

Новые 2-сахаринилметил(арил и арокси)ацетаты, применимые в качестве ингибиторов протеолитических ферментов, их композиции и способ их применения

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Publication number
RU92016490A
RU92016490A RU92016490/33A RU92016490A RU92016490A RU 92016490 A RU92016490 A RU 92016490A RU 92016490/33 A RU92016490/33 A RU 92016490/33A RU 92016490 A RU92016490 A RU 92016490A RU 92016490 A RU92016490 A RU 92016490A
Authority
RU
Russia
Prior art keywords
aryl
acetates
applicable
saharinilmethil
aroxy
Prior art date
Application number
RU92016490/33A
Other languages
English (en)
Other versions
RU2081871C1 (ru
Inventor
Гамильтон Лэйтимер Ли
Поль Данлэп Ричард
Original Assignee
Стерлинг Уинтроп Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Стерлинг Уинтроп Инк. filed Critical Стерлинг Уинтроп Инк.
Publication of RU92016490A publication Critical patent/RU92016490A/ru
Application granted granted Critical
Publication of RU2081871C1 publication Critical patent/RU2081871C1/ru

Links

Claims (1)

  1. 4-R4-R5-2-Сахаринилметил(арил- и арилокси)ацетаты, применимые для лечения перерожденных заболеваний, получают реакцией 4-R4-R5-2-галоидметилсахарин с арил- или арилоксиуксусной кислотой в присутствии акцептора кислоты.
RU9292016490A 1991-12-30 1992-12-29 2-сахаринилметил(арил или арилокси) ацетаты, или их соли, образованные добавлением кислот к этим соединениям основного характера, или их соли, образованные добавлением оснований к этим соединениям кислотного характера, и фармацевтическая композиция, ингибирующая активность протеолитических ферментов RU2081871C1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US81574091A 1991-12-30 1991-12-30
US815740 1991-12-30

Publications (2)

Publication Number Publication Date
RU92016490A true RU92016490A (ru) 1995-06-19
RU2081871C1 RU2081871C1 (ru) 1997-06-20

Family

ID=25218721

Family Applications (1)

Application Number Title Priority Date Filing Date
RU9292016490A RU2081871C1 (ru) 1991-12-30 1992-12-29 2-сахаринилметил(арил или арилокси) ацетаты, или их соли, образованные добавлением кислот к этим соединениям основного характера, или их соли, образованные добавлением оснований к этим соединениям кислотного характера, и фармацевтическая композиция, ингибирующая активность протеолитических ферментов

Country Status (17)

Country Link
US (3) US5385923A (ru)
EP (1) EP0550112A1 (ru)
JP (1) JPH05255286A (ru)
AU (1) AU651746B2 (ru)
CA (1) CA2086348A1 (ru)
CZ (1) CZ386992A3 (ru)
FI (1) FI925946A (ru)
HU (2) HUT65736A (ru)
IL (1) IL104259A (ru)
MX (1) MX9207274A (ru)
MY (1) MY108926A (ru)
NO (1) NO303446B1 (ru)
NZ (1) NZ245586A (ru)
PH (1) PH30411A (ru)
RU (1) RU2081871C1 (ru)
SG (1) SG48025A1 (ru)
TW (1) TW226016B (ru)

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US20090053221A1 (en) * 2006-01-17 2009-02-26 Cheung Nai-Kong V Immune response enhancing glucan
HRP20171415T4 (hr) 2009-06-25 2023-03-03 Alkermes Pharma Ireland Limited Heterociklični spojevi za liječenje neuroloških i psiholoških poremećaja
WO2010151711A1 (en) 2009-06-25 2010-12-29 Alkermes, Inc. Prodrugs of nh-acidic compounds
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EP2585066B1 (en) 2010-06-24 2018-09-26 Alkermes Pharma Ireland Limited Prodrugs of nh-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives
US9034867B2 (en) 2011-03-18 2015-05-19 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising sorbitan esters
NZ722096A (en) 2011-12-15 2016-11-25 Alkermes Pharma Ireland Ltd Prodrugs of secondary amine compounds
CA2867137C (en) 2012-03-19 2020-12-08 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising aripiprazole prodrugs and benzyl alcohol
JP6471089B2 (ja) 2012-03-19 2019-02-13 アルカームス ファーマ アイルランド リミテッド 脂肪酸エステルを含む医薬組成物
JP6219918B2 (ja) 2012-03-19 2017-10-25 アルカームス ファーマ アイルランド リミテッド グリセロールエステルを含む医薬組成物
ES2792149T3 (es) 2012-09-19 2020-11-10 Alkermes Pharma Ireland Ltd Composiciones farmacéuticas que tienen estabilidad de almacenamiento mejorada
MX2016008494A (es) 2013-12-31 2016-10-28 Saint Gobain Abrasives Inc Articulo abrasivo que incluye partículas abrasivas perfiladas.
US20150253127A1 (en) * 2014-03-04 2015-09-10 Honeywell Asca Inc. Thickness Determination of Web Product by Mid-infrared Wavelength Scanning Interferometry
MX2016012041A (es) 2014-03-20 2017-01-19 Alkermes Pharma Ireland Ltd Formulaciones de aripiprazol que tienen mayores velocidades de inyeccion.
US10346168B2 (en) 2015-06-26 2019-07-09 Microsoft Technology Licensing, Llc Decoupled processor instruction window and operand buffer
JP7384812B2 (ja) 2018-03-05 2023-11-21 アルカームス ファーマ アイルランド リミテッド アリピプラゾール投与戦略

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