RU2282447C2 - Никотинсодержащая фармацевтическая композиция и ее применение - Google Patents
Никотинсодержащая фармацевтическая композиция и ее применение Download PDFInfo
- Publication number
- RU2282447C2 RU2282447C2 RU2004108853/15A RU2004108853A RU2282447C2 RU 2282447 C2 RU2282447 C2 RU 2282447C2 RU 2004108853/15 A RU2004108853/15 A RU 2004108853/15A RU 2004108853 A RU2004108853 A RU 2004108853A RU 2282447 C2 RU2282447 C2 RU 2282447C2
- Authority
- RU
- Russia
- Prior art keywords
- nicotine
- smoking
- composition according
- cessation
- pharmaceutical composition
- Prior art date
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- SNICXCGAKADSCV-JTQLQIEISA-N (-)-Nicotine Chemical compound CN1CCC[C@H]1C1=CC=CN=C1 SNICXCGAKADSCV-JTQLQIEISA-N 0.000 title claims abstract description 86
- 229960002715 nicotine Drugs 0.000 title claims abstract description 86
- SNICXCGAKADSCV-UHFFFAOYSA-N nicotine Natural products CN1CCCC1C1=CC=CN=C1 SNICXCGAKADSCV-UHFFFAOYSA-N 0.000 title claims abstract description 86
- 239000008194 pharmaceutical composition Substances 0.000 title claims abstract 9
- 235000019219 chocolate Nutrition 0.000 claims abstract description 34
- 239000000203 mixture Substances 0.000 claims abstract description 34
- 230000000391 smoking effect Effects 0.000 claims abstract description 19
- 238000002560 therapeutic procedure Methods 0.000 claims abstract description 4
- 244000299461 Theobroma cacao Species 0.000 claims description 39
- 238000002670 nicotine replacement therapy Methods 0.000 claims description 15
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- 235000013355 food flavoring agent Nutrition 0.000 claims description 7
- 229910000029 sodium carbonate Inorganic materials 0.000 claims description 7
- 241000208125 Nicotiana Species 0.000 claims description 6
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- BVKZGUZCCUSVTD-UHFFFAOYSA-M Bicarbonate Chemical class OC([O-])=O BVKZGUZCCUSVTD-UHFFFAOYSA-M 0.000 claims description 2
- OCUCCJIRFHNWBP-IYEMJOQQSA-L Copper gluconate Chemical class [Cu+2].OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)C([O-])=O.OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)C([O-])=O OCUCCJIRFHNWBP-IYEMJOQQSA-L 0.000 claims description 2
- DGAQECJNVWCQMB-PUAWFVPOSA-M Ilexoside XXIX Chemical compound C[C@@H]1CC[C@@]2(CC[C@@]3(C(=CC[C@H]4[C@]3(CC[C@@H]5[C@@]4(CC[C@@H](C5(C)C)OS(=O)(=O)[O-])C)C)[C@@H]2[C@]1(C)O)C)C(=O)O[C@H]6[C@@H]([C@H]([C@@H]([C@H](O6)CO)O)O)O.[Na+] DGAQECJNVWCQMB-PUAWFVPOSA-M 0.000 claims description 2
- ZLMJMSJWJFRBEC-UHFFFAOYSA-N Potassium Chemical compound [K] ZLMJMSJWJFRBEC-UHFFFAOYSA-N 0.000 claims description 2
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- IPQVTOJGNYVQEO-UHFFFAOYSA-N 9-[2-carboxy-4-hydroxy-10-oxo-5-[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-9h-anthracen-9-yl]-4-hydroxy-10-oxo-5-[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-9h-anthracene-2-carboxylic acid Chemical class OC1C(O)C(O)C(CO)OC1OC1=CC=CC2=C1C(=O)C1=C(O)C=C(C(O)=O)C=C1C2C1C2=CC(C(O)=O)=CC(O)=C2C(=O)C2=C(OC3C(C(O)C(O)C(CO)O3)O)C=CC=C21 IPQVTOJGNYVQEO-UHFFFAOYSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23G—COCOA; COCOA PRODUCTS, e.g. CHOCOLATE; SUBSTITUTES FOR COCOA OR COCOA PRODUCTS; CONFECTIONERY; CHEWING GUM; ICE-CREAM; PREPARATION THEREOF
- A23G1/00—Cocoa; Cocoa products, e.g. chocolate; Substitutes therefor
- A23G1/30—Cocoa products, e.g. chocolate; Substitutes therefor
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23G—COCOA; COCOA PRODUCTS, e.g. CHOCOLATE; SUBSTITUTES FOR COCOA OR COCOA PRODUCTS; CONFECTIONERY; CHEWING GUM; ICE-CREAM; PREPARATION THEREOF
- A23G1/00—Cocoa; Cocoa products, e.g. chocolate; Substitutes therefor
- A23G1/30—Cocoa products, e.g. chocolate; Substitutes therefor
- A23G1/32—Cocoa products, e.g. chocolate; Substitutes therefor characterised by the composition containing organic or inorganic compounds
