PT88177A - Processo para a preparacao de eteres contendo por exemplo, grupos azabiciclicos - Google Patents

Processo para a preparacao de eteres contendo por exemplo, grupos azabiciclicos

Info

Publication number
PT88177A
PT88177A PT88177A PT8817788A PT88177A PT 88177 A PT88177 A PT 88177A PT 88177 A PT88177 A PT 88177A PT 8817788 A PT8817788 A PT 8817788A PT 88177 A PT88177 A PT 88177A
Authority
PT
Portugal
Prior art keywords
azabicylic
eteres
groups
preparation
eteres containing
Prior art date
Application number
PT88177A
Other languages
English (en)
Other versions
PT88177B (pt
Inventor
Ian Anthony Cliffe
Original Assignee
Wyeth John & Brother Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB878718444A external-priority patent/GB8718444D0/en
Priority claimed from GB888811975A external-priority patent/GB8811975D0/en
Application filed by Wyeth John & Brother Ltd filed Critical Wyeth John & Brother Ltd
Publication of PT88177A publication Critical patent/PT88177A/pt
Publication of PT88177B publication Critical patent/PT88177B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/06Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing isoquinuclidine ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06Oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT88177A 1987-08-04 1988-08-03 Processo para a preparacao de eteres contendo por exemplo, grupos azabiciclicos PT88177B (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB878718444A GB8718444D0 (en) 1987-08-04 1987-08-04 Ethers
GB888811975A GB8811975D0 (en) 1988-05-20 1988-05-20 Ethers

Publications (2)

Publication Number Publication Date
PT88177A true PT88177A (pt) 1989-06-30
PT88177B PT88177B (pt) 1995-03-01

Family

ID=26292571

Family Applications (1)

Application Number Title Priority Date Filing Date
PT88177A PT88177B (pt) 1987-08-04 1988-08-03 Processo para a preparacao de eteres contendo por exemplo, grupos azabiciclicos

Country Status (15)

