PL1853601T3 - Niesteroidowe modulatory receptora glukokortykoidowego - Google Patents

Niesteroidowe modulatory receptora glukokortykoidowego

Info

Publication number
PL1853601T3
PL1853601T3 PL06708243T PL06708243T PL1853601T3 PL 1853601 T3 PL1853601 T3 PL 1853601T3 PL 06708243 T PL06708243 T PL 06708243T PL 06708243 T PL06708243 T PL 06708243T PL 1853601 T3 PL1853601 T3 PL 1853601T3
Authority
PL
Poland
Prior art keywords
receptor modulators
glucocorticoid receptor
non steroidal
steroidal glucocorticoid
modulators
Prior art date
Application number
PL06708243T
Other languages
English (en)
Inventor
Ralf Plate
Guido Jenny Rudolf Zaman
Pedro Harold Han Hermkens
Christiaan Gerardus Johannes Maria Jans
Rogier Christian Buijsman
Man Adrianus Petrus Antonius De
Paolo Giovanni Martino Conti
Scott James Lusher
Willem Hendrik Abraham Dokter
Original Assignee
Msd Oss Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Msd Oss Bv filed Critical Msd Oss Bv
Publication of PL1853601T3 publication Critical patent/PL1853601T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
PL06708243T 2005-02-14 2006-02-14 Niesteroidowe modulatory receptora glukokortykoidowego PL1853601T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP05101086 2005-02-14
EP06708243A EP1853601B1 (en) 2005-02-14 2006-02-14 Non steroidal glucocorticoid receptor modulators
PCT/EP2006/050906 WO2006084917A1 (en) 2005-02-14 2006-02-14 Non steroidal glucocorticoid receptor modulators

Publications (1)

Publication Number Publication Date
PL1853601T3 true PL1853601T3 (pl) 2009-07-31

Family

ID=34938730

Family Applications (1)

Application Number Title Priority Date Filing Date
PL06708243T PL1853601T3 (pl) 2005-02-14 2006-02-14 Niesteroidowe modulatory receptora glukokortykoidowego

Country Status (30)

Country Link
US (1) US8133885B2 (pl)
EP (1) EP1853601B1 (pl)
JP (1) JP4922950B2 (pl)
KR (1) KR101285454B1 (pl)
CN (1) CN101119995B (pl)
AR (1) AR054329A1 (pl)
AT (1) ATE422497T1 (pl)
AU (1) AU2006212192B2 (pl)
BR (1) BRPI0607341A2 (pl)
CA (1) CA2597748C (pl)
CY (1) CY1109038T1 (pl)
DE (1) DE602006005138D1 (pl)
DK (1) DK1853601T3 (pl)
ES (1) ES2321227T3 (pl)
HR (1) HRP20090161T1 (pl)
IL (1) IL184374A (pl)
MX (1) MX2007008786A (pl)
MY (1) MY147632A (pl)
NO (1) NO20073702L (pl)
NZ (1) NZ556469A (pl)
PE (1) PE20061037A1 (pl)
PL (1) PL1853601T3 (pl)
PT (1) PT1853601E (pl)
RS (1) RS50778B (pl)
RU (1) RU2409577C2 (pl)
SI (1) SI1853601T1 (pl)
TW (1) TWI370129B (pl)
UA (1) UA91352C2 (pl)
WO (1) WO2006084917A1 (pl)
ZA (1) ZA200705899B (pl)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI297685B (en) 2002-04-04 2008-06-11 Organon Nv Non-steroidal progesterone receptor modulators
RS51970B (en) 2007-02-02 2012-02-29 Pfizer Products Inc. TRICYCLIC UNITS AND THEIR USE AS MODULATORS OF GLUCOCORTICOID RECEPTORS
TW200914029A (en) * 2007-05-07 2009-04-01 Organon Nv New progesterone receptor modulators
US8063037B2 (en) 2007-05-07 2011-11-22 N. V. Organon Progesterone receptor modulators
EP3607942A1 (en) 2008-11-07 2020-02-12 University of Sheffield Medicament and method of diagnosis
WO2017046096A1 (en) * 2015-09-15 2017-03-23 Leo Pharma A/S Non-steroidal glucocorticoid receptor modulators for local drug delivery

