PL3166945T3 - Nowe pochodne triazolopirymidynonu lub triazolopirydynonu i ich zastosowanie - Google Patents
Nowe pochodne triazolopirymidynonu lub triazolopirydynonu i ich zastosowanieInfo
- Publication number
- PL3166945T3 PL3166945T3 PL15818399T PL15818399T PL3166945T3 PL 3166945 T3 PL3166945 T3 PL 3166945T3 PL 15818399 T PL15818399 T PL 15818399T PL 15818399 T PL15818399 T PL 15818399T PL 3166945 T3 PL3166945 T3 PL 3166945T3
- Authority
- PL
- Poland
- Prior art keywords
- triazolopyrimidinone
- novel
- triazolopyridinone
- derivatives
- triazolopyridinone derivatives
- Prior art date
Links
- LJRXNXBFJXXRNQ-UHFFFAOYSA-N 2h-[1,2,4]triazolo[4,3-a]pyridin-3-one Chemical class C1=CC=CN2C(=O)NN=C21 LJRXNXBFJXXRNQ-UHFFFAOYSA-N 0.000 title 1
- DDCYOMQDEGIFNS-UHFFFAOYSA-N triazolo[4,5-d]pyrimidin-5-one Chemical compound O=C1N=CC2=NN=NC2=N1 DDCYOMQDEGIFNS-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Neurology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
- Cardiology (AREA)
- Neurosurgery (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Epidemiology (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR20140087798 | 2014-07-11 | ||
| KR1020150068375A KR101739003B1 (ko) | 2014-07-11 | 2015-05-15 | 신규한 트리아졸로피리미디논 또는 트리아졸로피리디논 유도체, 및 이들의 용도 |
| PCT/KR2015/007219 WO2016006974A2 (en) | 2014-07-11 | 2015-07-10 | Novel triazolopyrimidinone or triazolopyridinone derivatives, and use thereof |
| EP15818399.6A EP3166945B1 (en) | 2014-07-11 | 2015-07-10 | Novel triazolopyrimidinone or triazolopyridinone derivatives, and use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PL3166945T3 true PL3166945T3 (pl) | 2020-09-07 |
Family
ID=55308036
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL15818399T PL3166945T3 (pl) | 2014-07-11 | 2015-07-10 | Nowe pochodne triazolopirymidynonu lub triazolopirydynonu i ich zastosowanie |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US9914737B2 (pl) |
| EP (1) | EP3166945B1 (pl) |
| JP (1) | JP6257835B2 (pl) |
| KR (1) | KR101739003B1 (pl) |
| CN (1) | CN106488918B (pl) |
| DK (1) | DK3166945T3 (pl) |
| ES (1) | ES2763566T3 (pl) |
| HU (1) | HUE048394T2 (pl) |
| PL (1) | PL3166945T3 (pl) |
| PT (1) | PT3166945T (pl) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP7369968B2 (ja) * | 2017-12-27 | 2023-10-27 | 公益財団法人がん研究会 | 抗がん剤 |
| EP3787630A4 (en) | 2018-04-30 | 2022-01-26 | Indiana University Research and Technology Corporation | FERROCHELATASE INHIBITORS AND METHODS OF USE |
| US20240317737A1 (en) * | 2021-01-11 | 2024-09-26 | St Pharm Co., Ltd. | Pyrrolopyridine derivative preparation method |
| CN118284609A (zh) * | 2021-12-01 | 2024-07-02 | St制药株式会社 | 用于制备三唑并嘧啶酮衍生物的方法 |
| JP2026507361A (ja) * | 2023-03-10 | 2026-03-02 | エスティー ファーム カンパニー リミテッド | 新規固体分散体およびその製造方法 |
| WO2024191138A1 (ko) * | 2023-03-10 | 2024-09-19 | 에스티팜 주식회사 | 트리아졸로피리미디논 유도체와 mek 억제제의 병용 요법 |
| WO2024191139A1 (ko) * | 2023-03-10 | 2024-09-19 | 에스티팜 주식회사 | Kras 변이 암의 예방 또는 치료용 조성물 |
| WO2025084446A1 (ko) * | 2023-10-16 | 2025-04-24 | 에스티팜 주식회사 | 트리아졸로피리미디논 유도체의 결정형 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20040242568A1 (en) * | 2003-03-25 | 2004-12-02 | Syrrx, Inc. | Dipeptidyl peptidase inhibitors |
| US20080242661A1 (en) | 2006-12-11 | 2008-10-02 | Graeme James Dykes | Novel compounds useful for the treatment of degenerative & inflammatory diseases |
| MX2014000536A (es) | 2011-07-13 | 2014-12-05 | Novartis Ag | Compuestos de 4-piperidinilo para usarse como inhibidores de tanquirasa. |
| PL2831077T3 (pl) | 2012-03-28 | 2016-10-31 | Bicykliczne pochodne pirazynonowe | |
| WO2013182546A1 (en) | 2012-06-07 | 2013-12-12 | F. Hoffmann-La Roche Ag | Pyrazolopyrimidone and pyrazolopyridone inhibitors of tankyrase |
| KR20150005711A (ko) | 2012-06-07 | 2015-01-14 | 에프. 호프만-라 로슈 아게 | 탄키라제 억제제로서 피롤로피리미돈 및 피롤로피리돈 |
-
2015
- 2015-05-15 KR KR1020150068375A patent/KR101739003B1/ko active Active
- 2015-07-10 EP EP15818399.6A patent/EP3166945B1/en active Active
- 2015-07-10 PL PL15818399T patent/PL3166945T3/pl unknown
- 2015-07-10 JP JP2017501285A patent/JP6257835B2/ja active Active
- 2015-07-10 ES ES15818399T patent/ES2763566T3/es active Active
- 2015-07-10 HU HUE15818399A patent/HUE048394T2/hu unknown
- 2015-07-10 DK DK15818399.6T patent/DK3166945T3/da active
- 2015-07-10 CN CN201580037780.XA patent/CN106488918B/zh active Active
- 2015-07-10 PT PT158183996T patent/PT3166945T/pt unknown
- 2015-07-10 US US15/325,651 patent/US9914737B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| EP3166945B1 (en) | 2019-10-09 |
| JP2017521439A (ja) | 2017-08-03 |
| CN106488918B (zh) | 2020-02-28 |
| ES2763566T3 (es) | 2020-05-29 |
| CN106488918A (zh) | 2017-03-08 |
| JP6257835B2 (ja) | 2018-01-10 |
| US9914737B2 (en) | 2018-03-13 |
| DK3166945T3 (da) | 2020-01-13 |
| PT3166945T (pt) | 2020-01-08 |
| EP3166945A4 (en) | 2018-02-14 |
| HUE048394T2 (hu) | 2020-07-28 |
| KR101739003B1 (ko) | 2017-05-23 |
| EP3166945A2 (en) | 2017-05-17 |
| US20170145016A1 (en) | 2017-05-25 |
| KR20160007348A (ko) | 2016-01-20 |
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