RU2688167C1 - Применение изоксазолиновых соединений на домашней птице - Google Patents
Применение изоксазолиновых соединений на домашней птице Download PDFInfo
- Publication number
- RU2688167C1 RU2688167C1 RU2016129272A RU2016129272A RU2688167C1 RU 2688167 C1 RU2688167 C1 RU 2688167C1 RU 2016129272 A RU2016129272 A RU 2016129272A RU 2016129272 A RU2016129272 A RU 2016129272A RU 2688167 C1 RU2688167 C1 RU 2688167C1
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- Prior art keywords
- cas
- poultry
- isoxazoline compound
- trifluoromethyl
- drinking water
- Prior art date
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- 244000144977 poultry Species 0.000 title claims abstract description 70
- 150000002547 isoxazolines Chemical class 0.000 title description 18
- -1 isoxazoline compound Chemical class 0.000 claims abstract description 91
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- MLBZKOGAMRTSKP-UHFFFAOYSA-N fluralaner Chemical compound C1=C(C(=O)NCC(=O)NCC(F)(F)F)C(C)=CC(C=2CC(ON=2)(C=2C=C(Cl)C=C(Cl)C=2)C(F)(F)F)=C1 MLBZKOGAMRTSKP-UHFFFAOYSA-N 0.000 claims abstract description 36
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- FLEFKKUZMDEUIP-QFIPXVFZSA-N 1-[6-[(5s)-5-(3,5-dichloro-4-fluorophenyl)-5-(trifluoromethyl)-4h-1,2-oxazol-3-yl]spiro[1h-2-benzofuran-3,3'-azetidine]-1'-yl]-2-methylsulfonylethanone Chemical compound C1N(C(=O)CS(=O)(=O)C)CC21C1=CC=C(C=3C[C@](ON=3)(C=3C=C(Cl)C(F)=C(Cl)C=3)C(F)(F)F)C=C1CO2 FLEFKKUZMDEUIP-QFIPXVFZSA-N 0.000 claims abstract description 7
- HDKWFBCPLKNOCK-SFHVURJKSA-N 3-methyl-n-[2-oxo-2-(2,2,2-trifluoroethylamino)ethyl]-5-[(5s)-5-(3,4,5-trichlorophenyl)-5-(trifluoromethyl)-4h-1,2-oxazol-3-yl]thiophene-2-carboxamide Chemical compound S1C(C(=O)NCC(=O)NCC(F)(F)F)=C(C)C=C1C1=NO[C@](C(F)(F)F)(C=2C=C(Cl)C(Cl)=C(Cl)C=2)C1 HDKWFBCPLKNOCK-SFHVURJKSA-N 0.000 claims abstract description 7
- OXDDDHGGRFRLEE-UHFFFAOYSA-N 4-[5-[3-chloro-5-(trifluoromethyl)phenyl]-5-(trifluoromethyl)-4h-1,2-oxazol-3-yl]-n-[2-oxo-2-(2,2,2-trifluoroethylamino)ethyl]naphthalene-1-carboxamide Chemical compound C12=CC=CC=C2C(C(=O)NCC(=O)NCC(F)(F)F)=CC=C1C(C1)=NOC1(C(F)(F)F)C1=CC(Cl)=CC(C(F)(F)F)=C1 OXDDDHGGRFRLEE-UHFFFAOYSA-N 0.000 claims abstract description 5
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Classifications
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
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- A—HUMAN NECESSITIES
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- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
- A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
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- A—HUMAN NECESSITIES
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- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Zoology (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Plant Pathology (AREA)
- Environmental Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP13199007.9 | 2013-12-20 | ||
| EP13199007 | 2013-12-20 | ||
| PCT/EP2014/078636 WO2015091900A1 (en) | 2013-12-20 | 2014-12-19 | Use of isoxazoline derivatives for the treatment or prevention of arthropod infestations in poultry |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2019114185A Division RU2796536C9 (ru) | 2013-12-20 | 2014-12-19 | Применение изоксазолиновых соединений на домашней птице |
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| RU2016129272A RU2016129272A (ru) | 2018-01-25 |
