RU2190613C2 - Аналоги камптотецина, способы их получения и фармацевтическая композиция на их основе - Google Patents

Аналоги камптотецина, способы их получения и фармацевтическая композиция на их основе Download PDF

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Publication number
RU2190613C2
RU2190613C2 RU99115884/04A RU99115884A RU2190613C2 RU 2190613 C2 RU2190613 C2 RU 2190613C2 RU 99115884/04 A RU99115884/04 A RU 99115884/04A RU 99115884 A RU99115884 A RU 99115884A RU 2190613 C2 RU2190613 C2 RU 2190613C2
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RU
Russia
Prior art keywords
compound
ethyl
lower alkyl
formula
hydroxy
Prior art date
Application number
RU99115884/04A
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English (en)
Russian (ru)
Other versions
RU99115884A (ru
Inventor
Дени Бигг
Оливье ЛАВЕРНЬ
Джерри ХАРНЕТТ
Алан РОЛЛАН
Анн-Мари Либератор
Кристоф ЛАНКО
Original Assignee
Сосьете Де Консей Де Решерш Э Д`Аппликасьон Сьентифик (С.К.Р.А.С.)
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Publication of RU99115884A publication Critical patent/RU99115884A/ru
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
RU99115884/04A 1996-12-20 1997-12-05 Аналоги камптотецина, способы их получения и фармацевтическая композиция на их основе RU2190613C2 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9615775A FR2757515B1 (fr) 1996-12-20 1996-12-20 Formes prodrogues et nouveaux analogues de la camptothecine, leurs procedes de preparation, leur application comme medicaments et les compositions pharmaceutiques les contenant
FR96/15945 1996-12-24
FR96/15775 1996-12-24

Publications (2)

Publication Number Publication Date
RU99115884A RU99115884A (ru) 2001-05-27
RU2190613C2 true RU2190613C2 (ru) 2002-10-10

Family

ID=9498939

Family Applications (1)

Application Number Title Priority Date Filing Date
RU99115884/04A RU2190613C2 (ru) 1996-12-20 1997-12-05 Аналоги камптотецина, способы их получения и фармацевтическая композиция на их основе

Country Status (3)

Country Link
FR (1) FR2757515B1 (fr)
RU (1) RU2190613C2 (fr)
ZA (1) ZA9711270B (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2450008C2 (ru) * 2006-07-26 2012-05-10 Индена С.П.А. Производные камптотецина с противоопухолевой активностью

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2790261B1 (fr) * 1999-02-26 2004-09-10 Sod Conseils Rech Applic Nouveaux analogues optiquement purs de la camptothecine et leurs procedes de preparation

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT835258E (pt) * 1995-06-21 2003-02-28 Sod Conseils Rech Applic Novos analogos de camptotecina, processos para a sua preparacao, sua utilizacao como farmacos e composicoes farmaceuticas que os contem

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2450008C2 (ru) * 2006-07-26 2012-05-10 Индена С.П.А. Производные камптотецина с противоопухолевой активностью

Also Published As

Publication number Publication date
FR2757515B1 (fr) 2000-05-05
FR2757515A1 (fr) 1998-06-26
ZA9711270B (en) 1998-06-23

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PD4A Correction of name of patent owner
MM4A The patent is invalid due to non-payment of fees

Effective date: 20111206