PL3782617T3 - Farmaceutyczne kompozycje żelowe zawierające lewodopę, karbidopę i entakapon - Google Patents

Farmaceutyczne kompozycje żelowe zawierające lewodopę, karbidopę i entakapon

Info

Publication number
PL3782617T3
PL3782617T3 PL20200070.9T PL20200070T PL3782617T3 PL 3782617 T3 PL3782617 T3 PL 3782617T3 PL 20200070 T PL20200070 T PL 20200070T PL 3782617 T3 PL3782617 T3 PL 3782617T3
Authority
PL
Poland
Prior art keywords
entacapone
carbidopa
levodopa
gel compositions
pharmaceutical gel
Prior art date
Application number
PL20200070.9T
Other languages
English (en)
Polish (pl)
Inventor
Roger BOLSÖY
Original Assignee
Lobsor Pharmaceuticals Aktiebolag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE1451034A external-priority patent/SE538425C2/en
Application filed by Lobsor Pharmaceuticals Aktiebolag filed Critical Lobsor Pharmaceuticals Aktiebolag
Publication of PL3782617T3 publication Critical patent/PL3782617T3/pl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • A61K31/277Nitriles; Isonitriles having a ring, e.g. verapamil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0024Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1652Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Dermatology (AREA)
  • Neurology (AREA)
  • Inorganic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PL20200070.9T 2014-09-04 2015-09-04 Farmaceutyczne kompozycje żelowe zawierające lewodopę, karbidopę i entakapon PL3782617T3 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE1451034A SE538425C2 (en) 2014-09-04 2014-09-04 Pharmaceutical compositions comprising levodopa, carbidopa and a comt inhibitor and method of administration thereof
SE1550344 2015-03-24

Publications (1)

Publication Number Publication Date
PL3782617T3 true PL3782617T3 (pl) 2024-06-24

Family

ID=55440194

Family Applications (2)

Application Number Title Priority Date Filing Date
PL20200070.9T PL3782617T3 (pl) 2014-09-04 2015-09-04 Farmaceutyczne kompozycje żelowe zawierające lewodopę, karbidopę i entakapon
PL15838800T PL3188725T3 (pl) 2014-09-04 2015-09-04 Kompozycje farmaceutyczne zawierające lewodopę, inhibitor dekarboksylazy dopaminy i inhibitor comt oraz sposób ich podawania

Family Applications After (1)

Application Number Title Priority Date Filing Date
PL15838800T PL3188725T3 (pl) 2014-09-04 2015-09-04 Kompozycje farmaceutyczne zawierające lewodopę, inhibitor dekarboksylazy dopaminy i inhibitor comt oraz sposób ich podawania

Country Status (16)

Country Link
US (5) US10071069B2 (cg-RX-API-DMAC7.html)
EP (3) EP4356907A1 (cg-RX-API-DMAC7.html)
JP (2) JP6622310B2 (cg-RX-API-DMAC7.html)
CN (1) CN107072973A (cg-RX-API-DMAC7.html)
AU (3) AU2015312430B2 (cg-RX-API-DMAC7.html)
CA (2) CA2959307C (cg-RX-API-DMAC7.html)
DK (2) DK3782617T3 (cg-RX-API-DMAC7.html)
ES (2) ES2844500T3 (cg-RX-API-DMAC7.html)
FI (1) FI3782617T3 (cg-RX-API-DMAC7.html)
HR (2) HRP20210025T1 (cg-RX-API-DMAC7.html)
HU (2) HUE052857T2 (cg-RX-API-DMAC7.html)
PL (2) PL3782617T3 (cg-RX-API-DMAC7.html)
PT (2) PT3188725T (cg-RX-API-DMAC7.html)
RS (1) RS65337B1 (cg-RX-API-DMAC7.html)
SI (2) SI3188725T1 (cg-RX-API-DMAC7.html)
WO (1) WO2016036308A1 (cg-RX-API-DMAC7.html)