Country Link
US (3) US4929625A (pt)
EP (1) EP0306148B1 (pt)
JP (1) JP2711272B2 (pt)
KR (1) KR970002635B1 (pt)
AU (1) AU605896B2 (pt)
CA (1) CA1307790C (pt)
DE (1) DE3887039T2 (pt)
DK (1) DK170802B1 (pt)
ES (1) ES2061660T3 (pt)
FI (1) FI94250C (pt)
GB (1) GB2208510B (pt)
HU (1) HU203348B (pt)
IE (1) IE61026B1 (pt)
IL (1) IL87329A (pt)
PT (1) PT88177B (pt)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1230881B (it) * 1989-06-20 1991-11-08 Angeli Inst Spa Derivati del r(-) 3-chinuclidinolo
DK0456519T3 (da) * 1990-05-11 1994-11-07 Sankyo Co Piperidyloxy- og quinuclidinyloxyisoxazolderivater, deres fremstilling og deres terapeutiske anvendelse
YU84791A (sh) * 1990-05-19 1994-06-10 Boehringer Ingelheim Kg. Biciklicni 1-aza-cikloalkalni
GB9019973D0 (en) * 1990-09-12 1990-10-24 Wyeth John & Brother Ltd Azabicyclic derivatives
JPH05310732A (ja) * 1992-03-12 1993-11-22 Mitsubishi Kasei Corp シンノリン−3−カルボン酸誘導体
IL107184A (en) * 1992-10-09 1997-08-14 Abbott Lab Heterocyclic ether compounds that enhance cognitive function
US5948793A (en) * 1992-10-09 1999-09-07 Abbott Laboratories 3-pyridyloxymethyl heterocyclic ether compounds useful in controlling neurotransmitter release
GB9226573D0 (en) * 1992-12-21 1993-02-17 Ici Plc Heterocyclic compounds
US5998404A (en) * 1994-10-24 1999-12-07 Eli Lilly And Company Heterocyclic compounds and their use
US5605908A (en) * 1994-10-24 1997-02-25 Eli Lilly And Company Heterocyclic compounds and their use
US5929247A (en) * 1994-10-24 1999-07-27 Eli Lilly And Company Heterocyclic compounds and their preparation and use
US5512574A (en) * 1994-12-21 1996-04-30 American Home Products Corporation Quinuclidine and azabicyclo 2.2.1! heptane pyrazinyl ethers as muscarinic agonists
WO1997017955A1 (en) * 1995-11-13 1997-05-22 Eli Lilly And Company Method for treating anxiety
US5998434A (en) * 1995-12-06 1999-12-07 Eli Lilly And Company Composition for treating pain
US6133253A (en) * 1996-12-10 2000-10-17 Abbott Laboratories 3-Pyridyl enantiomers and their use as analgesics
US6455554B1 (en) 1999-06-07 2002-09-24 Targacept, Inc. Oxopyridinyl pharmaceutical compositions and methods for use
US20030147697A1 (en) * 2002-02-06 2003-08-07 Brady Patrick Richard Evaporative desorption soil treatment apparatus and process
US20050245567A1 (en) * 2002-08-14 2005-11-03 Dan Peters Novel quinuclidine derivatives and their use
GB0220581D0 (en) 2002-09-04 2002-10-09 Novartis Ag Organic Compound
US7418763B2 (en) * 2003-02-26 2008-09-02 Black & Decker Inc. Hand vacuum with filter indicator
BRPI0411608A (pt) * 2003-06-24 2006-08-08 Neurosearch As derivado de 8-aza-biciclo [3.2.1] octano, composição farmacêutica, uso do composto, e, método de tratamento, prevenção ou alìvio de uma doença, um distúrbio ou uma condição de um organismo animal vivo
AR049401A1 (es) 2004-06-18 2006-07-26 Novartis Ag Aza-biciclononanos
GB0415746D0 (en) 2004-07-14 2004-08-18 Novartis Ag Organic compounds
GB0521508D0 (en) 2005-10-21 2005-11-30 Novartis Ag Organic compounds
GB0525673D0 (en) 2005-12-16 2006-01-25 Novartis Ag Organic compounds
GB0525672D0 (en) 2005-12-16 2006-01-25 Novartis Ag Organic compounds
EP2018380B1 (en) * 2006-05-19 2011-10-19 Abbott Laboratories Cns active fused bicycloheterocycle substituted azabicyclic alkane derivatives

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2640829A (en) * 1950-11-10 1953-06-02 Smith Kline French Lab Isoquinolyl heterocyclic ethers
NL7109301A (pt) * 1970-07-15 1972-01-18
US4261990A (en) * 1979-03-09 1981-04-14 Ciba-Geigy Corporation N-alkyleneiminoalkyl-dicarboximides as antiallergics and antiasthmatics
FI74707C (fi) * 1982-06-29 1988-03-10 Sandoz Ag Foerfarande foer framstaellning av terapeutiskt anvaendbara alkylenoeverbryggade piperidylestrar eller -amider av bicykliska karboxylsyror.
GB8302483D0 (en) * 1983-01-29 1983-03-02 Beecham Group Plc Compounds
ZA848275B (en) * 1983-12-28 1985-08-28 Degussa New piridine-2-ethers or pyridine-2-thioethers having a nitrogen-containing cycloaliphatic ring
EP0405617A3 (en) * 1985-03-14 1992-11-25 Beecham Group P.L.C. Medicaments for the treatment of anxiety
DE3788057T2 (de) * 1986-12-17 1994-03-03 Glaxo Group Ltd Verwendung von heterocyclischen Verbindungen zur Behandlung von Depressionen.
US4766215A (en) * 1987-02-27 1988-08-23 American Home Products Corporation Histamine H1 -receptor antagonists
GB8718445D0 (en) * 1987-08-04 1987-09-09 Wyeth John & Brother Ltd Pyridyl-ethers
US4843074A (en) * 1988-05-17 1989-06-27 Marion Laboratories, Inc. 1-azabicyclo[2.2.2]octan-3-yl 2-aryl-3-azacyclo-2-hydroxypropionates and their quaternary salts
DE3839385A1 (de) * 1988-11-22 1990-05-23 Boehringer Ingelheim Kg Neue quinuclidine, ihre herstellung als arzneimittel und verfahren zu ihrer herstellung

