PT1373267E - Inibidores nao nucleosidicos da transcriptase reversa - Google Patents

Inibidores nao nucleosidicos da transcriptase reversa

Info

Publication number
PT1373267E
PT1373267E PT02716563T PT02716563T PT1373267E PT 1373267 E PT1373267 E PT 1373267E PT 02716563 T PT02716563 T PT 02716563T PT 02716563 T PT02716563 T PT 02716563T PT 1373267 E PT1373267 E PT 1373267E
Authority
PT
Portugal
Prior art keywords
alkyl
cycloalkyl
reverse transcriptase
dotted line
line represents
Prior art date
Application number
PT02716563T
Other languages
English (en)
Inventor
William W Ogilvie
D Ziel Robert
Naud Julie
O Meara Jeffrey
Dale R Cameron
Original Assignee
Boehringer Ingelheim Ca Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Ca Ltd filed Critical Boehringer Ingelheim Ca Ltd
Publication of PT1373267E publication Critical patent/PT1373267E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Saccharide Compounds (AREA)
PT02716563T 2001-03-22 2002-03-21 Inibidores nao nucleosidicos da transcriptase reversa PT1373267E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US27804401P 2001-03-22 2001-03-22

Publications (1)

Publication Number Publication Date
PT1373267E true PT1373267E (pt) 2005-05-31

Family

ID=23063458

Family Applications (1)

Application Number Title Priority Date Filing Date
PT02716563T PT1373267E (pt) 2001-03-22 2002-03-21 Inibidores nao nucleosidicos da transcriptase reversa

Country Status (11)

Country Link
US (1) US6716836B2 (pt)
EP (1) EP1373267B1 (pt)
JP (1) JP4148780B2 (pt)
AT (1) ATE288434T1 (pt)
AU (1) AU2002247573A1 (pt)
CA (1) CA2441996C (pt)
DE (1) DE60202853T2 (pt)
ES (1) ES2236500T3 (pt)
MX (1) MXPA03007966A (pt)
PT (1) PT1373267E (pt)
WO (1) WO2002076982A2 (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6706706B2 (en) 2002-03-27 2004-03-16 Boehringer Ingelheim International Gmbh Non-nucleoside reverse transcriptase inhibitors
US6806265B2 (en) * 2002-05-16 2004-10-19 Boehringer Ingelheim International Gmbh Non-nucleoside reverse transcriptase inhibitors
JP4391426B2 (ja) * 2002-09-19 2009-12-24 ベーリンガー インゲルハイム (カナダ) リミテッド 非ヌクレオシド逆転写酵素インヒビター
CA2495744A1 (en) 2002-09-19 2004-04-01 Boehringer Ingelheim (Canada) Ltd. Non-nucleoside reverse transcriptase inhibitors
JP2013149779A (ja) * 2012-01-19 2013-08-01 Semiconductor Components Industries Llc 半導体装置
EP3509588B1 (en) * 2016-09-12 2023-06-07 Integral Health,Inc. Bicyclic compounds useful as gpr120 modulators
EP3509587B1 (en) 2016-09-12 2023-12-06 Valo Health, Inc. Monocyclic compounds useful as gpr120 modulators

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5366972A (en) * 1989-04-20 1994-11-22 Boehringer Ingelheim Pharmaceuticals, Inc. 5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection
TW327171B (en) * 1994-02-18 1998-02-21 Boehringer Ingelheim Pharma 2-heteroaryl-5 for prevention or treatment of HIV infection
US5705499A (en) 1995-10-06 1998-01-06 Boehringer Ingelheim Pharmaceuticals, Inc. 8-arylalkyl- and 8-arylheteroalkyl-5,11-dihydro-6H-dipyrido 3,2-B:2',3'-e! 1!diazepines and their use in the treatment of HIV-1 infection
TWI270547B (en) 2000-06-16 2007-01-11 Boehringer Ingelheim Ca Ltd Non-nucleoside reverse transcriptase inhibitors

Also Published As

Publication number Publication date
WO2002076982A2 (en) 2002-10-03
MXPA03007966A (es) 2004-05-24
WO2002076982A3 (en) 2002-12-12
EP1373267A2 (en) 2004-01-02
US20030069226A1 (en) 2003-04-10
DE60202853D1 (de) 2005-03-10
ATE288434T1 (de) 2005-02-15
CA2441996A1 (en) 2002-10-03
EP1373267B1 (en) 2005-02-02
DE60202853T2 (de) 2006-02-09
JP4148780B2 (ja) 2008-09-10
ES2236500T3 (es) 2005-07-16
AU2002247573A1 (en) 2002-10-08
US6716836B2 (en) 2004-04-06
CA2441996C (en) 2011-07-19
JP2004523590A (ja) 2004-08-05

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