PT1080104E - Certos tiois heteroarilo substituidos inibidores da enzima conversora da endotelina - Google Patents
Certos tiois heteroarilo substituidos inibidores da enzima conversora da endotelinaInfo
- Publication number
- PT1080104E PT1080104E PT99923433T PT99923433T PT1080104E PT 1080104 E PT1080104 E PT 1080104E PT 99923433 T PT99923433 T PT 99923433T PT 99923433 T PT99923433 T PT 99923433T PT 1080104 E PT1080104 E PT 1080104E
- Authority
- PT
- Portugal
- Prior art keywords
- heteroarilian
- endotheline
- thyroids
- substitute
- inhibitors
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biophysics (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Genetics & Genomics (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Enzymes And Modification Thereof (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US6497998A | 1998-04-23 | 1998-04-23 |
Publications (1)
Publication Number | Publication Date |
---|---|
PT1080104E true PT1080104E (pt) | 2005-06-30 |
Family
ID=22059547
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT99923433T PT1080104E (pt) | 1998-04-23 | 1999-04-21 | Certos tiois heteroarilo substituidos inibidores da enzima conversora da endotelina |
Country Status (11)
Country | Link |
---|---|
EP (1) | EP1080104B1 (pt) |
JP (1) | JP3646062B2 (pt) |
AT (1) | ATE288922T1 (pt) |
AU (1) | AU750048B2 (pt) |
CA (1) | CA2324251A1 (pt) |
DE (1) | DE69923676T2 (pt) |
ES (1) | ES2237917T3 (pt) |
IL (1) | IL138688A0 (pt) |
PT (1) | PT1080104E (pt) |
WO (1) | WO1999055723A1 (pt) |
ZA (1) | ZA200004679B (pt) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6426354B1 (en) | 1998-04-23 | 2002-07-30 | Novartis Ag | Certain heteroaryl substituted thiol inhibitors of endothelin-converting enzyme |
US6423727B1 (en) | 1998-04-23 | 2002-07-23 | Novartis Ag | Certain thiol inhibitors of endothelin-converting enzyme |
JP4603646B2 (ja) * | 1999-11-15 | 2010-12-22 | 富士フイルムファインケミカルズ株式会社 | 新規なジピリジル誘導体 |
NL1014353C2 (nl) * | 2000-02-11 | 2001-08-15 | Dsm Nv | Werkwijze voor de bereiding van (R) -2-broom-3-fenylpropaanzuur. |
US20020028799A1 (en) * | 2000-07-06 | 2002-03-07 | Naylor Alasdair Mark | Treatment of male sexual dysfunction |
US6670479B2 (en) * | 2001-03-07 | 2003-12-30 | Advanced Research And Technology Institute, Inc. | Amination process |
US6777443B2 (en) | 2001-05-15 | 2004-08-17 | Novartis Ag | Dipeptide derivatives |
PT1430045E (pt) | 2001-09-21 | 2007-01-31 | Novartis Ag | Derivados de pirano como inibidores de ace e nep |
AU2003244467A1 (en) | 2002-02-04 | 2003-09-02 | Kaneka Corporation | Process for production of optically active 2-halogeno- carboxylic acids |
TWI259079B (en) | 2002-02-08 | 2006-08-01 | Merck & Co Inc | N-biphenyl(substituted methyl)aminocycloalkanecarboxamide derivatives |
ES2256727T3 (es) | 2002-02-08 | 2006-07-16 | MERCK & CO., INC. | Derivados de n-bifenilmetil aminocicloalcanocarboxamida. |
JP3975226B2 (ja) | 2006-01-11 | 2007-09-12 | 生化学工業株式会社 | シクロアルキルカルボニルアミノ酸誘導体及びその製造方法 |
JP4047365B2 (ja) | 2006-01-11 | 2008-02-13 | 生化学工業株式会社 | シクロアルカンカルボキサミド誘導体及びその製造方法 |
WO2007080884A1 (ja) * | 2006-01-11 | 2007-07-19 | Seikagaku Corporation | シクロアルキルカルボニルアミノ酸エステル誘導体及びその製造方法 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5432186A (en) * | 1993-11-16 | 1995-07-11 | Ciba-Geigy Corporation | Cyclic amino acid derivatives |
FR2745571B1 (fr) * | 1996-03-04 | 1998-06-19 | Inst Nat Sante Rech Med | Nouveaux derives soufres comportant une liaison amide, leur procede de preparation, leur application a titre de medicaments, et les compositions pharmaceutiques les renfermant |
FR2745570B1 (fr) * | 1996-03-04 | 1998-06-19 | Roussel Uclaf | Nouveaux derives soufres comportant une liaison retroamide, leur procede et intermediaires de preparation, leur application a titre de medicaments, et les compositions pharmaceutiques les renfermant |
-
1999
- 1999-04-21 PT PT99923433T patent/PT1080104E/pt unknown
- 1999-04-21 AU AU40319/99A patent/AU750048B2/en not_active Ceased
- 1999-04-21 JP JP2000545881A patent/JP3646062B2/ja not_active Expired - Fee Related
- 1999-04-21 EP EP99923433A patent/EP1080104B1/en not_active Expired - Lifetime
- 1999-04-21 WO PCT/EP1999/002694 patent/WO1999055723A1/en active IP Right Grant
- 1999-04-21 IL IL13868899A patent/IL138688A0/xx unknown
- 1999-04-21 ES ES99923433T patent/ES2237917T3/es not_active Expired - Lifetime
- 1999-04-21 CA CA002324251A patent/CA2324251A1/en not_active Abandoned
- 1999-04-21 DE DE69923676T patent/DE69923676T2/de not_active Expired - Fee Related
- 1999-04-21 AT AT99923433T patent/ATE288922T1/de not_active IP Right Cessation
-
2000
- 2000-09-06 ZA ZA200004679A patent/ZA200004679B/en unknown
Also Published As
Publication number | Publication date |
---|---|
EP1080104B1 (en) | 2005-02-09 |
DE69923676D1 (de) | 2005-03-17 |
DE69923676T2 (de) | 2006-01-12 |
ATE288922T1 (de) | 2005-02-15 |
CA2324251A1 (en) | 1999-11-04 |
EP1080104A1 (en) | 2001-03-07 |
WO1999055723A1 (en) | 1999-11-04 |
ZA200004679B (en) | 2002-04-24 |
JP3646062B2 (ja) | 2005-05-11 |
AU4031999A (en) | 1999-11-16 |
ES2237917T3 (es) | 2005-08-01 |
AU750048B2 (en) | 2002-07-11 |
JP2002513029A (ja) | 2002-05-08 |
IL138688A0 (en) | 2001-10-31 |
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