HUE059430T2 - Szubsztituált triazolo-kinoxalin származékok - Google Patents

Szubsztituált triazolo-kinoxalin származékok

Info

Publication number
HUE059430T2
HUE059430T2 HUE19742596A HUE19742596A HUE059430T2 HU E059430 T2 HUE059430 T2 HU E059430T2 HU E19742596 A HUE19742596 A HU E19742596A HU E19742596 A HUE19742596 A HU E19742596A HU E059430 T2 HUE059430 T2 HU E059430T2
Authority
HU
Hungary
Prior art keywords
quinoxaline derivatives
substituted triazolo
triazolo quinoxaline
substituted
derivatives
Prior art date
Application number
HUE19742596A
Other languages
English (en)
Inventor
Florian Jakob
Jo Alen
Simon Lucas
Tobias Craan
Ingo Konetzki
Achim Kless
Stefan Schunk
Paul Ratcliffe
Sebastian Wachten
Simon Cruwys
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of HUE059430T2 publication Critical patent/HUE059430T2/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
HUE19742596A 2018-07-20 2019-07-22 Szubsztituált triazolo-kinoxalin származékok HUE059430T2 (hu)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP18184613 2018-07-20

Publications (1)

Publication Number Publication Date
HUE059430T2 true HUE059430T2 (hu) 2022-11-28

Family

ID=63014350

Family Applications (1)

Application Number Title Priority Date Filing Date
HUE19742596A HUE059430T2 (hu) 2018-07-20 2019-07-22 Szubsztituált triazolo-kinoxalin származékok

Country Status (20)

Country Link
US (1) US20210139488A1 (hu)
EP (1) EP3823971B1 (hu)
JP (1) JP7336506B2 (hu)
CN (1) CN112673009B (hu)
AU (1) AU2019304532A1 (hu)
BR (1) BR112021000950A2 (hu)
CA (1) CA3106752A1 (hu)
DK (1) DK3823971T3 (hu)
EA (1) EA202190271A1 (hu)
ES (1) ES2929206T3 (hu)
HR (1) HRP20221020T1 (hu)
HU (1) HUE059430T2 (hu)
IL (1) IL280212B2 (hu)
LT (1) LT3823971T (hu)
MX (1) MX2021000762A (hu)
PL (1) PL3823971T3 (hu)
PT (1) PT3823971T (hu)
RS (1) RS63671B1 (hu)
SI (1) SI3823971T1 (hu)
WO (1) WO2020016453A1 (hu)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR117951A1 (es) * 2018-07-20 2021-09-08 Gruenenthal Gmbh Derivados de triazolquinoxalina adicionalmente sustituidos
EP4090661A1 (en) * 2020-01-17 2022-11-23 Grünenthal GmbH Quinoxaline derivatives as modulators of the glucocorticoid receptor
WO2021144439A1 (en) * 2020-01-17 2021-07-22 Grünenthal GmbH Quinoxaline derivatives
CN115124471B (zh) * 2021-03-24 2024-02-13 中国工程物理研究院化工材料研究所 一类具有高能和低熔点特性的吡唑环类炸药及其合成方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE148120T1 (de) * 1993-05-06 1997-02-15 Novo Nordisk As (1,2,4-triazolo(4,3-a>chinoxalinverbindungen deren herstellung und verwendung
MXPA05010293A (es) * 2003-03-27 2005-11-17 Pfizer Prod Inc 4-amino[1,2,4]triazolo[4,3-a]quinoxalinas sustituidas.
EP1617806B1 (en) * 2003-04-23 2009-11-04 Merck & Co., Inc. Selective spirocyclic glucocorticoid receptor modulators
WO2006019716A1 (en) * 2004-07-14 2006-02-23 Ligand Pharmaceuticals, Inc. Intracellular receptor modulator compounds and methods
TWI410422B (zh) * 2007-01-15 2013-10-01 Mitsubishi Tanabe Pharma Corp 縮合四氫喹啉衍生物及其醫藥用途
WO2008146871A1 (ja) * 2007-05-29 2008-12-04 Santen Pharmaceutical Co., Ltd. グルココルチコイド受容体結合活性を有する、スルホン酸エステル又はスルホン酸アミド構造を導入したフェニル基を置換基として有する新規1,2,3,4-テトラヒドロキノキサリン誘導体
JP2009046435A (ja) * 2007-08-21 2009-03-05 Mitsubishi Tanabe Pharma Corp グルココルチコイド受容体モジュレーター
WO2009035067A1 (ja) 2007-09-13 2009-03-19 Santen Pharmaceutical Co., Ltd. 1,3,3-トリメチル-7-フェニル-3,4-ジヒドロ-1h-キノキサリン-2-オン誘導体からなるグルココルチコイド受容体アゴニスト
WO2009103007A2 (en) * 2008-02-13 2009-08-20 Ligand Pharmaceuticals Incorporated Steroid hormone receptor modulator compounds and methods
WO2017034006A1 (ja) 2015-08-25 2017-03-02 参天製薬株式会社 [4-(1,3,3-トリメチル-2-オキソ-3,4-ジヒドロ-1h-キノキサリン-7-イル)フェノキシ]エチルオキシ化合物またはその塩
AR117951A1 (es) * 2018-07-20 2021-09-08 Gruenenthal Gmbh Derivados de triazolquinoxalina adicionalmente sustituidos

