RU2286341C2 - Фармацевтические соли ребоксетина - Google Patents
Фармацевтические соли ребоксетина Download PDFInfo
- Publication number
- RU2286341C2 RU2286341C2 RU2005100846/04A RU2005100846A RU2286341C2 RU 2286341 C2 RU2286341 C2 RU 2286341C2 RU 2005100846/04 A RU2005100846/04 A RU 2005100846/04A RU 2005100846 A RU2005100846 A RU 2005100846A RU 2286341 C2 RU2286341 C2 RU 2286341C2
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- RU
- Russia
- Prior art keywords
- salt
- reboxetine
- fumarate
- succinate
- morpholine
- Prior art date
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- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
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- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
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- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
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- Engineering & Computer Science (AREA)
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|---|---|---|---|
| EP02077366.9 | 2002-06-17 | ||
| EP02077366 | 2002-06-17 |
Publications (2)
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| RU2005100846A RU2005100846A (ru) | 2005-06-10 |
| RU2286341C2 true RU2286341C2 (ru) | 2006-10-27 |
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| RU2005100846/04A RU2286341C2 (ru) | 2002-06-17 | 2003-06-04 | Фармацевтические соли ребоксетина |
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| US (2) | US20070010517A1 (https=) |
| EP (1) | EP1515959B1 (https=) |
| JP (1) | JP4563172B2 (https=) |
| KR (1) | KR100779786B1 (https=) |
| CN (2) | CN1662511B (https=) |
| AR (1) | AR040222A1 (https=) |
| AT (1) | ATE439354T1 (https=) |
| AU (1) | AU2003227755B2 (https=) |
| BR (1) | BR0311878A (https=) |
| CA (1) | CA2489763C (https=) |
| DE (1) | DE60328787D1 (https=) |
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| PE (1) | PE20040565A1 (https=) |
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| GB0319793D0 (en) | 2003-08-22 | 2003-09-24 | Lilly Co Eli | Pyridinylmorpholine derivatives |
| WO2005082869A1 (en) * | 2004-02-20 | 2005-09-09 | Pharmacia & Upjohn Company Llc | Method for the preparation of aryl ethers |
| US8580776B2 (en) * | 2007-07-10 | 2013-11-12 | The Board Of Trustees Of The University Of Illinois | Compositions and methods for treating neurodegenerating diseases |
| US20100069389A1 (en) * | 2008-09-06 | 2010-03-18 | Bionevia Pharmaceuticals, Inc. | Novel forms of reboxetine |
| US20190185438A1 (en) * | 2016-12-06 | 2019-06-20 | Tonix Pharmaceuticals Holding Corp. | Salts and polymorphs of esreboxetine |
| US12565478B1 (en) | 2025-01-21 | 2026-03-03 | Axsome Therapeutics, Inc. | (S)-2-((S)-(2-ethoxyphenoxy)(phenyl)methyl)-4-nitrosomorpholine |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2167407A (en) * | 1984-11-22 | 1986-05-29 | Erba Farmitalia | Enantiomers of phenoxy derivatives of benzyl morpholine and salts thereof |
| WO2001001973A2 (en) * | 1999-07-01 | 2001-01-11 | Pharmacia & Upjohn Company | Highly selective norepinephrine reuptake inhibitors and methods of using the same |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU9214498A (en) * | 1997-09-23 | 1999-04-12 | Eli Lilly And Company | Treatment of attention-deficit/hyperactivity disorder |
| UA57107C2 (uk) * | 1997-09-23 | 2003-06-16 | Елі Ліллі Енд Компані | Спосіб лікування розладу поведінки |
| UA56257C2 (uk) * | 1997-09-23 | 2003-05-15 | Елі Ліллі Енд Компані | Спосіб лікування неадекватної визивної поведінки |
| IT1305322B1 (it) * | 1998-04-23 | 2001-05-04 | Pharmacia & Upjohn Spa | Uso di reboxetina per il trattamento di disturbi nervosi |
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- 2003-06-04 RU RU2005100846/04A patent/RU2286341C2/ru not_active IP Right Cessation
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- 2003-06-04 CN CNA200810093308XA patent/CN101298440A/zh active Pending
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- 2003-06-04 NZ NZ537023A patent/NZ537023A/en unknown
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- 2003-06-04 KR KR1020047020412A patent/KR100779786B1/ko not_active Expired - Fee Related
- 2003-06-04 EP EP03725195A patent/EP1515959B1/en not_active Expired - Lifetime
- 2003-06-04 US US10/588,808 patent/US20070010517A1/en not_active Abandoned
- 2003-06-04 BR BR0311878-9A patent/BR0311878A/pt not_active IP Right Cessation
- 2003-06-04 JP JP2004513273A patent/JP4563172B2/ja not_active Expired - Fee Related
- 2003-06-11 TW TW092115889A patent/TWI267510B/zh not_active IP Right Cessation
- 2003-06-11 MY MYPI20032183A patent/MY131231A/en unknown
- 2003-06-13 AR ARP030102115A patent/AR040222A1/es unknown
- 2003-06-17 PE PE2003000594A patent/PE20040565A1/es not_active Application Discontinuation
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2004
- 2004-11-29 ZA ZA200409624A patent/ZA200409624B/xx unknown
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2005
- 2005-01-12 NO NO20050183A patent/NO329346B1/no not_active IP Right Cessation
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2009
- 2009-05-21 US US12/469,780 patent/US20090291953A1/en not_active Abandoned
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2167407A (en) * | 1984-11-22 | 1986-05-29 | Erba Farmitalia | Enantiomers of phenoxy derivatives of benzyl morpholine and salts thereof |
| WO2001001973A2 (en) * | 1999-07-01 | 2001-01-11 | Pharmacia & Upjohn Company | Highly selective norepinephrine reuptake inhibitors and methods of using the same |
Non-Patent Citations (1)
| Title |
|---|
| MELLONI P. et al. ″Configurational studies on 2-[α-(2-ethoxyphenoxy)benzyl] morpholine FCE 20124″, Tetrahedron, v.41, n.7, pp.13931399, 1985. * |
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