PT3823971T - Derivados substituídos de triazolo quinoxalina - Google Patents

Derivados substituídos de triazolo quinoxalina

Info

Publication number
PT3823971T
PT3823971T PT197425960T PT19742596T PT3823971T PT 3823971 T PT3823971 T PT 3823971T PT 197425960 T PT197425960 T PT 197425960T PT 19742596 T PT19742596 T PT 19742596T PT 3823971 T PT3823971 T PT 3823971T
Authority
PT
Portugal
Prior art keywords
quinoxaline derivatives
substituted triazolo
triazolo quinoxaline
substituted
derivatives
Prior art date
Application number
PT197425960T
Other languages
English (en)
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of PT3823971T publication Critical patent/PT3823971T/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PT197425960T 2018-07-20 2019-07-22 Derivados substituídos de triazolo quinoxalina PT3823971T (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP18184613 2018-07-20

Publications (1)

Publication Number Publication Date
PT3823971T true PT3823971T (pt) 2022-10-26

Family

ID=63014350

Family Applications (1)

Application Number Title Priority Date Filing Date
PT197425960T PT3823971T (pt) 2018-07-20 2019-07-22 Derivados substituídos de triazolo quinoxalina

Country Status (20)

Country Link
US (1) US20210139488A1 (pt)
EP (1) EP3823971B1 (pt)
JP (1) JP7336506B2 (pt)
CN (1) CN112673009B (pt)
AU (1) AU2019304532A1 (pt)
BR (1) BR112021000950A2 (pt)
CA (1) CA3106752A1 (pt)
DK (1) DK3823971T3 (pt)
EA (1) EA202190271A1 (pt)
ES (1) ES2929206T3 (pt)
HR (1) HRP20221020T1 (pt)
HU (1) HUE059430T2 (pt)
IL (1) IL280212B2 (pt)
LT (1) LT3823971T (pt)
MX (1) MX2021000762A (pt)
PL (1) PL3823971T3 (pt)
PT (1) PT3823971T (pt)
RS (1) RS63671B1 (pt)
SI (1) SI3823971T1 (pt)
WO (1) WO2020016453A1 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI811400B (zh) * 2018-07-20 2023-08-11 德商歌林達有限公司 經進一步取代之三唑并喹噁啉衍生物
EP4090661A1 (en) * 2020-01-17 2022-11-23 Grünenthal GmbH Quinoxaline derivatives as modulators of the glucocorticoid receptor
EP4090660B1 (en) * 2020-01-17 2024-01-31 Grünenthal GmbH Quinoxaline derivatives
CN115124471B (zh) * 2021-03-24 2024-02-13 中国工程物理研究院化工材料研究所 一类具有高能和低熔点特性的吡唑环类炸药及其合成方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1994026746A1 (en) * 1993-05-06 1994-11-24 Novo Nordisk A/S [1,2,4]TRIAZOLO[4,3-a]QUINOXALINE COMPOUNDS, THEIR PREPARATION AND USE
MXPA05010293A (es) * 2003-03-27 2005-11-17 Pfizer Prod Inc 4-amino[1,2,4]triazolo[4,3-a]quinoxalinas sustituidas.
AU2004232301B2 (en) * 2003-04-23 2009-11-12 Merck Sharp & Dohme Corp. Selective spirocyclic glucocorticoid receptor modulators
CN101018552A (zh) * 2004-07-14 2007-08-15 利亘制药公司 细胞内受体调节剂化合物和方法
TWI410422B (zh) * 2007-01-15 2013-10-01 Mitsubishi Tanabe Pharma Corp 縮合四氫喹啉衍生物及其醫藥用途
US8193187B2 (en) * 2007-05-29 2012-06-05 Santen Pharmaceutical Co., Ltd. 1,2,3,4-tetrahydroquinoxaline compound with a phenyl group substituent having a sulfonic acid ester structure or a sulfonic acid amide structure introduced therein and having glucocorticoid receptor-binding activity
JP2009046435A (ja) * 2007-08-21 2009-03-05 Mitsubishi Tanabe Pharma Corp グルココルチコイド受容体モジュレーター
JP2009084273A (ja) * 2007-09-13 2009-04-23 Santen Pharmaceut Co Ltd 1,3,3−トリメチル−7−フェニル−3,4−ジヒドロ−1h−キノキサリン−2−オン誘導体からなるグルココルチコイド受容体アゴニスト
WO2009103007A2 (en) * 2008-02-13 2009-08-20 Ligand Pharmaceuticals Incorporated Steroid hormone receptor modulator compounds and methods
CA2996278A1 (en) * 2015-08-25 2017-03-02 Santen Pharmaceutical Co., Ltd. [4-(1,3,3-trimethyl-2-oxo-3,4-dihydro-1h-quinoxalin-7-yl)-phenoxy]ethyloxy compound or salt thereof
TWI811400B (zh) * 2018-07-20 2023-08-11 德商歌林達有限公司 經進一步取代之三唑并喹噁啉衍生物

Also Published As

Publication number Publication date
SI3823971T1 (sl) 2022-10-28
JP7336506B2 (ja) 2023-08-31
HRP20221020T1 (hr) 2022-11-11
US20210139488A1 (en) 2021-05-13
CN112673009B (zh) 2023-09-19
RS63671B1 (sr) 2022-11-30
BR112021000950A2 (pt) 2021-04-20
DK3823971T3 (da) 2022-09-05
MX2021000762A (es) 2021-03-29
EP3823971B1 (en) 2022-07-27
HUE059430T2 (hu) 2022-11-28
IL280212A (en) 2021-03-01
EP3823971A1 (en) 2021-05-26
ES2929206T3 (es) 2022-11-25
LT3823971T (lt) 2022-09-12
IL280212B1 (en) 2023-05-01
CA3106752A1 (en) 2020-01-23
CN112673009A (zh) 2021-04-16
AU2019304532A1 (en) 2021-03-18
WO2020016453A1 (en) 2020-01-23
JP2021532103A (ja) 2021-11-25
IL280212B2 (en) 2023-09-01
PL3823971T3 (pl) 2023-01-09
EA202190271A1 (ru) 2021-06-07

Similar Documents

Publication Publication Date Title
IL261885A (en) Pyrazolopyrimidine history
HK1252752A1 (zh) 新型吡唑並嘧啶衍生物
IL254870A0 (en) Quinoxaline histories are transmuted
SI3419978T1 (sl) Derivati pirazolo(1,5-A)pirazin-4-ila kot zaviralci z janusom povezane kinaze (JAK)
HK1256751A1 (zh) [1,2,4]三唑並[1,5-a]嘧啶-7-基化合物
SG11202010679SA (en) Substituted dihydropyrazolo pyrazine carboxamide derivatives
IL280211A (en) History of triazoloquinoxaline with additional transformations
IL280212B1 (en) Transmuted triazoloquinoxaline histories
IL283990A (en) Modified oxopyridine derivatives
IL279938A (en) History of spirochroman
LT3796975T (lt) Sulfonilaminobenzamido dariniai
GB201601431D0 (en) Pyrrolobenzodiazepines
PL3770162T3 (pl) Pochodne dihydrochromenu
SG11202006837XA (en) Dihydroindolizinone derivative
FI3627028T3 (fi) Putkiyhde
GB201806948D0 (en) Derivatives
ZA201902361B (en) Trailer