PT84553B - Processo de preparacao de derivados de indenopirimidina - Google Patents

Processo de preparacao de derivados de indenopirimidina

Info

Publication number
PT84553B
PT84553B PT84553A PT8455387A PT84553B PT 84553 B PT84553 B PT 84553B PT 84553 A PT84553 A PT 84553A PT 8455387 A PT8455387 A PT 8455387A PT 84553 B PT84553 B PT 84553B
Authority
PT
Portugal
Prior art keywords
indenopyrimidine
derivatives
preparation
indenopyrimidine derivatives
Prior art date
Application number
PT84553A
Other languages
English (en)
Other versions
PT84553A (en
Inventor
Eriks Victor Krumkalns
Kenneth Steven Hirsch
Charles David Jones
Donald Grant Saunders
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PT84553A publication Critical patent/PT84553A/pt
Publication of PT84553B publication Critical patent/PT84553B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/26Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT84553A 1986-03-31 1987-03-25 Processo de preparacao de derivados de indenopirimidina PT84553B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/846,541 US4769378A (en) 1986-03-31 1986-03-31 Indenopyrimidine aromatase inhibitors

Publications (2)

Publication Number Publication Date
PT84553A PT84553A (en) 1987-04-01
PT84553B true PT84553B (pt) 1989-11-10

Family

ID=25298228

Family Applications (1)

Application Number Title Priority Date Filing Date
PT84553A PT84553B (pt) 1986-03-31 1987-03-25 Processo de preparacao de derivados de indenopirimidina

Country Status (21)

Country Link
US (1) US4769378A (pt)
EP (1) EP0240263B1 (pt)
JP (1) JPH0751568B2 (pt)
KR (1) KR890003838B1 (pt)
CN (1) CN1013673B (pt)
AR (1) AR245109A1 (pt)
AT (1) ATE78251T1 (pt)
AU (1) AU581809B2 (pt)
CA (1) CA1265140A (pt)
DE (1) DE3780338T2 (pt)
DK (1) DK165245C (pt)
ES (1) ES2042552T3 (pt)
GR (1) GR3005204T3 (pt)
HU (1) HU196379B (pt)
IE (1) IE59762B1 (pt)
IL (1) IL81978A (pt)
NZ (1) NZ219748A (pt)
PH (1) PH23398A (pt)
PT (1) PT84553B (pt)
SU (1) SU1470185A3 (pt)
ZA (1) ZA872162B (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5780465A (en) * 1997-04-03 1998-07-14 Dow Agrosciences Llc 4-substituted 5-polycyclylpyrimidine herbicides
SE0401790D0 (sv) * 2004-07-07 2004-07-07 Forskarpatent I Syd Ab Tamoxifen response in pre- and postmenopausal breast cancer patients
US7960400B2 (en) 2007-08-27 2011-06-14 Duquesne University Of The Holy Ghost Tricyclic compounds having cytostatic and/or cytotoxic activity and methods of use thereof
US7982035B2 (en) 2007-08-27 2011-07-19 Duquesne University Of The Holy Spirit Tricyclic compounds having antimitotic and/or antitumor activity and methods of use thereof
WO2009125299A2 (en) * 2008-03-05 2009-10-15 Lewis James D Quick-change fishing lure system and method of using
US20150311450A1 (en) * 2012-11-30 2015-10-29 Lg Chem, Ltd. New compounds and organic electronic device using the same

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133922A (en) * 1964-05-19 Z-cyano-
GB956269A (en) * 1960-04-01 1964-04-22 Manuf Prod Pharma Substituted indeno-pyrimidines
US3177216A (en) * 1961-12-28 1965-04-06 Searle & Co 4-trifluoromethyl-2-thio-5h-alka[d]-pyrimidines and congeners
US3763178A (en) * 1968-09-05 1973-10-02 American Home Prod Imidazolinyl phenyl carbonyl acid addition salts and related compounds
BE795636A (fr) * 1972-02-19 1973-08-20 Schering Ag Nitroimidazolylpyrimidines, et leur procede de preparation
US3925384A (en) * 1974-10-21 1975-12-09 Squibb & Sons Inc 2-Amino-4,5-dihydro-4-arylindeno pyrimidines
US4235893A (en) * 1978-05-08 1980-11-25 Brodie Angela M Ester derivatives of 4-hydroxy-4-androstene-3,17-dione and a method for inhibiting estrogen biosynthesis
NZ206968A (en) * 1983-02-02 1986-06-11 Lilly Co Eli Pyrimidine derivatives pharmaceutical formulations

Also Published As

Publication number Publication date
DE3780338T2 (de) 1993-03-04
SU1470185A3 (ru) 1989-03-30
US4769378A (en) 1988-09-06
KR890003838B1 (ko) 1989-10-05
DK165245C (da) 1993-03-22
EP0240263A3 (en) 1988-09-28
DE3780338D1 (de) 1992-08-20
JPH0751568B2 (ja) 1995-06-05
HUT43834A (en) 1987-12-28
ES2042552T3 (es) 1993-12-16
GR3005204T3 (pt) 1993-05-24
IE59762B1 (en) 1994-03-23
CN87102424A (zh) 1987-10-07
ZA872162B (en) 1988-10-26
PT84553A (en) 1987-04-01
CA1265140A (en) 1990-01-30
IL81978A0 (en) 1987-10-20
JPS62238275A (ja) 1987-10-19
EP0240263A2 (en) 1987-10-07
AU581809B2 (en) 1989-03-02
DK161187D0 (da) 1987-03-30
HU196379B (en) 1988-11-28
EP0240263B1 (en) 1992-07-15
ATE78251T1 (de) 1992-08-15
NZ219748A (en) 1989-05-29
IE870812L (en) 1987-09-30
CN1013673B (zh) 1991-08-28
AR245109A1 (es) 1993-12-30
PH23398A (en) 1989-07-26
IL81978A (en) 1991-03-10
DK165245B (da) 1992-10-26
AU7075287A (en) 1987-10-08
KR870008857A (ko) 1987-10-21
DK161187A (da) 1987-10-01

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