| RU2688167C1 true RU2688167C1 (ru) | 2019-05-20 |
Family
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| RU2016129272A RU2688167C1 (ru) | 2013-12-20 | 2014-12-19 | Применение изоксазолиновых соединений на домашней птице |
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| EP (2) | EP3878281B1 (OSRAM) |
| JP (1) | JP6506763B2 (OSRAM) |
| CN (2) | CN110839641A (OSRAM) |
| BR (1) | BR112016014216B1 (OSRAM) |
| ES (2) | ES2874054T3 (OSRAM) |
| HU (2) | HUE063842T2 (OSRAM) |
| MX (2) | MX376210B (OSRAM) |
| PL (2) | PL3082806T3 (OSRAM) |
| PT (1) | PT3082806T (OSRAM) |
| RU (1) | RU2688167C1 (OSRAM) |
| WO (1) | WO2015091900A1 (OSRAM) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP4430947A1 (en) | 2023-03-17 | 2024-09-18 | Przedsiebiorstwo Wielobranzowe "Vet-Agro" Sp. Z O.O. | Therapeutic use of isoxazoline compounds, composition of isoxazoline compounds and kit for therapeutic use |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX376210B (es) * | 2013-12-20 | 2025-03-07 | Intervet Int Bv | Uso de derivados de isoxazolina para el tratamiento o prevención de infestaciones por artrópodos en aves de corral. |
| JP6581586B2 (ja) * | 2013-12-20 | 2019-09-25 | インターベット インターナショナル ベー． フェー． | イソオキサゾリン組成物および動物における寄生虫侵襲の予防または処置におけるその使用 |
| HUE059228T2 (hu) * | 2015-06-23 | 2022-10-28 | Intervet Int Bv | E vitamint tartalmazó izoxazolin oldat, fertõtlenített ivóvízzel való felhasználásra |
| WO2018039508A1 (en) * | 2016-08-25 | 2018-03-01 | Merial, Inc. | Method for reducing unwanted effects in parasiticidal treatments |
| TWI834690B (zh) * | 2018-07-18 | 2024-03-11 | 美商富曼西公司 | 用於防治無脊椎動物害蟲之異噁唑啉化合物 |
| TW202012399A (zh) * | 2018-09-12 | 2020-04-01 | 美商富曼西公司 | 用於防制無脊椎動物害蟲之異口咢唑啉化合物 |
| WO2020201440A1 (en) * | 2019-04-03 | 2020-10-08 | Virbac | Low dose fluralaner compositions for protection against parasitic invertebrate pest |
| BR112022011046A2 (pt) * | 2019-12-16 | 2022-08-23 | Intervet Int Bv | Composição para controle de piolhos em avinos |
| EP4077286A1 (en) | 2019-12-18 | 2022-10-26 | Elanco Tiergesundheit AG | Isoxazoline derivatives as pesticides |
| WO2022020585A1 (en) | 2020-07-24 | 2022-01-27 | Elanco Us Inc. | Process for making an isoxazoline compound and intermediate thereof |
| US11903962B1 (en) * | 2023-05-07 | 2024-02-20 | Michael Farber | Isoxazoline complexes and compositions thereof |
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| WO2013050302A1 (en) * | 2011-10-03 | 2013-04-11 | Syngenta Participations Ag | Isoxazoline derivatives as insecticidal compounds |
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| WO2007053902A1 (en) | 2005-11-10 | 2007-05-18 | Bomac Animal Health Pty Limited | Method of treating parasites |
| TW200803740A (en) | 2005-12-16 | 2008-01-16 | Du Pont | 5-aryl isoxazolines for controlling invertebrate pests |
| TWI412322B (zh) | 2005-12-30 | 2013-10-21 | Du Pont | 控制無脊椎害蟲之異唑啉 |
| TWI430995B (zh) | 2007-06-26 | 2014-03-21 | Du Pont | 萘異唑啉無脊椎有害動物控制劑 |
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| EP2364147A2 (en) | 2008-11-19 | 2011-09-14 | Merial Limited | Compositions comprising 1-arylpyrazole alone or in combination with formamidine for the treatment of parasitic infection |
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| US20130203591A1 (en) * | 2010-06-09 | 2013-08-08 | Syngenta Crop Protection Llc | Pesticidal mixtures including isoxazoline derivatives |
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2014
