PT85547A - Processo de preparacao de composicao farmaceuticas a base de derivados de 2-mercapto-imidazol e de preparacao destes derivados - Google Patents
Processo de preparacao de composicao farmaceuticas a base de derivados de 2-mercapto-imidazol e de preparacao destes derivadosInfo
- Publication number
- PT85547A PT85547A PT85547A PT8554787A PT85547A PT 85547 A PT85547 A PT 85547A PT 85547 A PT85547 A PT 85547A PT 8554787 A PT8554787 A PT 8554787A PT 85547 A PT85547 A PT 85547A
- Authority
- PT
- Portugal
- Prior art keywords
- derivatives
- mercapto
- preparation
- pharmaceutical compositions
- compositions based
- Prior art date
Links
- OXFSTTJBVAAALW-UHFFFAOYSA-N 1,3-dihydroimidazole-2-thione Chemical class SC1=NC=CN1 OXFSTTJBVAAALW-UHFFFAOYSA-N 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 241000124008 Mammalia Species 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 230000003389 potentiating effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/84—Sulfur atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Enzymes And Modification Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US89816586A | 1986-08-18 | 1986-08-18 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT85547A true PT85547A (pt) | 1988-08-17 |
| PT85547B PT85547B (pt) | 1995-03-01 |
Family
ID=25409053
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT85547A PT85547B (pt) | 1986-08-18 | 1987-08-17 | Processo de preparacao de composicao farmaceuticas a base de derivados de 2-mercapto-imidazol e de preparacao destes derivados |
Country Status (15)
| Country | Link |
|---|---|
| EP (2) | EP0288488A4 (pt) |
| CN (1) | CN87105734A (pt) |
| AT (1) | ATE72430T1 (pt) |
| AU (1) | AU7910287A (pt) |
| DE (1) | DE3776613D1 (pt) |
| DK (1) | DK210488A (pt) |
| ES (1) | ES2038185T3 (pt) |
| GR (1) | GR3004345T3 (pt) |
| HU (2) | HU204037B (pt) |
| NZ (1) | NZ221427A (pt) |
| PH (1) | PH23530A (pt) |
| PT (1) | PT85547B (pt) |
| WO (1) | WO1988001267A1 (pt) |
| ZA (1) | ZA876073B (pt) |
| ZW (1) | ZW15387A1 (pt) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4835154A (en) * | 1987-06-01 | 1989-05-30 | Smithkline Beckman Corporation | 1-aralykyl-5-piperazinylmethyl-2-mercaptoimidazoles and 2-alkylthioimidazoles and their use as dopamine-βhydroxylase inhibitors |
| US4882348A (en) * | 1987-12-29 | 1989-11-21 | Smithkline Beckman Corporation | 2-(aminoalkylthio)imidazoles as dopamine-β-hydroxylase inhibitors |
| FR2928544A1 (fr) * | 2008-03-17 | 2009-09-18 | Oreal | Utilisation d'inhibiteurs de la dopamine-beta hydroxylase pour la pigmentation capillaire. |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5671074A (en) * | 1979-11-12 | 1981-06-13 | Takeda Chem Ind Ltd | 1,2-disubstituted-4-halogenoimidazole-5-acetic acid derivative |
| PT78388B (en) * | 1983-04-12 | 1986-09-15 | Smithkline Beckman Corp | Dopamine-beta-hydroxylase inhibitors |
| US4532331A (en) * | 1983-04-12 | 1985-07-30 | Smithkline Beckman Corporation | 1-Benzyl-2-aminomethyl imidazole derivatives |
-
1987
- 1987-08-12 NZ NZ221427A patent/NZ221427A/en unknown
- 1987-08-14 PH PH35675A patent/PH23530A/en unknown
- 1987-08-14 ZW ZW153/87A patent/ZW15387A1/xx unknown
- 1987-08-17 EP EP19870905838 patent/EP0288488A4/en active Pending
- 1987-08-17 AU AU79102/87A patent/AU7910287A/en not_active Abandoned
- 1987-08-17 WO PCT/US1987/002011 patent/WO1988001267A1/en not_active Ceased
- 1987-08-17 ZA ZA876073A patent/ZA876073B/xx unknown
- 1987-08-17 DE DE8787307259T patent/DE3776613D1/de not_active Expired - Fee Related
- 1987-08-17 EP EP87307259A patent/EP0260814B1/en not_active Expired - Lifetime
- 1987-08-17 HU HU874557A patent/HU204037B/hu unknown
- 1987-08-17 ES ES198787307259T patent/ES2038185T3/es not_active Expired - Lifetime
- 1987-08-17 PT PT85547A patent/PT85547B/pt not_active IP Right Cessation
- 1987-08-17 AT AT87307259T patent/ATE72430T1/de not_active IP Right Cessation
- 1987-08-17 HU HU911945A patent/HU911945D0/hu unknown
- 1987-08-18 CN CN198787105734A patent/CN87105734A/zh active Pending
-
1988
- 1988-04-18 DK DK210488A patent/DK210488A/da not_active Application Discontinuation
-
1992
- 1992-04-15 GR GR920400699T patent/GR3004345T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NZ221427A (en) | 1990-12-21 |
| ATE72430T1 (de) | 1992-02-15 |
| WO1988001267A1 (en) | 1988-02-25 |
| ES2038185T3 (es) | 1993-07-16 |
| CN87105734A (zh) | 1988-02-24 |
| EP0288488A1 (en) | 1988-11-02 |
| HU911945D0 (en) | 1991-12-30 |
| EP0288488A4 (en) | 1990-09-12 |
| DE3776613D1 (de) | 1992-03-19 |
| GR3004345T3 (pt) | 1993-03-31 |
| EP0260814B1 (en) | 1992-02-05 |
| PT85547B (pt) | 1995-03-01 |
| HUT50461A (en) | 1990-02-28 |
| ZW15387A1 (en) | 1987-11-18 |
| PH23530A (en) | 1989-08-25 |
| ZA876073B (en) | 1988-08-31 |
| DK210488D0 (da) | 1988-04-18 |
| AU7910287A (en) | 1988-03-08 |
| HU204037B (en) | 1991-11-28 |
| DK210488A (da) | 1988-04-18 |
| EP0260814A1 (en) | 1988-03-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG3A | Patent granted, date of granting |
Effective date: 19940811 |
|
| MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 19960229 |