PT74293B - Chemical methods and intermediates for preparing substituted pyrimidinones - Google Patents
Chemical methods and intermediates for preparing substituted pyrimidinonesInfo
- Publication number
- PT74293B PT74293B PT74293A PT7429382A PT74293B PT 74293 B PT74293 B PT 74293B PT 74293 A PT74293 A PT 74293A PT 7429382 A PT7429382 A PT 7429382A PT 74293 B PT74293 B PT 74293B
- Authority
- PT
- Portugal
- Prior art keywords
- intermediates
- chemical methods
- preparing substituted
- substituted pyrimidinones
- pyrimidine
- Prior art date
Links
- 239000000543 intermediate Substances 0.000 title 1
- 239000000126 substance Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000006570 (C5-C6) heteroaryl group Chemical group 0.000 abstract 1
- BBZZGDLNBVRFFI-UHFFFAOYSA-N 4,5-dihydropyrimidine Chemical compound C1CN=CN=C1 BBZZGDLNBVRFFI-UHFFFAOYSA-N 0.000 abstract 1
- CZPWVGJYEJSRLH-UHFFFAOYSA-N Pyrimidine Chemical compound C1=CN=CN=C1 CZPWVGJYEJSRLH-UHFFFAOYSA-N 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 239000000739 antihistaminic agent Substances 0.000 abstract 1
- -1 hydroxy, mercapto Chemical group 0.000 abstract 1
- 125000002816 methylsulfanyl group Chemical group [H]C([H])([H])S[*] 0.000 abstract 1
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
- C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/56—One oxygen atom and one sulfur atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/232,105 US4352933A (en) | 1981-02-06 | 1981-02-06 | Chemical methods and intermediates for preparing substituted pyrimidinones |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT74293A PT74293A (en) | 1982-02-01 |
| PT74293B true PT74293B (pt) | 1983-06-28 |
Family
ID=22871897
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT74293A PT74293B (pt) | 1981-02-06 | 1982-01-15 | Chemical methods and intermediates for preparing substituted pyrimidinones |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US4352933A (forum.php) |
| EP (2) | EP0141973A3 (forum.php) |
| JP (1) | JPS57163378A (forum.php) |
| KR (1) | KR880001473B1 (forum.php) |
| AT (1) | ATE29882T1 (forum.php) |
| DE (1) | DE3277373D1 (forum.php) |
| DK (1) | DK49782A (forum.php) |
| ES (1) | ES8302723A1 (forum.php) |
| GR (1) | GR75406B (forum.php) |
| IE (1) | IE53005B1 (forum.php) |
| IL (1) | IL64621A (forum.php) |
| PT (1) | PT74293B (forum.php) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4477663A (en) * | 1981-02-06 | 1984-10-16 | Smithkline Beckman Corporation | Intermediates for preparing substituted pyrimidinones |
| US4620001A (en) * | 1981-02-06 | 1986-10-28 | Smithkline Beckman Corporation | Chemical methods and intermediates for preparing substituted pyrimidinones |
| US4675406A (en) * | 1981-02-06 | 1987-06-23 | Smithkline Beckman Corporation | Substituted pyrimidinones |
| DK230482A (da) * | 1981-05-30 | 1982-12-01 | Smith Kline French Lab | Pyrimidonsalt og fremstilling heraf |
| DE3365869D1 (en) * | 1982-07-30 | 1986-10-09 | Smith Kline French Lab | Amino pyrimidinones and their preparation |
| US4772704A (en) * | 1983-09-21 | 1988-09-20 | Bristol-Myers Company | 2,5-disubstituted-4(3H)-pyrimidones having histamine H2 -receptor antagonist activity |
| JP2807577B2 (ja) * | 1990-06-15 | 1998-10-08 | エーザイ株式会社 | 環状アミド誘導体 |
| ES2203988T3 (es) | 1997-11-06 | 2004-04-16 | Smithkline Beecham Plc | Compuestos de pirimidinona y composiciones farmaceuticas que los contienen. |
| EP2382865A1 (de) | 2010-04-28 | 2011-11-02 | Bayer CropScience AG | Synergistische Wirkstoffkombinationen |
| US9241486B2 (en) | 2012-08-31 | 2016-01-26 | Bayer Cropscience Lp | Combination and methods for controlling turfgrass pests |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1419994A (en) * | 1973-05-03 | 1976-01-07 | Smith Kline French Lab | Heterocyclicalkylaminotheterocyclic compounds methods for their preparation and compositions comprising them |
| US4153793A (en) * | 1973-05-03 | 1979-05-08 | Smith Kline & French Laboratories Limited | Imidazo alkylamino pyrimidones |
| US4145546A (en) * | 1975-10-02 | 1979-03-20 | Smith Kline & French Laboratories Limited | 4-Pyrimidone compounds |
| US4154834A (en) * | 1975-12-29 | 1979-05-15 | Smith Kline & French Laboratories Limited | Substituted isocytosines having histamine H2 -antagonist activity |
| US4216318A (en) * | 1975-12-29 | 1980-08-05 | Smith Kline & French Laboratories Limited | Heterocyclic alkyl 4-pyrimidones |