- 2014-12-19 MX MX2016008119A patent/MX376210B/es active IP Right Grant
- 2014-12-19 CN CN201911241170.8A patent/CN110839641A/zh active Pending
- 2014-12-19 ES ES14816243T patent/ES2874054T3/es active Active
- 2014-12-19 PL PL14816243T patent/PL3082806T3/pl unknown
- 2014-12-19 US US15/105,197 patent/US10272071B2/en active Active
- 2014-12-19 BR BR112016014216-0A patent/BR112016014216B1/pt active IP Right Grant
- 2014-12-19 EP EP21166872.8A patent/EP3878281B1/en active Active
- 2014-12-19 PT PT148162431T patent/PT3082806T/pt unknown
- 2014-12-19 EP EP14816243.1A patent/EP3082806B1/en active Active
- 2014-12-19 HU HUE21166872A patent/HUE063842T2/hu unknown
- 2014-12-19 RU RU2016129272A patent/RU2688167C1/ru active
- 2014-12-19 WO PCT/EP2014/078636 patent/WO2015091900A1/en not_active Ceased
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2016
- 2016-06-17 MX MX2020010997A patent/MX2020010997A/es unknown
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2019
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2020
- 2020-04-15 US US16/849,487 patent/US11304934B2/en active Active
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2022
- 2022-03-08 US US17/653,950 patent/US12128032B2/en active Active
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| WO2009003075A1 (en) * | 2007-06-27 | 2008-12-31 | E.I. Du Pont De Nemours And Company | Animal pest control method |
| WO2012107533A1 (en) * | 2011-02-10 | 2012-08-16 | Novartis Ag | Isoxazoline derivatives for controlling invertebrate pests |
| WO2013026695A1 (en) * | 2011-08-25 | 2013-02-28 | Syngenta Participations Ag | Isoxazoline derivatives as insecticidal compounds |
| WO2013026931A1 (en) * | 2011-08-25 | 2013-02-28 | Syngenta Participations Ag | Isoxazoline derivatives as insecticidal compounds |
| WO2013050302A1 (en) * | 2011-10-03 | 2013-04-11 | Syngenta Participations Ag | Isoxazoline derivatives as insecticidal compounds |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP4430947A1 (en) | 2023-03-17 | 2024-09-18 | Przedsiebiorstwo Wielobranzowe "Vet-Agro" Sp. Z O.O. | Therapeutic use of isoxazoline compounds, composition of isoxazoline compounds and kit for therapeutic use |
Also Published As
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| ES2950885T3 (es) | 2023-10-16 |
| PL3082806T3 (pl) | 2021-09-13 |
| US20190192486A1 (en) | 2019-06-27 |
| US20220193040A1 (en) | 2022-06-23 |
| HUE063842T2 (hu) | 2024-02-28 |
| CN110839641A (zh) | 2020-02-28 |
| PT3082806T (pt) | 2021-06-04 |
| US10272071B2 (en) | 2019-04-30 |
| US20160317502A1 (en) | 2016-11-03 |
| PL3878281T3 (pl) | 2023-07-31 |
| HUE055444T2 (hu) | 2021-11-29 |
| ES2874054T3 (es) | 2021-11-04 |
| EP3082806A1 (en) | 2016-10-26 |
| RU2019114185A (ru) | 2019-06-27 |
| EP3878281A1 (en) | 2021-09-15 |
| BR112016014216B1 (pt) | 2022-08-30 |
| RU2016129272A (ru) | 2018-01-25 |
| WO2015091900A1 (en) | 2015-06-25 |
| JP6506763B2 (ja) | 2019-04-24 |
| US11304934B2 (en) | 2022-04-19 |
| CN105979944A (zh) | 2016-09-28 |
| US10653675B2 (en) | 2020-05-19 |
| EP3878281B1 (en) | 2023-05-24 |
| US20200237727A1 (en) | 2020-07-30 |
| US12128032B2 (en) | 2024-10-29 |
| BR112016014216A2 (OSRAM) | 2017-08-08 |
| EP3082806B1 (en) | 2021-05-12 |
| MX2020010997A (es) | 2020-11-09 |
| MX2016008119A (es) | 2016-09-16 |
| JP2016540028A (ja) | 2016-12-22 |
| MX376210B (es) | 2025-03-07 |
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