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EP4356907A1 (en) 2014-09-04 2024-04-24 LobSor Pharmaceuticals Aktiebolag Pharmaceutical compositions comprising levodopa, a dopamine decarboxylase inhibitor and a comtinhibitor and method of administration thereof
WO2016083863A1 (en) * 2014-11-28 2016-06-02 Bial - Portela & Ca, S.A. Medicaments for slowing parkinson's disease
CN107847722B (zh) 2015-05-06 2021-05-18 辛纳吉勒公司 包含药物粒子的药用悬浮液、用于其配给的装置、以及其使用方法
WO2017039525A1 (en) 2015-09-04 2017-03-09 Lobsor Pharmaceuticals Aktiebolag Method of treating a dopamine related disorder in a subject by administering levodopa, in combination with a dopamine decarboxylase inhibitor and a catechol-o-methyltransferase inhibitor
US10874629B2 (en) * 2016-04-11 2020-12-29 University Of Canberra Ophthalmic compositions comprising levodopa, an antioxidant and an aqueous carrier
AU2017299710A1 (en) * 2016-07-20 2019-01-31 Abbvie Inc. Levodopa and carbidopa intestinal gel and methods of use
EP3275433A1 (en) 2016-07-29 2018-01-31 Som Innovation Biotech S.L. Sustained release composition comprising micronized tolcapone
JP7257322B2 (ja) 2017-02-13 2023-04-13 バイエル・アニマル・ヘルス・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング プラドフロキサシンを含有する液体組成物
WO2019129120A1 (en) * 2017-12-28 2019-07-04 Rpxds Co., Ltd Tolcapone for prevention and/or treatment of obesity and related metabolic diseases
KR20250043584A (ko) 2018-03-23 2025-03-28 롭서 파마슈티컬스 악티에볼라그 신경퇴행성 장애의 치료를 위한 약제학적 조성물의 연속 투여
EP3593819A1 (en) * 2018-07-10 2020-01-15 Medday Pharmaceuticals Compositions for therapeutic uses containing 5-htp and carbidopa
MX368750B (es) * 2018-08-31 2019-10-15 Cell Therapy And Tech S A De C V Composiciones farmaceuticas semisolidas de base oleosa conteniendo pirfenidona para su aplicacion en la reparacion tisular.
EP4417258A3 (en) * 2018-12-18 2024-10-30 Eli Lilly and Company Dose regimens for use of ly3154207 in the treatment of dopaminergic cns disorders
JP7506371B2 (ja) * 2020-01-20 2024-06-26 国立大学法人浜松医科大学 ドーパミン減少抑制剤
CA3174918A1 (en) * 2020-03-13 2021-09-16 Bial - Portela & Ca, S.A. Micronised opicapone
CN111643493B (zh) * 2020-05-26 2023-01-10 上海京新生物医药有限公司 一种高浓度左旋多巴制剂及其制备方法及其应用
PL4200280T3 (pl) 2020-10-07 2024-05-20 Eli Lilly And Company Pochodne fenylo-3,4-dihydroizochinolin-2(1h)-ylo-etan-1-onu jako dodatnie modulatory allosteryczne receptora dopaminy d1
WO2022158991A1 (en) * 2021-01-20 2022-07-28 Bial-Portela & Ca., S.A. Treatment of pain associated with parkinson's disease with opicapone in combination with levodopa
WO2025162373A1 (en) * 2024-01-30 2025-08-07 National Institute Of Biological Sciences, Beijing Electrophile-containing catechol-o-methyltransferase (comt) inhibitors for targeting the keap1/nrf2 pathway

