RS63671B1 - Supstitutisani derivati triazolo hinoksalina - Google Patents

Supstitutisani derivati triazolo hinoksalina

Info

Publication number
RS63671B1
RS63671B1 RS20220977A RSP20220977A RS63671B1 RS 63671 B1 RS63671 B1 RS 63671B1 RS 20220977 A RS20220977 A RS 20220977A RS P20220977 A RSP20220977 A RS P20220977A RS 63671 B1 RS63671 B1 RS 63671B1
Authority
RS
Serbia
Prior art keywords
quinoxaline derivatives
substituted triazolo
triazolo quinoxaline
substituted
derivatives
Prior art date
Application number
RS20220977A
Other languages
English (en)
Inventor
Florian Jakob
Jo Alen
Simon Lucas
Tobias Craan
Ingo Konetzki
Achim Kless
Stefan Schunk
Paul Ratcliffe
Sebastian Wachten
Simon Cruwys
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of RS63671B1 publication Critical patent/RS63671B1/sr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
RS20220977A 2018-07-20 2019-07-22 Supstitutisani derivati triazolo hinoksalina RS63671B1 (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP18184613 2018-07-20
PCT/EP2019/069611 WO2020016453A1 (en) 2018-07-20 2019-07-22 Substituted triazolo quinoxaline derivatives
EP19742596.0A EP3823971B1 (en) 2018-07-20 2019-07-22 Substituted triazolo quinoxaline derivatives

Publications (1)

Publication Number Publication Date
RS63671B1 true RS63671B1 (sr) 2022-11-30

Family

ID=63014350

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20220977A RS63671B1 (sr) 2018-07-20 2019-07-22 Supstitutisani derivati triazolo hinoksalina

Country Status (20)

Country Link
US (1) US20210139488A1 (sr)
EP (1) EP3823971B1 (sr)
JP (1) JP7336506B2 (sr)
CN (1) CN112673009B (sr)
AU (1) AU2019304532A1 (sr)
BR (1) BR112021000950A2 (sr)
CA (1) CA3106752A1 (sr)
DK (1) DK3823971T3 (sr)
EA (1) EA202190271A1 (sr)
ES (1) ES2929206T3 (sr)
HR (1) HRP20221020T1 (sr)
HU (1) HUE059430T2 (sr)
IL (1) IL280212B2 (sr)
LT (1) LT3823971T (sr)
MX (1) MX2021000762A (sr)
PL (1) PL3823971T3 (sr)
PT (1) PT3823971T (sr)
RS (1) RS63671B1 (sr)
SI (1) SI3823971T1 (sr)
WO (1) WO2020016453A1 (sr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI811400B (zh) * 2018-07-20 2023-08-11 德商歌林達有限公司 經進一步取代之三唑并喹噁啉衍生物
WO2021144440A1 (en) * 2020-01-17 2021-07-22 Grünenthal GmbH Quinoxaline derivatives as modulators of the glucocorticoid receptor
EP4090660B1 (en) * 2020-01-17 2024-01-31 Grünenthal GmbH Quinoxaline derivatives
CN115124471B (zh) * 2021-03-24 2024-02-13 中国工程物理研究院化工材料研究所 一类具有高能和低熔点特性的吡唑环类炸药及其合成方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1994026746A1 (en) * 1993-05-06 1994-11-24 Novo Nordisk A/S [1,2,4]TRIAZOLO[4,3-a]QUINOXALINE COMPOUNDS, THEIR PREPARATION AND USE
JP2006521343A (ja) * 2003-03-27 2006-09-21 ファイザー・プロダクツ・インク 置換4−アミノ[1,2,4]トリアゾロ[4,3−a]キノキサリン
DE602004023926D1 (de) * 2003-04-23 2009-12-17 Merck & Co Inc Selektive spirocyclische glucocorticoid-rezeptor-modulatoren
CN101018552A (zh) * 2004-07-14 2007-08-15 利亘制药公司 细胞内受体调节剂化合物和方法
TWI410422B (zh) * 2007-01-15 2013-10-01 Mitsubishi Tanabe Pharma Corp 縮合四氫喹啉衍生物及其醫藥用途
PL2151436T3 (pl) * 2007-05-29 2013-09-30 Santen Pharmaceutical Co Ltd Nowe pochodne 1,2,3,4-tetrahydrochinoksaliny, które jako podstawnik zawierają grupę fenylową z wprowadzoną strukturą estru kwasu sulfonowego lub amidu kwasu sulfonowego i które mają aktywność wiążącą wobec receptora glukokortykoidowego
JP2009046435A (ja) * 2007-08-21 2009-03-05 Mitsubishi Tanabe Pharma Corp グルココルチコイド受容体モジュレーター
JP2009084273A (ja) * 2007-09-13 2009-04-23 Santen Pharmaceut Co Ltd 1,3,3−トリメチル−7−フェニル−3,4−ジヒドロ−1h−キノキサリン−2−オン誘導体からなるグルココルチコイド受容体アゴニスト
WO2009103007A2 (en) * 2008-02-13 2009-08-20 Ligand Pharmaceuticals Incorporated Steroid hormone receptor modulator compounds and methods
KR20180043329A (ko) 2015-08-25 2018-04-27 산텐 세이야꾸 가부시키가이샤 [4-(1,3,3-트리메틸-2-옥소-3,4-디히드로-1h-퀴녹살린-7-일)페녹시]에틸옥시 화합물 또는 그의 염
TWI811400B (zh) * 2018-07-20 2023-08-11 德商歌林達有限公司 經進一步取代之三唑并喹噁啉衍生物

Also Published As

Publication number Publication date
IL280212B2 (en) 2023-09-01
EP3823971B1 (en) 2022-07-27
WO2020016453A1 (en) 2020-01-23
AU2019304532A1 (en) 2021-03-18
LT3823971T (lt) 2022-09-12
PT3823971T (pt) 2022-10-26
CN112673009B (zh) 2023-09-19
IL280212B1 (en) 2023-05-01
EA202190271A1 (ru) 2021-06-07
EP3823971A1 (en) 2021-05-26
SI3823971T1 (sl) 2022-10-28
MX2021000762A (es) 2021-03-29
DK3823971T3 (da) 2022-09-05
IL280212A (en) 2021-03-01
CN112673009A (zh) 2021-04-16
HRP20221020T1 (hr) 2022-11-11
CA3106752A1 (en) 2020-01-23
JP7336506B2 (ja) 2023-08-31
US20210139488A1 (en) 2021-05-13
PL3823971T3 (pl) 2023-01-09
JP2021532103A (ja) 2021-11-25
ES2929206T3 (es) 2022-11-25
BR112021000950A2 (pt) 2021-04-20
HUE059430T2 (hu) 2022-11-28

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