PT2016064E - Métodos para a preparação de compostos contendo pirazole - Google Patents

Métodos para a preparação de compostos contendo pirazole Download PDF

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Publication number
PT2016064E
PT2016064E PT07761874T PT07761874T PT2016064E PT 2016064 E PT2016064 E PT 2016064E PT 07761874 T PT07761874 T PT 07761874T PT 07761874 T PT07761874 T PT 07761874T PT 2016064 E PT2016064 E PT 2016064E
Authority
PT
Portugal
Prior art keywords
preparation
pyrazole
methods
containing compounds
disorders
Prior art date
Application number
PT07761874T
Other languages
English (en)
Inventor
Xiaohu Deng
Jimmy T Liang
Neelakandha Mani
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of PT2016064E publication Critical patent/PT2016064E/pt

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D317/00Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/10Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
    • C07D317/14Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D317/16Radicals substituted by halogen atoms or nitro radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PT07761874T 2006-05-05 2007-05-04 Métodos para a preparação de compostos contendo pirazole PT2016064E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US74649706P 2006-05-05 2006-05-05

Publications (1)

Publication Number Publication Date
PT2016064E true PT2016064E (pt) 2010-04-16

Family

ID=38566748

Family Applications (1)

Application Number Title Priority Date Filing Date
PT07761874T PT2016064E (pt) 2006-05-05 2007-05-04 Métodos para a preparação de compostos contendo pirazole

Country Status (12)

Country Link
US (1) US7915404B2 (pt)
EP (1) EP2016064B1 (pt)
CN (1) CN101479252B (pt)
AT (1) ATE459614T1 (pt)
CY (1) CY1110087T1 (pt)
DE (1) DE602007005117D1 (pt)
DK (1) DK2016064T3 (pt)
ES (1) ES2340217T3 (pt)
PL (1) PL2016064T3 (pt)
PT (1) PT2016064E (pt)
SI (1) SI2016064T1 (pt)
WO (1) WO2007131153A2 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE420881T1 (de) * 2003-09-17 2009-01-15 Janssen Pharmaceutica Nv Kondensierte heterocyclische verbindungen als modulatoren des serotoninrezeptors
US7598255B2 (en) * 2005-08-04 2009-10-06 Janssen Pharmaceutica Nv Pyrimidine compounds as serotonin receptor modulators
WO2009058810A1 (en) * 2007-11-02 2009-05-07 Janssen Pharmaceutica N.V. Process for the preparation of substituted 2,4,5,6,7,8-hexahydro-1,2,6-triaza-azulene derivatives
EP2370437B1 (en) * 2008-11-25 2013-09-04 Nerviano Medical Sciences S.r.l. Bicyclic pyrazole and isoxazole derivatives as antitumor and antineurodegenerative agents

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0272866A1 (en) * 1986-12-23 1988-06-29 Merck & Co. Inc. 1,4-Benzodiazepines with 5-membered heterocyclic rings
ATE420881T1 (de) * 2003-09-17 2009-01-15 Janssen Pharmaceutica Nv Kondensierte heterocyclische verbindungen als modulatoren des serotoninrezeptors
US7598255B2 (en) 2005-08-04 2009-10-06 Janssen Pharmaceutica Nv Pyrimidine compounds as serotonin receptor modulators

Also Published As

Publication number Publication date
DK2016064T3 (da) 2010-06-07
US7915404B2 (en) 2011-03-29
DE602007005117D1 (de) 2010-04-15
US20070260057A1 (en) 2007-11-08
WO2007131153A2 (en) 2007-11-15
PL2016064T3 (pl) 2010-08-31
CN101479252B (zh) 2014-01-29
ATE459614T1 (de) 2010-03-15
EP2016064A2 (en) 2009-01-21
SI2016064T1 (sl) 2010-07-30
WO2007131153A3 (en) 2008-01-10
ES2340217T3 (es) 2010-05-31
CN101479252A (zh) 2009-07-08
EP2016064B1 (en) 2010-03-03
CY1110087T1 (el) 2015-01-14

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