- A23G1/42—Cocoa products, e.g. chocolate; Substitutes therefor characterised by the composition containing organic or inorganic compounds containing microorganisms or enzymes; containing paramedical or dietetical agents, e.g. vitamins
- A23G1/426—Cocoa products, e.g. chocolate; Substitutes therefor characterised by the composition containing organic or inorganic compounds containing microorganisms or enzymes; containing paramedical or dietetical agents, e.g. vitamins containing vitamins or antibiotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/465—Nicotine; Derivatives thereof
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2068—Compounds of unknown constitution, e.g. material from plants or animals
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Organic Chemistry (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Food Science & Technology (AREA)
- Psychology (AREA)
- Polymers & Plastics (AREA)
- Nutrition Science (AREA)
- Child & Adolescent Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Microbiology (AREA)
- Obesity (AREA)
- Inorganic Chemistry (AREA)
- Zoology (AREA)
- Physiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0103210-1 | 2001-09-27 | ||
| SE0103210A SE0103210D0 (sv) | 2001-09-27 | 2001-09-27 | New formulations and use thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU2004108853A RU2004108853A (ru) | 2005-04-20 |
| RU2282447C2 true RU2282447C2 (ru) | 2006-08-27 |
Family
ID=20285456
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2004108853/15A RU2282447C2 (ru) | 2001-09-27 | 2002-09-10 | Никотинсодержащая фармацевтическая композиция и ее применение |
Country Status (19)
| Country | Link |
|---|---|
| EP (1) | EP1429770B1 (enExample) |
| JP (1) | JP4262094B2 (enExample) |
| KR (1) | KR20040047868A (enExample) |
| CN (1) | CN1561213A (enExample) |
| AR (1) | AR036679A1 (enExample) |
| AT (1) | ATE431144T1 (enExample) |
| AU (1) | AU2002334523B2 (enExample) |
| BR (1) | BR0212834A (enExample) |
| CA (1) | CA2461757C (enExample) |
| DE (1) | DE60232344D1 (enExample) |
| DK (1) | DK1429770T3 (enExample) |
| ES (1) | ES2325684T3 (enExample) |
| IL (1) | IL160886A0 (enExample) |
| MX (1) | MXPA04002876A (enExample) |
| NZ (1) | NZ532528A (enExample) |
| RU (1) | RU2282447C2 (enExample) |
| SE (1) | SE0103210D0 (enExample) |
| WO (1) | WO2003026656A1 (enExample) |
| ZA (1) | ZA200402091B (enExample) |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2320674C1 (ru) * | 2006-07-12 | 2008-03-27 | Каш Тенгис | Способ получения сополимера n-винилпирролидона с лаурилметакрилатом для трансдермального введения никотина, сополимер, полученный этим способом, гель для трансдермального введения никотина |
| RU2448573C1 (ru) * | 2010-12-27 | 2012-04-27 | Олег Иванович Квасенков | Способ получения некурительного изделия из махорки |
| EA019621B1 (ru) * | 2010-12-27 | 2014-05-30 | Федеральное Государственное Автономное Образовательное Учреждение Высшего Профессионального Образования "Сибирский Федеральный Университет" (Сфу) | Устройство для бестраншейной замены трубопроводов |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7767698B2 (en) | 2002-06-03 | 2010-08-03 | Mcneil Ab | Formulation and use thereof |
| BRPI0415741B1 (pt) | 2003-11-07 | 2013-07-23 | composições de tabaco e métodos de fabricação de uma composição de tabaco | |
| US8627828B2 (en) | 2003-11-07 | 2014-01-14 | U.S. Smokeless Tobacco Company Llc | Tobacco compositions |
| CZ301596B6 (cs) * | 2009-02-11 | 2010-04-28 | Heglund A.S. | Kompozice urcená k bukální absorpci nikotinu za úcelem odvykání kourení |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2147501A (en) * | 1983-10-03 | 1985-05-15 | Avner Rotman | Encapsulated medicament in sweet matrix |
| US5662920A (en) * | 1993-07-26 | 1997-09-02 | Pharmacia Ab | Nicotine lozenge and therapeutic method for smoking cessation |
