RU2499583C2 - Заместительное трансдермальное введение фентанила один раз в день - Google Patents

Заместительное трансдермальное введение фентанила один раз в день Download PDF

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Publication number
RU2499583C2
RU2499583C2 RU2010119491/14A RU2010119491A RU2499583C2 RU 2499583 C2 RU2499583 C2 RU 2499583C2 RU 2010119491/14 A RU2010119491/14 A RU 2010119491/14A RU 2010119491 A RU2010119491 A RU 2010119491A RU 2499583 C2 RU2499583 C2 RU 2499583C2
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RU
Russia
Prior art keywords
fentanyl
day
patch
reservoir
drug
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RU2010119491/14A
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English (en)
Russian (ru)
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RU2010119491A (ru
Inventor
Стефен С. ХВАНГ
Роберт М. ГЕЙЛ
Original Assignee
Алза Корпорейшн
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40567772&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RU2499583(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Алза Корпорейшн filed Critical Алза Корпорейшн
Publication of RU2010119491A publication Critical patent/RU2010119491A/ru
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • A61K9/7061—Polyacrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4468—Non condensed piperidines, e.g. piperocaine having a nitrogen directly attached in position 4, e.g. clebopride, fentanyl
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids

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  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Hydrogenated Pyridines (AREA)
RU2010119491/14A 2007-10-15 2008-10-15 Заместительное трансдермальное введение фентанила один раз в день RU2499583C2 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US97991107P 2007-10-15 2007-10-15
US60/979,911 2007-10-15
PCT/US2008/080029 WO2009052204A1 (en) 2007-10-15 2008-10-15 Once-a-day replacement transdermal administration of fentanyl

Publications (2)

Publication Number Publication Date
RU2010119491A RU2010119491A (ru) 2011-11-27
RU2499583C2 true RU2499583C2 (ru) 2013-11-27

Family

ID=40567772

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2010119491/14A RU2499583C2 (ru) 2007-10-15 2008-10-15 Заместительное трансдермальное введение фентанила один раз в день

Country Status (10)

Country Link
US (3) US20090258061A1 (enExample)
EP (1) EP2207507B1 (enExample)
JP (6) JP5687901B2 (enExample)
KR (1) KR101583680B1 (enExample)
CN (2) CN101902996B (enExample)
AU (5) AU2008312507B2 (enExample)
MY (3) MY188123A (enExample)
NZ (1) NZ584190A (enExample)
RU (1) RU2499583C2 (enExample)
WO (1) WO2009052204A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2499583C2 (ru) 2007-10-15 2013-11-27 Алза Корпорейшн Заместительное трансдермальное введение фентанила один раз в день
CN101925355B (zh) * 2008-01-28 2013-05-29 帝国制药株式会社 含芬太尼的外用贴剂
CN102026629B (zh) * 2008-03-25 2015-01-14 帝国制药株式会社 透皮吸收制剂
DE102014013448A1 (de) * 2014-09-16 2016-03-17 Alfred E. Tiefenbacher (Gmbh & Co. Kg) Transdermales Therapeutisches System umfassend Buprenorphin
EP3233081B1 (en) * 2014-12-19 2021-09-22 Kindeva Drug Delivery L.P. Transdermal drug delivery device including fentanyl
MX2022000274A (es) * 2019-07-11 2022-02-03 Henkel Ag & Co Kgaa Polimero acrilico y composiciones adhesivas.
CN110693857B (zh) * 2019-10-17 2023-08-11 宜昌人福药业有限责任公司 一种舒芬太尼透皮贴剂及其制备方法

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US5186939A (en) * 1987-04-23 1993-02-16 Cygnus Therapeutic Systems Laminated composite for transdermal administration of fentanyl
RU2255744C1 (ru) * 2004-10-08 2005-07-10 Субботина Ольга Александровна Способ и набор для лечения воспалительных и аллергических заболеваний

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Also Published As

Publication number Publication date
JP2021038269A (ja) 2021-03-11
AU2018202501B2 (en) 2019-11-14
EP2207507A4 (en) 2013-10-23
HK1151449A1 (en) 2012-02-03
JP5687901B2 (ja) 2015-03-25
JP6810216B2 (ja) 2021-01-06
CN101902996A (zh) 2010-12-01
JP2011500604A (ja) 2011-01-06
AU2016244227A1 (en) 2016-11-03
JP2015232027A (ja) 2015-12-24
MY162831A (en) 2017-07-31
AU2008312507A1 (en) 2009-04-23
AU2020200951A1 (en) 2020-02-27
JP6600658B2 (ja) 2019-10-30
RU2010119491A (ru) 2011-11-27
JP7003211B2 (ja) 2022-01-20
US20090258061A1 (en) 2009-10-15
JP2017125057A (ja) 2017-07-20
EP2207507A1 (en) 2010-07-21
JP5802221B2 (ja) 2015-10-28
JP2013060470A (ja) 2013-04-04
JP6169139B2 (ja) 2017-07-26
AU2018202501A1 (en) 2018-05-10
MY154027A (en) 2015-04-30
AU2016244227B2 (en) 2018-01-18
AU2020200951B2 (en) 2021-07-15
AU2008312507B2 (en) 2014-03-27
CN104398496B (zh) 2018-03-20
CN104398496A (zh) 2015-03-11
US20170105944A1 (en) 2017-04-20
NZ584190A (en) 2012-09-28
JP2019206585A (ja) 2019-12-05
US20190022026A1 (en) 2019-01-24
CN101902996B (zh) 2014-11-26
WO2009052204A1 (en) 2009-04-23
HK1208156A1 (en) 2016-02-26
MY188123A (en) 2021-11-22
KR20100080800A (ko) 2010-07-12
EP2207507B1 (en) 2018-11-21
KR101583680B1 (ko) 2016-01-08
AU2014203502B2 (en) 2016-07-14
AU2014203502A1 (en) 2014-07-17

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