PT95112A - Processo para a preparacao de derivados de peptido farmacologicamente activos - Google Patents

Processo para a preparacao de derivados de peptido farmacologicamente activos

Info

Publication number
PT95112A
PT95112A PT95112A PT9511290A PT95112A PT 95112 A PT95112 A PT 95112A PT 95112 A PT95112 A PT 95112A PT 9511290 A PT9511290 A PT 9511290A PT 95112 A PT95112 A PT 95112A
Authority
PT
Portugal
Prior art keywords
preparation
pharmacologically active
active peptide
peptide derivatives
derivatives
Prior art date
Application number
PT95112A
Other languages
English (en)
Other versions
PT95112B (pt
Inventor
Tiberto Bruzzese
Massimo Signorini
Alberto Carlo Fanciano
Roberta Termini
Original Assignee
Prodotti Antibiotici Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Prodotti Antibiotici Spa filed Critical Prodotti Antibiotici Spa
Publication of PT95112A publication Critical patent/PT95112A/pt
Publication of PT95112B publication Critical patent/PT95112B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0802Tripeptides with the first amino acid being neutral
    • C07K5/0804Tripeptides with the first amino acid being neutral and aliphatic
    • C07K5/0806Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0802Tripeptides with the first amino acid being neutral
    • C07K5/0804Tripeptides with the first amino acid being neutral and aliphatic
    • C07K5/081Tripeptides with the first amino acid being neutral and aliphatic the side chain containing O or S as heteroatoms, e.g. Cys, Ser
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
PT95112A 1989-08-28 1990-08-28 Processo para a preparacao de derivados de peptido farmacologicamente activos PT95112B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT8921567A IT1231342B (it) 1989-08-28 1989-08-28 Derivati peptidici farmacologicamente attivi e preparazioni farmaceutiche che li contengono

Publications (2)

Publication Number Publication Date
PT95112A true PT95112A (pt) 1991-04-18
PT95112B PT95112B (pt) 1997-04-30

Family

ID=11183718

Family Applications (1)

Application Number Title Priority Date Filing Date
PT95112A PT95112B (pt) 1989-08-28 1990-08-28 Processo para a preparacao de derivados de peptido farmacologicamente activos

Country Status (8)

Country Link
US (1) US5182265A (pt)
EP (1) EP0421074B1 (pt)
JP (1) JPH0390098A (pt)
KR (1) KR910004659A (pt)
DE (1) DE69018914T2 (pt)
ES (1) ES2071710T3 (pt)
IT (1) IT1231342B (pt)
PT (1) PT95112B (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2378480A1 (en) * 1999-08-09 2001-02-15 Tripep Ab Pharmaceutical compositions containing tripeptides
US6258932B1 (en) 1999-08-09 2001-07-10 Tripep Ab Peptides that block viral infectivity and methods of use thereof
DE60130641T2 (de) 2000-02-07 2008-06-26 Wisconsin Alumni Research Foundation, Madison Pharmakologisch aktive antivirale peptide und methoden zu ihrer anwendung
US6593455B2 (en) 2001-08-24 2003-07-15 Tripep Ab Tripeptide amides that block viral infectivity and methods of use thereof
US6455670B1 (en) 2001-09-06 2002-09-24 Tripep Ab Pentamer peptide amide, ALGPG-NH2, that inhibits viral infectivity and methods of use thereof
EP1436317A1 (en) 2001-09-19 2004-07-14 Tripep Ab Molecules that block viral infectivity and methods of use thereof
WO2005060541A2 (en) * 2003-12-01 2005-07-07 Wisconsin Alumni Research Foundation Peptides and methods for inducing cellular resistance to infection
KR200447742Y1 (ko) * 2009-07-10 2010-02-12 조용진 법단

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1063727A (en) * 1965-04-12 1967-03-30 Ici Ltd Amide derivatives
GB1465235A (en) * 1975-04-29 1977-02-23 Sagami Chem Res Process for preparing peptides
GB8322414D0 (en) * 1983-08-19 1983-09-21 Szelke M Renin inhibitors
JPS61148198A (ja) * 1984-12-22 1986-07-05 Ajinomoto Co Inc 新規トリペプチド化合物および甘味剤
IT1190433B (it) * 1985-12-11 1988-02-16 Prodotti Antibiotici Spa Peptidi correlati al lisozima

Also Published As

Publication number Publication date
IT1231342B (it) 1991-11-28
KR910004659A (ko) 1991-03-29
ES2071710T3 (es) 1995-07-01
EP0421074A1 (en) 1991-04-10
US5182265A (en) 1993-01-26
EP0421074B1 (en) 1995-04-26
JPH0390098A (ja) 1991-04-16
DE69018914T2 (de) 1995-11-16
DE69018914D1 (de) 1995-06-01
IT8921567A0 (it) 1989-08-28
PT95112B (pt) 1997-04-30

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Legal Events

Date Code Title Description
BB1A Laying open of patent application

Effective date: 19901207

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20000731