PT75728A - 6-fluoro-3-<3-(1-heterocyclo)propyl>-1,2-benzisoxazoles a process for their preparation pharmaceutical compositions thereof and their use as medicaments - Google Patents
6-fluoro-3-<3-(1-heterocyclo)propyl>-1,2-benzisoxazoles a process for their preparation pharmaceutical compositions thereof and their use as medicamentsInfo
- Publication number
- PT75728A PT75728A PT75728A PT7572882A PT75728A PT 75728 A PT75728 A PT 75728A PT 75728 A PT75728 A PT 75728A PT 7572882 A PT7572882 A PT 7572882A PT 75728 A PT75728 A PT 75728A
- Authority
- PT
- Portugal
- Prior art keywords
- fluoro
- heterocyclo
- benzisoxazoles
- medicaments
- propyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/10—Spiro-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/366,245 US4458075A (en) | 1982-04-09 | 1982-04-09 | 6-Fluoro-3-[3-(1-heterocyclo)propyl]-1,2-benzisoxazoles |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT75728A true PT75728A (en) | 1982-11-01 |
| PT75728B PT75728B (en) | 1985-11-11 |
Family
ID=23442245
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT75728A PT75728B (en) | 1982-04-09 | 1982-10-22 | 6-fluoro-3-<3-(1-heterocyclo)propyl>-1,2-benzisoxazoles a process for their preparation pharmaceutical compositions thereof and their use as medicaments |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US4458075A (pt) |
| EP (1) | EP0091512B1 (pt) |
| JP (1) | JPS58177981A (pt) |
| AT (1) | ATE34172T1 (pt) |
| AU (1) | AU560513B2 (pt) |
| CA (1) | CA1189858A (pt) |
| DE (1) | DE3278472D1 (pt) |
| DK (1) | DK474582A (pt) |
| ES (1) | ES516828A0 (pt) |
| FI (1) | FI823434L (pt) |
| GR (1) | GR77705B (pt) |
| HU (1) | HU191076B (pt) |
| IL (1) | IL66868A (pt) |
| NO (1) | NO823557L (pt) |
| NZ (1) | NZ202045A (pt) |
| PH (1) | PH18365A (pt) |
| PT (1) | PT75728B (pt) |
| ZA (1) | ZA827814B (pt) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4894461A (en) * | 1981-04-27 | 1990-01-16 | Hoechst-Roussel Pharmaceuticals, Inc. | 3-(γ-chloropropyl)-6-fluoro-1,2-benzisoxazole |
| US4980365A (en) * | 1987-07-13 | 1990-12-25 | Hoechst-Roussel Pharmaceuticals Inc. | N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents |
| US4954511A (en) * | 1988-03-14 | 1990-09-04 | Hoechst-Roussell Pharmaceuticals Inc. | 4-pentafluorophenoxypiperidines |
| US4914204A (en) * | 1988-03-14 | 1990-04-03 | Hoechst-Roussel Pharmaceuticals Incorporated | 4-Pentafluorophenoxypiperidines |
| US4861889A (en) * | 1988-03-14 | 1989-08-29 | Hoechst-Roussel Pharmaceuticals, Inc. | 3-(2,3,4,5,6-pentafluorophenoxy)-8-azabicyclo[3.2.1]octanes |
| US5114936A (en) * | 1990-08-23 | 1992-05-19 | Hoechst-Roussel Pharmaceuticals Incorporated | 6,7-dihydro-3-phenyl-1,2-benzisoxazol-4(5h)-ones and -ols, compositions and pharmaceutical use |
| US5750542A (en) | 1993-09-28 | 1998-05-12 | Pfizer | Benzisoxazole and benzisothizole derivatives as cholinesterase inhibitors |
| EP1535912A1 (en) * | 2000-04-28 | 2005-06-01 | Arcadia Pharmaceuticals Inc. | Muscarinic agonists |
| CN1249051C (zh) * | 2000-04-28 | 2006-04-05 | 阿卡蒂亚药品公司 | 毒蕈碱性激动剂 |
| DE102019103847A1 (de) | 2019-02-15 | 2020-08-20 | Vetron Typical Europe Gmbh | Nähmaschine |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS4970963A (pt) * | 1972-11-09 | 1974-07-09 | ||