Also Published As

Publication number Publication date
JP2021532103A (ja) 2021-11-25
IL280212B2 (en) 2023-09-01
EP3823971B1 (en) 2022-07-27
ES2929206T3 (es) 2022-11-25
AU2019304532A1 (en) 2021-03-18
EP3823971A1 (en) 2021-05-26
CN112673009B (zh) 2023-09-19
CA3106752A1 (en) 2020-01-23
EA202190271A1 (ru) 2021-06-07
IL280212A (en) 2021-03-01
US20210139488A1 (en) 2021-05-13
RS63671B1 (sr) 2022-11-30
PL3823971T3 (pl) 2023-01-09
BR112021000950A2 (pt) 2021-04-20
IL280212B1 (en) 2023-05-01
JP7336506B2 (ja) 2023-08-31
WO2020016453A1 (en) 2020-01-23
MX2021000762A (es) 2021-03-29
HRP20221020T1 (hr) 2022-11-11
CN112673009A (zh) 2021-04-16
LT3823971T (lt) 2022-09-12
SI3823971T1 (sl) 2022-10-28
DK3823971T3 (da) 2022-09-05
PT3823971T (pt) 2022-10-26

Similar Documents

Publication Publication Date Title
IL261885A (en) Pyrazolopyrimidine history
HK1252752A1 (zh) 新型吡唑並嘧啶衍生物
IL254870A0 (en) Quinoxaline histories are transmuted
SI3419978T1 (sl) Derivati pirazolo(1,5-A)pirazin-4-ila kot zaviralci z janusom povezane kinaze (JAK)
HK1256751A1 (zh) [1,2,4]三唑並[1,5-a]嘧啶-7-基化合物
SG11202010679SA (en) Substituted dihydropyrazolo pyrazine carboxamide derivatives
IL280211A (en) History of triazoloquinoxaline with additional transformations
IL280212A (en) Transmuted triazoloquinoxaline histories
IL283990A (en) Modified oxopyridine derivatives
IL279938A (en) History of spirochroman
HUE064831T2 (hu) Szulfonil-amino-benzamid származékok
GB201601431D0 (en) Pyrrolobenzodiazepines
PL3770162T3 (pl) Pochodne dihydrochromenu
SG11202006837XA (en) Dihydroindolizinone derivative
FI3627028T3 (fi) Putkiyhde
GB201806948D0 (en) Derivatives
ZA201902361B (en) Trailer