| GB1582528A (en) * | 1977-03-25 | 1981-01-07 | Smith Kline French Lab | Amino pyrimidone derivatives |
| IN151188B (forum.php) * | 1978-02-13 | 1983-03-05 | Smith Kline French Lab | |
| AU527202B2 (en) * | 1978-04-11 | 1983-02-24 | Smith Kline & French Laboratories Limited | 2-aminopyrimidones |
| ZA793443B (en) * | 1978-07-26 | 1980-12-31 | Glaxo Group Ltd | Heterocyclic derivatives |
| US4374836A (en) * | 1978-10-16 | 1983-02-22 | Imperial Chemical Industries Ltd. | Antisecretory heterocyclic derivatives, process for their manufacture and pharmaceutical compositions containing them |
| DE2962609D1 (en) * | 1979-04-11 | 1982-06-09 | Estel Hoogovens Bv | Expandable coiler mandrel |
| CA1140129A (en) * | 1979-08-21 | 1983-01-25 | Ronald J. King | 4-pyrimidone derivatives |
-
1981
- 1981-02-06 US US06/232,105 patent/US4352933A/en not_active Expired - Fee Related
- 1981-12-22 IL IL64621A patent/IL64621A/xx unknown
-
1982
- 1982-01-15 PT PT74293A patent/PT74293B/pt unknown
- 1982-02-03 ES ES509274A patent/ES8302723A1/es not_active Expired
- 1982-02-04 EP EP84111114A patent/EP0141973A3/en not_active Ceased
- 1982-02-04 EP EP82300562A patent/EP0058055B1/en not_active Expired
- 1982-02-04 DE DE8282300562T patent/DE3277373D1/de not_active Expired
- 1982-02-04 AT AT82300562T patent/ATE29882T1/de not_active IP Right Cessation
- 1982-02-05 JP JP57018094A patent/JPS57163378A/ja active Pending
- 1982-02-05 GR GR67224A patent/GR75406B/el unknown
- 1982-02-05 DK DK49782A patent/DK49782A/da not_active Application Discontinuation
- 1982-02-06 KR KR8200509A patent/KR880001473B1/ko not_active Expired
- 1982-02-08 IE IE270/82A patent/IE53005B1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES509274A0 (es) | 1983-01-16 |
| EP0141973A3 (en) | 1986-02-26 |
| EP0058055B1 (en) | 1987-09-23 |
| IL64621A0 (en) | 1982-03-31 |
| IE53005B1 (en) | 1988-05-11 |
| IL64621A (en) | 1985-10-31 |
| DK49782A (da) | 1982-08-07 |
| EP0058055A3 (en) | 1982-10-27 |
| IE820270L (en) | 1982-08-06 |
| US4352933A (en) | 1982-10-05 |
| KR880001473B1 (ko) | 1988-08-13 |
| DE3277373D1 (en) | 1987-10-29 |
| GR75406B (forum.php) | 1984-07-13 |
| EP0058055A2 (en) | 1982-08-18 |
| PT74293A (en) | 1982-02-01 |
| ES8302723A1 (es) | 1983-01-16 |
| KR830009088A (ko) | 1983-12-17 |
| EP0141973A2 (en) | 1985-05-22 |
| ATE29882T1 (de) | 1987-10-15 |
| JPS57163378A (en) | 1982-10-07 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ES2072276T5 (es) | Alfa-arilacrilatos substituidos con heterociclos y fungicidas que contienen estos compuestos. | |
| ES8706146A1 (es) | Un procedimiento para preparar derivados de piridina | |
| ES2063929T3 (es) | Derivados de acido oxi-fenoxiacetico heterociclicos y su uso como herbicidas. | |
| GB1447108A (en) | Pyrimidone compounds | |
| PT74293B (pt) | Chemical methods and intermediates for preparing substituted pyrimidinones | |
| KR830005216A (ko) | 이미다조[4,5-b] 피리딘 유도체의 제조방법 | |
| IE32035L (en) | Preparation of substituted vinyl pyrimidines and¹imidazolines | |
| KR870006033A (ko) | 피리디닐 피리미딘 유도체의 제조 방법 | |
| ES2177580T3 (es) | Procedimiento para la preparacion de derivados heterociclicos de fluoralqueniltio. | |
| GB1366540A (en) | Fused 1 2 4 thiadiazolines and a process for their preparation | |
| AU553927B2 (en) | Oxazolo- thiazolo- imidazolo (5,4-b) pyridines | |
| ATE111097T1 (de) | Fungizide. | |
| GB1340160A (en) | 7-ureidocephalosporins | |
| GB1185039A (en) | Pyrimidine Derivatives and Compositions containing them | |
| ATE17943T1 (de) | Als schaedlingsbekaempfungsmittel wirksame pyrimidin derivate. | |
| ES8304094A1 (es) | Procedimiento para preparar una sal de pirimidona. | |
| KR830001931A (ko) | 히스타민 길항체의 제조방법 | |
| ES8705876A1 (es) | Un procedimiento para preparar 3-(piperidinil)-y 3-(pirrolidinil)-1h-indazoles | |
| SU1496220A1 (ru) | Трис(2-гидроксиэтил)аммониевые соли гетерилтиоуксусных кислот, обладающие гиполипидемическим действием | |
| JPS57176981A (en) | Dihydropyrimidine compound and its salts | |
| JPS56167696A (en) | Pyrimidine, its preparation and insecticide, acaricide and nematocide containing the same as active constituent | |
| SE7702797L (sv) | Forfarande for framstellning av 5-fluorouracilderivat | |
| ES8205410A1 (es) | Un procedimiento para preparar una pirazolo-piridinona | |
| KR870010040A (ko) | N-(2-피리미디닐) 피페라지닐 부틸 아자스피로 데칸디온의 제조방법 | |
| KR830005159A (ko) | 살균제 티오글리클산 아닐리드와 그의 제조방법 및 동물질을 함유하는 살충조성물 |