| GB1488003A (en) * | 1973-10-23 | 1977-10-05 | Lilly Industries Ltd | 1,2-benzisoxazole derivatives processes for their preparation and their use as pharmaceuticals |
| FI60390C (fi) * | 1975-03-05 | 1982-01-11 | Sumitomo Chemical Co | Foerfarande foer framstaellning av neuroleptiska butyrofenoner |
| JPS51136666A (en) * | 1975-05-19 | 1976-11-26 | Dainippon Pharmaceut Co Ltd | Process for preparing 3-aminoalkyl-1,2-benzisoxazole derivatives. |
| JPS6043064B2 (ja) * | 1979-11-28 | 1985-09-26 | ウェルファイド株式会社 | 新規イソオキサゾ−ル誘導体 |
-
1982
- 1982-04-09 US US06/366,245 patent/US4458075A/en not_active Expired - Lifetime
- 1982-09-24 IL IL66868A patent/IL66868A/xx unknown
- 1982-09-30 NZ NZ202045A patent/NZ202045A/en unknown
- 1982-10-08 FI FI823434A patent/FI823434L/fi not_active Application Discontinuation
- 1982-10-22 PT PT75728A patent/PT75728B/pt unknown
- 1982-10-22 GR GR69602A patent/GR77705B/el unknown
- 1982-10-23 EP EP82109802A patent/EP0091512B1/en not_active Expired
- 1982-10-23 AT AT82109802T patent/ATE34172T1/de not_active IP Right Cessation
- 1982-10-23 DE DE8282109802T patent/DE3278472D1/de not_active Expired
- 1982-10-26 PH PH28038A patent/PH18365A/en unknown
- 1982-10-26 DK DK474582A patent/DK474582A/da not_active Application Discontinuation
- 1982-10-26 HU HU823416A patent/HU191076B/hu unknown
- 1982-10-26 JP JP57186908A patent/JPS58177981A/ja active Pending
- 1982-10-26 ES ES516828A patent/ES516828A0/es active Granted
- 1982-10-26 NO NO823557A patent/NO823557L/no unknown
- 1982-10-26 AU AU89777/82A patent/AU560513B2/en not_active Ceased
- 1982-10-26 CA CA000414158A patent/CA1189858A/en not_active Expired
- 1982-10-26 ZA ZA827814A patent/ZA827814B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AU8977782A (en) | 1983-10-13 |
| IL66868A0 (en) | 1982-12-31 |
| PT75728B (en) | 1985-11-11 |
| ES8308560A1 (es) | 1983-09-16 |
| US4458075A (en) | 1984-07-03 |
| DK474582A (da) | 1983-10-10 |
| ATE34172T1 (de) | 1988-05-15 |
| ES516828A0 (es) | 1983-09-16 |
| PH18365A (en) | 1985-06-13 |
| HU191076B (en) | 1987-01-28 |
| FI823434A0 (fi) | 1982-10-08 |
| EP0091512B1 (en) | 1988-05-11 |
| FI823434L (fi) | 1983-10-10 |
| JPS58177981A (ja) | 1983-10-18 |
| ZA827814B (en) | 1983-08-31 |
| NO823557L (no) | 1983-10-10 |
| EP0091512A2 (en) | 1983-10-19 |
| CA1189858A (en) | 1985-07-02 |
| EP0091512A3 (en) | 1984-12-12 |
| NZ202045A (en) | 1986-03-14 |
| DE3278472D1 (en) | 1988-06-16 |
| AU560513B2 (en) | 1987-04-09 |
| GR77705B (pt) | 1984-09-25 |
| IL66868A (en) | 1987-07-31 |
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| PT75728A (en) | 6-fluoro-3-<3-(1-heterocyclo)propyl>-1,2-benzisoxazoles a process for their preparation pharmaceutical compositions thereof and their use as medicaments | |
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| ZA827815B (en) | 1-(3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl)-4-(substituted)-piperazines and-piperidines,and a process for the preparation thereof,pharmaceutical compositions containing the same and their use as medicaments | |
| IL65598A (en) | 1-(3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl)-4-hydroxy-4-phenylpiperidines,a process for their preparation and their use as medicaments |