RS61908B1 - Postupak za proizvodnju kondenzovanih imidazolo derivata - Google Patents

Postupak za proizvodnju kondenzovanih imidazolo derivata

Info

Publication number
RS61908B1
RS61908B1 RS20210655A RSP20210655A RS61908B1 RS 61908 B1 RS61908 B1 RS 61908B1 RS 20210655 A RS20210655 A RS 20210655A RS P20210655 A RSP20210655 A RS P20210655A RS 61908 B1 RS61908 B1 RS 61908B1
Authority
RS
Serbia
Prior art keywords
production
condensed
derivatives
imidazolo derivatives
condensed imidazolo
Prior art date
Application number
RS20210655A
Other languages
English (en)
Inventor
Andreas Bertogg
Hanspeter Schilling
Original Assignee
Recordati Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Recordati Ag filed Critical Recordati Ag
Publication of RS61908B1 publication Critical patent/RS61908B1/sr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41881,3-Diazoles condensed with other heterocyclic ring systems, e.g. biotin, sorbinil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26Androgens
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/38Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/46Drugs for disorders of the endocrine system of the suprarenal hormones for decreasing, blocking or antagonising the activity of glucocorticosteroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
RS20210655A 2015-01-29 2016-01-28 Postupak za proizvodnju kondenzovanih imidazolo derivata RS61908B1 (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562109307P 2015-01-29 2015-01-29
PCT/IB2016/050433 WO2016120821A1 (en) 2015-01-29 2016-01-28 Process for the production of condensed imidazolo derivatives
EP16702814.1A EP3250555B1 (en) 2015-01-29 2016-01-28 Process for the production of condensed imidazolo derivatives

Publications (1)

Publication Number Publication Date
RS61908B1 true RS61908B1 (sr) 2021-06-30

Family

ID=55299696

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20210655A RS61908B1 (sr) 2015-01-29 2016-01-28 Postupak za proizvodnju kondenzovanih imidazolo derivata

Country Status (21)

Country Link
US (1) US10556869B2 (sr)
EP (1) EP3250555B1 (sr)
JP (1) JP6857126B2 (sr)
KR (1) KR102559242B1 (sr)
CN (1) CN107207518B (sr)
AU (1) AU2016210899B2 (sr)
BR (1) BR112017014706A2 (sr)
CA (1) CA2973539A1 (sr)
CY (1) CY1124340T1 (sr)
DK (1) DK3250555T3 (sr)
ES (1) ES2870461T3 (sr)
HR (1) HRP20210654T1 (sr)
HU (1) HUE054248T2 (sr)
LT (1) LT3250555T (sr)
MX (1) MX2017009839A (sr)
PL (1) PL3250555T3 (sr)
PT (1) PT3250555T (sr)
RS (1) RS61908B1 (sr)
RU (1) RU2734818C2 (sr)
SI (1) SI3250555T1 (sr)
WO (1) WO2016120821A1 (sr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111592546B (zh) * 2020-05-26 2023-08-25 上海鲲博玖瑞医药科技发展有限公司 奥德司他的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4617307A (en) * 1984-06-20 1986-10-14 Ciba-Geigy Corporation Substituted imidazo[1,5-A]pyridine derivatives as aromatase inhibitors
GT200600381A (es) * 2005-08-25 2007-03-28 Compuestos organicos
BR112012017458B1 (pt) * 2010-01-14 2020-10-20 Recordati Ag Uso de di-hidrogeno fosfato de 4-[(5r)-6,7-di-hidro-5h-pirrolo[1,2-c]imidazol-5-il]-3- flurorbenzonitrila
PE20142358A1 (es) * 2012-01-17 2015-01-30 Novartis Ag Nuevas formas y sales de un dihidropirrolo[1,2-c]imidazolilo, inhibidor de la aldosterona sintasa o aromatasa

Also Published As

Publication number Publication date
US10556869B2 (en) 2020-02-11
PT3250555T (pt) 2021-04-27
EP3250555B1 (en) 2021-03-03
CN107207518A (zh) 2017-09-26
RU2017127127A3 (sr) 2019-09-23
KR102559242B1 (ko) 2023-07-25
LT3250555T (lt) 2021-06-25
SI3250555T1 (sl) 2021-08-31
HUE054248T2 (hu) 2021-08-30
HRP20210654T1 (hr) 2021-05-28
ES2870461T3 (es) 2021-10-27
CY1124340T1 (el) 2022-07-22
BR112017014706A2 (pt) 2018-02-06
EP3250555A1 (en) 2017-12-06
AU2016210899B2 (en) 2019-03-07
US20180002292A1 (en) 2018-01-04
PL3250555T3 (pl) 2021-08-02
DK3250555T3 (da) 2021-04-26
WO2016120821A1 (en) 2016-08-04
KR20170106353A (ko) 2017-09-20
CA2973539A1 (en) 2016-08-04
RU2017127127A (ru) 2019-02-28
AU2016210899A1 (en) 2017-07-20
JP6857126B2 (ja) 2021-04-14
RU2734818C2 (ru) 2020-10-23
JP2018503659A (ja) 2018-02-08
MX2017009839A (es) 2017-11-02
CN107207518B (zh) 2021-03-30

Similar Documents

Publication Publication Date Title
GB2550003B (en) Process for the production of formaldehyde-stabilised urea
ZA201706795B (en) Process for the preparation of dicycloplatin
SI3630738T1 (sl) Postopek za ustvarjanje ozanimoda
ZA201902125B (en) Process for the production of 2-alkylalkanol
IL248267A0 (en) A process for preparing converted cycloserines
SI3160985T1 (sl) Postopek za pripravo D-arginil-2,6-dimetil-L-tirosil-L-lisil-L- fenilalaninamida
PT3362405T (pt) Processo e unidade de produção para a produção de metanol
ZA201801650B (en) Process for producing novel 4-benzoazonine derivatives
PT3182981T (pt) Processo de produção de isomaltooligosacarídeos
IL257814B (en) A method for preparing praziquantel
ZA201704196B (en) Method for the production of praziquantel
GB2564185B (en) Process for the preparation of derivatives of benzodioxole
ZA201608307B (en) Process for the purification of l-alpha-glycerophosphorylcholine
PT3368513T (pt) Processo para a síntese de pirfenidona
HUE055317T2 (hu) Eljárás izoidid elõállítására
IL262889B (en) Process for the manufacture of 6-alkynyl-pyridine derivatives
IL267305A (en) Process for the manufacture of diazepine derivatives
FR3024729B1 (fr) Procede de preparation du trioxane
PT3250555T (pt) Processo para a produção de derivados de imidazolo condensado
HRP20181918T1 (hr) Postupak za sintezu derivata benzazepina
GB201717809D0 (en) Process for the production of cobimetinib
GB201414880D0 (en) Process for making phosphate derivatives