RU2498984C2 - Перхаридины в качестве ингибиторов cdk - Google Patents
Перхаридины в качестве ингибиторов cdk Download PDFInfo
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- RU2498984C2 RU2498984C2 RU2010108507/04A RU2010108507A RU2498984C2 RU 2498984 C2 RU2498984 C2 RU 2498984C2 RU 2010108507/04 A RU2010108507/04 A RU 2010108507/04A RU 2010108507 A RU2010108507 A RU 2010108507A RU 2498984 C2 RU2498984 C2 RU 2498984C2
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| IBIB2007/003655 | 2007-09-12 | ||
| PCT/IB2008/003106 WO2009034475A2 (en) | 2007-09-12 | 2008-09-12 | Perharidines as cdk inhibitors |
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| WO2013059634A1 (en) | 2011-10-20 | 2013-04-25 | The Regents Of The University Of California | Use of cdk9 inhibitors to reduce cartilage degradation |
| CN105481858B (zh) * | 2014-10-11 | 2019-05-17 | 上海医药集团股份有限公司 | 一种含氮稠杂环化合物、其制备方法、组合物及应用 |
| SMT202500028T1 (it) | 2018-09-10 | 2025-03-12 | Mirati Therapeutics Inc | Terapie combinate |
| CN111217814B (zh) * | 2018-11-26 | 2022-08-26 | 天津科技大学 | 一类联哌啶衍生物及其作为抗肿瘤药物的应用 |
| US20230115907A1 (en) | 2019-12-20 | 2023-04-13 | Evopoint Biosciences Co., Ltd. | Heterocyclic compound and pharmaceutical composition, preparation method, intermediate and use thereof |
| GB202108572D0 (en) * | 2021-06-16 | 2021-07-28 | Carrick Therapeutics Ltd | Therapeutic compounds and their use |
| CN115104576A (zh) * | 2022-07-12 | 2022-09-27 | 河北医科大学 | Cdk5调控eEF2在糖尿病肾病防治中的操作方法 |
| CN118598874A (zh) * | 2024-05-21 | 2024-09-06 | 江南大学 | 一种取代的9h嘌呤类化合物、药物组合物及其用途 |
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| SU566842A1 (ru) * | 1976-01-06 | 1977-07-30 | Донецкое Отделение Физико-Органической Химии Института Физической Химии Им.Л.В.Писаржевского Ан Украинской Сср | Способ получени замещенных имидазопиридинов |
| EP1352910A1 (en) * | 2002-04-10 | 2003-10-15 | Grünenthal GmbH | New analogs of nitrobenzylthioinosine |
| UA74593C2 (en) * | 2000-12-08 | 2006-01-16 | 3M Innovative Properties Co | Substituted imidazopyridines |
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| AU7738000A (en) * | 1999-09-30 | 2001-04-30 | Neurogen Corporation | Certain alkylene diamine-substituted heterocycles |
| CA2491680C (en) * | 2002-07-02 | 2012-04-17 | Southern Research Institute | Inhibitors of ftsz and uses thereof |
| CA2576159A1 (en) * | 2004-08-27 | 2006-03-02 | Cyclacel Limited | Purine and pyrimidine cdk inhibitors and their use for the treatment of autoimmune diseases |
| TW200616624A (en) * | 2004-09-09 | 2006-06-01 | Solvay Pharm Bv | 2-substituted-1-deaza purine derivatives with adenosine receptor modulating activity |
| EP1824850A2 (en) * | 2004-12-09 | 2007-08-29 | Nycomed GmbH | SUBSTITUTED IMIDAZO[4,5-b]PYRIDINES AS INHIBITORS OF GASTRIC ACID SECRETION |
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2007
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2008
- 2008-09-12 KR KR1020107007885A patent/KR20100075907A/ko not_active Withdrawn
- 2008-09-12 RU RU2010108507/04A patent/RU2498984C2/ru not_active IP Right Cessation
- 2008-09-12 JP JP2010524600A patent/JP2010539155A/ja active Pending
- 2008-09-12 EP EP08831015A patent/EP2185557A2/en not_active Withdrawn
- 2008-09-12 CA CA2699040A patent/CA2699040A1/en not_active Abandoned
- 2008-09-12 WO PCT/IB2008/003106 patent/WO2009034475A2/en not_active Ceased
- 2008-09-12 BR BRPI0816799-0A2A patent/BRPI0816799A2/pt not_active IP Right Cessation
- 2008-09-12 CN CN200880106879A patent/CN101809020A/zh active Pending
- 2008-09-12 MX MX2010002477A patent/MX2010002477A/es active IP Right Grant
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Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SU566842A1 (ru) * | 1976-01-06 | 1977-07-30 | Донецкое Отделение Физико-Органической Химии Института Физической Химии Им.Л.В.Писаржевского Ан Украинской Сср | Способ получени замещенных имидазопиридинов |
| UA74593C2 (en) * | 2000-12-08 | 2006-01-16 | 3M Innovative Properties Co | Substituted imidazopyridines |
| EP1352910A1 (en) * | 2002-04-10 | 2003-10-15 | Grünenthal GmbH | New analogs of nitrobenzylthioinosine |
Also Published As
| Publication number | Publication date |
|---|---|
| KR20100075907A (ko) | 2010-07-05 |
| CN101809020A (zh) | 2010-08-18 |
| WO2009034411A1 (en) | 2009-03-19 |
| EP2185557A2 (en) | 2010-05-19 |
| US20100280065A1 (en) | 2010-11-04 |
| RU2010108507A (ru) | 2011-10-20 |
| CA2699040A1 (en) | 2009-03-19 |
| WO2009034475A3 (en) | 2009-08-13 |
| WO2009034475A2 (en) | 2009-03-19 |
| BRPI0816799A2 (pt) | 2015-03-03 |
| MX2010002477A (es) | 2010-08-09 |
| US8450342B2 (en) | 2013-05-28 |
| JP2010539155A (ja) | 2010-12-16 |
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