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GB9004348D0 (en) 1990-02-27 1990-04-25 Orion Yhtymae Oy New use of catechol derivatives and their physiologically acceptable salts and esters
SE9203594D0 (sv) 1992-11-30 1992-11-30 Christer Nystroem Laekemedel i dispersa system
EP1135118A1 (en) * 1998-11-10 2001-09-26 Teva Pharmaceutical Industries Ltd. Dispersible compositions containing l-dopa ethyl ester
FI109453B (fi) 1999-06-30 2002-08-15 Orion Yhtymae Oyj Farmaseuttinen koostumus
US20100221321A1 (en) 2003-02-27 2010-09-02 Innercap Technologies, Inc. Apparatus And Methods For Delivering A Plurality Of Medicaments For Management Of Co-Morbid Diseases, Illnesses Or Conditions
CN1845728B (zh) * 2003-08-29 2013-06-19 转化医药公司 包含左旋多巴和卡比多巴的药物组合物
WO2005023185A2 (en) 2003-08-29 2005-03-17 Transform Pharmaceuticals, Inc. Pharmaceutical compositions and method of using levodopa and carbidopa
WO2005099678A1 (en) 2004-04-06 2005-10-27 Transform Pharmaceuticals, Inc. Pharmaceutical compositions and method of using levodopa and carbidopa
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CA2653683A1 (en) * 2006-05-31 2007-12-06 Solvay Pharmaceuticals Gmbh Long term 24-hour intestinal administration of levodopa/carbidopa
US8741342B2 (en) 2006-10-30 2014-06-03 Wockhardt Research Centre Pharmaceutical compositions comprising entacapone, levodopa, and carbidopa
PT2252284E (pt) * 2008-02-06 2011-08-23 Wockhardt Research Center COMPOSIÇÕES FARMACjUTICAS DE ENTACAPONE, LEVODOPA E CARBIDOPA COM BIODISPONIBILIDADE MELHORADA
US20130253056A1 (en) 2009-05-19 2013-09-26 Neuroderm, Ltd. Continuous Administration of Levodopa and/or Dopa Decarboxylase Inhibitors and Compositions for Same
PT2432454T (pt) * 2009-05-19 2017-06-12 Neuroderm Ltd Composições para administração contínua de inibidores de dopa decarboxilase
HUE047841T2 (hu) 2010-11-15 2020-05-28 Neuroderm Ltd L-dopa, dopa dekarboxiláz inhibitorok, katekol-o-metil transzferáz inhibitorok folyamatos adagolására szolgáló készítmények
WO2012147099A1 (en) 2011-04-25 2012-11-01 Suven Nishtaa Pharma Pvt. Ltd. Pharmaceutical compositions of levodopa, carbidopa and entacapone
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EP4356907A1 (en) 2014-09-04 2024-04-24 LobSor Pharmaceuticals Aktiebolag Pharmaceutical compositions comprising levodopa, a dopamine decarboxylase inhibitor and a comtinhibitor and method of administration thereof
SE538425C2 (en) 2014-09-04 2016-06-21 Lobsor Pharmaceuticals Ab Pharmaceutical compositions comprising levodopa, carbidopa and a comt inhibitor and method of administration thereof
WO2017039525A1 (en) 2015-09-04 2017-03-09 Lobsor Pharmaceuticals Aktiebolag Method of treating a dopamine related disorder in a subject by administering levodopa, in combination with a dopamine decarboxylase inhibitor and a catechol-o-methyltransferase inhibitor

Also Published As

Publication number Publication date
US12156858B2 (en) 2024-12-03
CA2959307A1 (en) 2016-03-10
ES2973289T3 (es) 2024-06-19
JP6889231B2 (ja) 2021-06-18
AU2020239682B2 (en) 2021-12-23
FI3782617T3 (fi) 2024-03-13
EP3782617B1 (en) 2024-01-03
US20210023033A1 (en) 2021-01-28
AU2022200291A1 (en) 2022-02-10
DK3782617T3 (da) 2024-03-04
EP4356907A1 (en) 2024-04-24
PL3188725T3 (pl) 2021-08-02
PT3782617T (pt) 2024-02-29
US11413262B2 (en) 2022-08-16
HUE052857T2 (hu) 2021-05-28
EP3188725B1 (en) 2020-10-28
US20220362193A1 (en) 2022-11-17
CA2959307C (en) 2023-03-28
AU2015312430A1 (en) 2017-03-30
CN107072973A (zh) 2017-08-18
US10071069B2 (en) 2018-09-11
US20250041257A1 (en) 2025-02-06
PT3188725T (pt) 2021-01-27
JP6622310B2 (ja) 2019-12-18
US20170231937A1 (en) 2017-08-17
DK3188725T3 (da) 2021-01-18
JP2017527623A (ja) 2017-09-21
EP3188725A4 (en) 2018-04-25
ES2844500T3 (es) 2021-07-22
WO2016036308A1 (en) 2016-03-10
US10786472B2 (en) 2020-09-29
AU2020239682A1 (en) 2020-10-15
EP3188725A1 (en) 2017-07-12
HRP20240314T1 (hr) 2024-05-24
EP3782617A1 (en) 2021-02-24
HRP20210025T1 (hr) 2021-03-05
AU2015312430B2 (en) 2020-06-25
AU2022200291B2 (en) 2024-01-25
RS65337B1 (sr) 2024-04-30
SI3782617T1 (sl) 2024-04-30
HUE066097T2 (hu) 2024-07-28
US20180338944A1 (en) 2018-11-29
SI3188725T1 (sl) 2021-04-30
CA3175785A1 (en) 2016-03-10
JP2020045353A (ja) 2020-03-26

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