Also Published As

Publication number Publication date
GB8818323D0 (en) 1988-09-07
AU2035988A (en) 1989-02-09
HUT48247A (en) 1989-05-29
IL87329A (en) 1992-12-01
US4997839A (en) 1991-03-05
DE3887039D1 (de) 1994-02-24
JP2711272B2 (ja) 1998-02-10
CA1307790C (en) 1992-09-22
FI94250C (fi) 1995-08-10
FI883632A (fi) 1989-02-05
FI883632A0 (fi) 1988-08-03
DK434488A (da) 1989-02-05
PT88177B (pt) 1995-03-01
DK434488D0 (da) 1988-08-03
EP0306148A2 (en) 1989-03-08
IE61026B1 (en) 1994-09-07
HU203348B (en) 1991-07-29
KR890003753A (ko) 1989-04-17
GB2208510A (en) 1989-04-05
US4929625A (en) 1990-05-29
GB2208510B (en) 1991-03-06
IE882375L (en) 1989-02-04
AU605896B2 (en) 1991-01-24
EP0306148B1 (en) 1994-01-12
IL87329A0 (en) 1989-01-31
DK170802B1 (da) 1996-01-22
FI94250B (fi) 1995-04-28
EP0306148A3 (en) 1990-05-23
DE3887039T2 (de) 1994-04-28
JPH0193585A (ja) 1989-04-12
ES2061660T3 (es) 1994-12-16
KR970002635B1 (ko) 1997-03-07
US5082843A (en) 1992-01-21

Similar Documents

Publication Publication Date Title
PT88177A (pt) Processo para a preparacao de eteres contendo por exemplo, grupos azabiciclicos
BR8803759A (pt) Processo para a preparacao de 2,2,6,6-tetrametil-4-piperidilaminas
BR8803908A (pt) Processo para a preparacao de um polimero de 1-olefina
BR8802484A (pt) Processo para a preparacao de isocianatos
BR8806789A (pt) Processo para a preparacao de um polibuteno
BR8801098A (pt) Processo para a preparacao de um composto de imidazola
PT94059A (pt) Processo para a preparacao de copolimetros hidrossoluveis, de n-vinilamidas
PT90119A (pt) Processo para a preparacao de um adocante
PT84316B (pt) Processo para a preparacao de cicloalcano {1,2 -b} indole-sulfamidas
PT83481B (pt) Processo para a preparacao de heteropolissacarideos de baixa viscosidade
BR8605269A (pt) Processo para preparacao de(2,2)-paraciclofano
BR8705524A (pt) Processo para preparacao de compostos
BR8707028A (pt) Processo para a preparacao de mercaptometilfenois
BR8506909A (pt) Processo para a preparacao de poliais polimericos
PT80956B (pt) Processo para a preparacao de 1,4-di-hidropiridinas
PT89039A (pt) Processo para a preparacao de l-ramnose
PT84108B (pt) Processo para a preparacao de acidos 7-piperazinil(substituido)-1-etil-6-fluoro-1,4-di-hidro-4-oxo-3-quinolinocarboxilicos
BR8803678A (pt) Processo para a preparacao de polieteramidas
PT84072B (pt) Processo para a preparacao de esteroides aminoglicosidicos
PT89056A (pt) Processo para a preparacao de hidroxilaminas substituidas
BR8704446A (pt) Processo para a preparacao de um hidrogel amplamente isento de monomeros
BR8706408A (pt) Processo para a preparacao de aldeidos
PT87946A (pt) Processo para a preparacao de derivados 4-amino susbtituido-1,2-dihidroxinaftaleno
BR8806351A (pt) Processo para a preparacao de fenil-ureias
PT81061B (pt) Processo para a preparacao de um polipeptideo vacinico

Legal Events

Date Code Title Description
FG3A Patent granted, date of granting

Effective date: 19940811