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4054572A (en) * 1973-04-26 1977-10-18 Akzona Incorporated Hexahydro pyridine [1,2d] dibenza [b,f] (1,4)-diazepines
TWI297685B (en) * 2002-04-04 2008-06-11 Organon Nv Non-steroidal progesterone receptor modulators
US7074806B2 (en) 2002-06-06 2006-07-11 Boehringer Ingelheim Pharmaceuticals, Inc. Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof

Also Published As

Publication number Publication date
ATE422497T1 (de) 2009-02-15
SI1853601T1 (sl) 2009-06-30
ES2321227T3 (es) 2009-06-03
JP4922950B2 (ja) 2012-04-25
TWI370129B (en) 2012-08-11
MY147632A (en) 2012-12-31
IL184374A (en) 2012-02-29
CY1109038T1 (el) 2014-07-02
WO2006084917A1 (en) 2006-08-17
DE602006005138D1 (de) 2009-03-26
IL184374A0 (en) 2007-10-31
MX2007008786A (es) 2007-08-03
RU2409577C2 (ru) 2011-01-20
CN101119995A (zh) 2008-02-06
CA2597748C (en) 2013-09-24
EP1853601B1 (en) 2009-02-11
KR101285454B1 (ko) 2013-07-15
RS50778B (sr) 2010-08-31
US20090062262A1 (en) 2009-03-05
AR054329A1 (es) 2007-06-20
DK1853601T3 (da) 2009-05-18
PE20061037A1 (es) 2006-10-26
PT1853601E (pt) 2009-04-09
BRPI0607341A2 (pt) 2010-03-23
RU2007134226A (ru) 2009-03-20
CN101119995B (zh) 2012-01-25
ZA200705899B (en) 2008-07-30
CA2597748A1 (en) 2006-08-17
HRP20090161T1 (en) 2009-05-31
EP1853601A1 (en) 2007-11-14
JP2008530056A (ja) 2008-08-07
US8133885B2 (en) 2012-03-13
NO20073702L (no) 2007-09-28
AU2006212192A1 (en) 2006-08-17
KR20070107750A (ko) 2007-11-07
NZ556469A (en) 2009-08-28
TW200640923A (en) 2006-12-01
AU2006212192B2 (en) 2011-06-16
UA91352C2 (en) 2010-07-26

Similar Documents

Publication Publication Date Title
IL190281A0 (en) Modulation of glucocorticoid receptor expression
IL183543A0 (en) Estrogen receptor modulators
IL182829A0 (en) Estrogen receptor modulators
EP2179061A4 (en) GREAT LIKE RECEPTOR MODULATORS
ZA200807551B (en) Selective androgen receptor modulators
GB0400440D0 (en) Receptor modulators
IL180955A0 (en) Progesterone receptor modulators comprising pyrrole- oxindole derivatives and uses thereof
IL191710A0 (en) Glucocorticoid receptor modulators as antiinflammatory agents
IL176935A0 (en) Androgen receptor modulators
HK1131396A1 (en) 11-phosphorous steroid derivatives useful as progesterone receptor modulators
IL184374A0 (en) Non steroidal glucocorticoid receptor modulators
ZA200804871B (en) Estrogen modulators
IL188314A0 (en) Cyanopyrrole-sulfonamide progesterone receptor modulators and uses thereof
EP1784187A4 (en) MODULATORS OF THE ANDROGEN RECEPTOR
EP1945213A4 (en) MODULATORS OF THE R3-PIPERIDINE-4-YL-INDOLE ORL-1 RECEPTOR
ZA200800690B (en) Non-steroidal progesterone receptor modulators
HK1144287A1 (en) Steroids derivatives as selective progesterone receptor modulators
HK1126767A1 (en) Pyridooxazepine progesteron receptor modulators
ZA200806237B (en) Cannibinoid receptor modulators
AP2008004481A0 (en) Estrogen modulators
HK1096405A1 (en) Progesterone receptor modulators
ZA200907546B (en) New progesterone receptor modulators
HK1131787A1 (en) Oxa-steroids derivatives as selective progesterone receptor modulators