PT882045E - Processo para a preparacao de granisetron - Google Patents

Processo para a preparacao de granisetron

Info

Publication number
PT882045E
PT882045E PT97904526T PT97904526T PT882045E PT 882045 E PT882045 E PT 882045E PT 97904526 T PT97904526 T PT 97904526T PT 97904526 T PT97904526 T PT 97904526T PT 882045 E PT882045 E PT 882045E
Authority
PT
Portugal
Prior art keywords
granisetron
preparation
cyclising
compound
preparing
Prior art date
Application number
PT97904526T
Other languages
English (en)
Inventor
David Alan Jones
Neal Ward
Victor Witold Jacewicz
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of PT882045E publication Critical patent/PT882045E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/14Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing 9-azabicyclo [3.3.1] nonane ring systems, e.g. granatane, 2-aza-adamantane; Cyclic acetals thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
PT97904526T 1996-02-13 1997-02-11 Processo para a preparacao de granisetron PT882045E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9602866.7A GB9602866D0 (en) 1996-02-13 1996-02-13 Novel process

Publications (1)

Publication Number Publication Date
PT882045E true PT882045E (pt) 2004-10-29

Family

ID=10788578

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97904526T PT882045E (pt) 1996-02-13 1997-02-11 Processo para a preparacao de granisetron

Country Status (9)

Country Link
US (1) US6268498B1 (pt)
EP (1) EP0882045B1 (pt)
JP (1) JP2000504715A (pt)
AT (1) ATE269863T1 (pt)
DE (1) DE69729631T2 (pt)
ES (1) ES2221951T3 (pt)
GB (1) GB9602866D0 (pt)
PT (1) PT882045E (pt)
WO (1) WO1997030049A1 (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9506119D0 (en) * 1995-03-25 1995-05-10 Smithkline Beecham Plc Chemical process
ES2197001B1 (es) * 2002-03-26 2004-11-16 Laboratorios Vita, S.A. Procedimiento de obtencion de un compuesto farmaceuticamente activo.
KR100965040B1 (ko) 2005-07-11 2010-06-21 미쓰비시 타나베 파마 코퍼레이션 옥심 유도체 및 그의 제조 방법
WO2007088557A1 (en) * 2006-02-01 2007-08-09 Natco Pharma Limited Process for highly pure crystalline granisetron base
ES2573324T3 (es) 2007-06-13 2016-06-07 Inke, S.A. Forma polimórfica de Granisetrón base, procedimientos para su obtención y formulación que la contiene

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3650772T2 (de) * 1985-04-27 2003-04-03 Hoffmann La Roche Derivate von Indazole-3-carboxamide und -3-carboxylsäure

Also Published As

Publication number Publication date
US6268498B1 (en) 2001-07-31
GB9602866D0 (en) 1996-04-10
EP0882045A1 (en) 1998-12-09
DE69729631T2 (de) 2005-06-09
DE69729631D1 (de) 2004-07-29
JP2000504715A (ja) 2000-04-18
ATE269863T1 (de) 2004-07-15
EP0882045B1 (en) 2004-06-23
ES2221951T3 (es) 2005-01-16
WO1997030049A1 (en) 1997-08-21

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