PL364580A1 - Pochodne cyklopropyloindolu jako selektywne inhibitory zwrotnego wychwytu serotoniny - Google Patents

Pochodne cyklopropyloindolu jako selektywne inhibitory zwrotnego wychwytu serotoniny

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Publication number
PL364580A1
PL364580A1 PL02364580A PL36458002A PL364580A1 PL 364580 A1 PL364580 A1 PL 364580A1 PL 02364580 A PL02364580 A PL 02364580A PL 36458002 A PL36458002 A PL 36458002A PL 364580 A1 PL364580 A1 PL 364580A1
Authority
PL
Poland
Prior art keywords
cyclopropylindole
derivatives
serotonin reuptake
reuptake inhibitors
selective serotonin
Prior art date
Application number
PL02364580A
Other languages
English (en)
Inventor
Ronald Mattson
Derek Denhart
Jeffrey DESKUS
Jonathan Ditta
Lawrence MARCIN
James Epperson
John Catt
Dalton King
Mendi Higgins
Original Assignee
Bristol-Myers Squibb Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol-Myers Squibb Company filed Critical Bristol-Myers Squibb Company
Publication of PL364580A1 publication Critical patent/PL364580A1/pl

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    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
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    • C07D209/04—Indoles; Hydrogenated indoles
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    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
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    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
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    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
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    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
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    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
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    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Obesity (AREA)
  • Child & Adolescent Psychology (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychology (AREA)
  • Anesthesiology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
PL02364580A 2001-03-29 2002-03-05 Pochodne cyklopropyloindolu jako selektywne inhibitory zwrotnego wychwytu serotoniny PL364580A1 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US27988801P 2001-03-29 2001-03-29
US29312201P 2001-05-23 2001-05-23
US32780401P 2001-10-09 2001-10-09

Publications (1)

Publication Number Publication Date
PL364580A1 true PL364580A1 (pl) 2004-12-13

Family

ID=27403105

Family Applications (1)

Application Number Title Priority Date Filing Date
PL02364580A PL364580A1 (pl) 2001-03-29 2002-03-05 Pochodne cyklopropyloindolu jako selektywne inhibitory zwrotnego wychwytu serotoniny

Country Status (17)

Country Link
US (2) US6777437B2 (pl)
EP (1) EP1373203A1 (pl)
JP (1) JP2004531506A (pl)
AR (1) AR035793A1 (pl)
BG (1) BG108207A (pl)
CA (1) CA2442525A1 (pl)
CZ (1) CZ20032644A3 (pl)
EE (1) EE200300478A (pl)
HU (1) HUP0400343A2 (pl)
IL (1) IL158044A0 (pl)
IS (1) IS6969A (pl)
MX (1) MXPA03008807A (pl)
NO (1) NO20034307L (pl)
PE (1) PE20020975A1 (pl)
PL (1) PL364580A1 (pl)
SK (1) SK12012003A3 (pl)
WO (1) WO2002079152A1 (pl)

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ATE407671T1 (de) * 2003-05-09 2008-09-15 Esteve Labor Dr Verwendung von sulfonamid-derivate zur herstellung eines medikaments für die vorbeugung oder behandlung von essstörungen
DE10337184A1 (de) * 2003-08-13 2005-03-10 Gruenenthal Gmbh Substituierte 3-Pyrrolidin-Indol-Derivate
MX2007006408A (es) * 2004-11-29 2007-06-22 Warner Lambert Co Pirazolo[3,4-b]piridinas e indazoles terapeuticos.
EP1896076A2 (en) * 2005-06-27 2008-03-12 Daniel Drai Compositions and methods for enhancement of sexual function
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WO2007025144A1 (en) * 2005-08-24 2007-03-01 University Of Illinois - Chicago 5-ht2c receptor agonists as anorectic agents
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DE602007014206D1 (de) * 2006-06-22 2011-06-09 Univ Ramot Neuartige serotonin-wiederaufnahmehemmer als arzneimittel mit peripheriesystem-beschränkter aktivität
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WO2011106573A2 (en) 2010-02-24 2011-09-01 Oryzon Genomics, S.A. Lysine demethylase inhibitors for diseases and disorders associated with hepadnaviridae
US9616058B2 (en) 2010-02-24 2017-04-11 Oryzon Genomics, S.A. Potent selective LSD1 inhibitors and dual LSD1/MAO-B inhibitors for antiviral use
TWI429628B (zh) * 2010-03-29 2014-03-11 Univ Taipei Medical 吲哚基或吲哚啉基羥肟酸化合物
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