RU2368608C2 - Производные пиперидина в качестве модуляторов хемокинового рецептора ccr5 - Google Patents

Производные пиперидина в качестве модуляторов хемокинового рецептора ccr5 Download PDF

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RU2368608C2
RU2368608C2 RU2006138663/04A RU2006138663A RU2368608C2 RU 2368608 C2 RU2368608 C2 RU 2368608C2 RU 2006138663/04 A RU2006138663/04 A RU 2006138663/04A RU 2006138663 A RU2006138663 A RU 2006138663A RU 2368608 C2 RU2368608 C2 RU 2368608C2
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Алан ФАУЛЛ (GB)
Алан ФАУЛЛ
Хауард ТАКЕР (GB)
Хауард ТАКЕР
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Астразенека Аб
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Priority claimed from SE0401057A external-priority patent/SE0401057D0/xx
Priority claimed from SE0500057A external-priority patent/SE0500057D0/sv
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
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  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
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  • Immunology (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
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  • Dermatology (AREA)
  • Endocrinology (AREA)
  • Virology (AREA)
  • Biomedical Technology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Rheumatology (AREA)
  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
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  • Psychiatry (AREA)
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RU2006138663/04A 2004-04-23 2005-04-20 Производные пиперидина в качестве модуляторов хемокинового рецептора ccr5 RU2368608C2 (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
SE0401057A SE0401057D0 (sv) 2004-04-23 2004-04-23 Chemical Compounds
SE0401057-5 2004-04-23
SE0500057A SE0500057D0 (sv) 2005-01-10 2005-01-10 Chemical compounds
SE0500057-5 2005-01-10

Publications (2)

Publication Number Publication Date
RU2006138663A RU2006138663A (ru) 2008-05-27
RU2368608C2 true RU2368608C2 (ru) 2009-09-27

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RU2006138663/04A RU2368608C2 (ru) 2004-04-23 2005-04-20 Производные пиперидина в качестве модуляторов хемокинового рецептора ccr5

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US (2) US7615555B2 (enExample)
EP (1) EP1742934A2 (enExample)
JP (1) JP2007533735A (enExample)
KR (1) KR20070007345A (enExample)
AR (1) AR048834A1 (enExample)
AU (1) AU2005235169B2 (enExample)
BR (1) BRPI0510126A (enExample)
CA (1) CA2562417A1 (enExample)
IL (1) IL178650A0 (enExample)
MX (1) MXPA06012045A (enExample)
NO (1) NO20065319L (enExample)
RU (1) RU2368608C2 (enExample)
SA (1) SA05260099B1 (enExample)
TW (1) TW200610761A (enExample)
UY (1) UY28870A1 (enExample)
WO (1) WO2005101989A2 (enExample)

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TW200831093A (en) * 2006-12-11 2008-08-01 Astrazeneca Ab Chemical compound
TW200831483A (en) * 2006-12-11 2008-08-01 Astrazeneca Ab Chemical compound
EP2112880A4 (en) * 2006-12-14 2011-12-21 Merck Sharp & Dohme ACYLBIPIPERIDINYL COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND TREATMENT METHOD
ES2536404T3 (es) * 2007-02-23 2015-05-25 K.H.S. Pharma Holding Gmbh Procedimiento para la preparación de ésteres de azoniaspironortropina
US7977358B2 (en) 2007-07-26 2011-07-12 Hoffmann-La Roche Inc. Pyrazol derivatives
RS52712B (sr) 2008-04-11 2013-08-30 Janssen Pharmaceutica N.V. Tiazolopiridin-2-iloksi-fenil i tiazolopirazin-2-iloksi-fenil amini kao modulatori leukotrien a4 hidrolaze
US8217060B2 (en) 2009-05-15 2012-07-10 Janssen Pharmaceutica, Nv Benzimidazole derivatives useful as TRP M8 receptor modulators
ES2564457T3 (es) 2009-07-24 2016-03-22 Glaxosmithkline Llc Derivados de azabiciclo[3,2,1]octilo para su uso en el tratamiento de VIH
CN102241664B (zh) * 2010-05-13 2014-11-12 上海医药工业研究院 芳烷二胺类衍生物及其作为抗抑郁症药物的应用
BR112012029395A2 (pt) 2010-05-17 2016-07-26 Array Biopharma Inc lactamas piperdinil-substituídas como moduladores de gpr119
WO2013074641A1 (en) * 2011-11-16 2013-05-23 Array Biopharma Inc. Piperidinyl- substituted cyclic ureas as gpr119 modulators
JP6303250B2 (ja) 2012-12-21 2018-04-04 石原産業株式会社 有害生物防除剤
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