| WO2000030641A1 (en) * | 1998-11-23 | 2000-06-02 | Pharmacia & Upjohn Ab | Nicotine-containing pharmaceutical compositions giving a rapid transmucosal absorption |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0103211D0 (sv) * | 2001-09-27 | 2001-09-27 | Pharmacia Ab | New formulations and use thereof |
-
2001
- 2001-09-27 SE SE0103210A patent/SE0103210D0/xx unknown
-
2002
- 2002-09-10 AT AT02799531T patent/ATE431144T1/de not_active IP Right Cessation
- 2002-09-10 RU RU2004108853/15A patent/RU2282447C2/ru not_active IP Right Cessation
- 2002-09-10 CA CA002461757A patent/CA2461757C/en not_active Expired - Lifetime
- 2002-09-10 IL IL16088602A patent/IL160886A0/xx unknown
- 2002-09-10 MX MXPA04002876A patent/MXPA04002876A/es active IP Right Grant
- 2002-09-10 NZ NZ532528A patent/NZ532528A/en not_active IP Right Cessation
- 2002-09-10 KR KR10-2004-7004483A patent/KR20040047868A/ko not_active Ceased
- 2002-09-10 JP JP2003530292A patent/JP4262094B2/ja not_active Expired - Fee Related
- 2002-09-10 AU AU2002334523A patent/AU2002334523B2/en not_active Ceased
- 2002-09-10 DK DK02799531T patent/DK1429770T3/da active
- 2002-09-10 CN CNA028190386A patent/CN1561213A/zh active Pending
- 2002-09-10 WO PCT/SE2002/001612 patent/WO2003026656A1/en not_active Ceased
- 2002-09-10 BR BR0212834-9A patent/BR0212834A/pt not_active IP Right Cessation
- 2002-09-10 DE DE60232344T patent/DE60232344D1/de not_active Expired - Lifetime
- 2002-09-10 ES ES02799531T patent/ES2325684T3/es not_active Expired - Lifetime
- 2002-09-10 EP EP02799531A patent/EP1429770B1/en not_active Expired - Lifetime
- 2002-09-26 AR ARP020103631A patent/AR036679A1/es unknown
-
2004
- 2004-03-16 ZA ZA2004/02091A patent/ZA200402091B/en unknown
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2147501A (en) * | 1983-10-03 | 1985-05-15 | Avner Rotman | Encapsulated medicament in sweet matrix |
| US5662920A (en) * | 1993-07-26 | 1997-09-02 | Pharmacia Ab | Nicotine lozenge and therapeutic method for smoking cessation |
| RU2153338C2 (ru) * | 1993-07-26 | 2000-07-27 | Фармасиа Энд Апджон Аб | Никотинсодержащая таблетка и способ лечения от курения |
| WO2000030641A1 (en) * | 1998-11-23 | 2000-06-02 | Pharmacia & Upjohn Ab | Nicotine-containing pharmaceutical compositions giving a rapid transmucosal absorption |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2320674C1 (ru) * | 2006-07-12 | 2008-03-27 | Каш Тенгис | Способ получения сополимера n-винилпирролидона с лаурилметакрилатом для трансдермального введения никотина, сополимер, полученный этим способом, гель для трансдермального введения никотина |
| RU2448573C1 (ru) * | 2010-12-27 | 2012-04-27 | Олег Иванович Квасенков | Способ получения некурительного изделия из махорки |
| EA019621B1 (ru) * | 2010-12-27 | 2014-05-30 | Федеральное Государственное Автономное Образовательное Учреждение Высшего Профессионального Образования "Сибирский Федеральный Университет" (Сфу) | Устройство для бестраншейной замены трубопроводов |
Also Published As
| Publication number | Publication date |
|---|---|
| ATE431144T1 (de) | 2009-05-15 |
| MXPA04002876A (es) | 2005-06-20 |
| WO2003026656A1 (en) | 2003-04-03 |
| EP1429770B1 (en) | 2009-05-13 |
| IL160886A0 (en) | 2004-08-31 |
| CA2461757C (en) | 2008-09-02 |
| ES2325684T3 (es) | 2009-09-14 |
| BR0212834A (pt) | 2004-10-13 |
| JP2005503429A (ja) | 2005-02-03 |
| DK1429770T3 (da) | 2009-08-03 |
| EP1429770A1 (en) | 2004-06-23 |
| AR036679A1 (es) | 2004-09-29 |
| CN1561213A (zh) | 2005-01-05 |
| DE60232344D1 (de) | 2009-06-25 |
| KR20040047868A (ko) | 2004-06-05 |
| NZ532528A (en) | 2005-10-28 |
| ZA200402091B (en) | 2005-06-29 |
| SE0103210D0 (sv) | 2001-09-27 |
| CA2461757A1 (en) | 2003-04-03 |
| AU2002334523B2 (en) | 2007-02-15 |
| JP4262094B2 (ja) | 2009-05-13 |
| RU2004108853A (ru) | 2005-04-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM4A | The patent is invalid due to non-payment of fees |
Effective date: 20160911 |