PL1844036T3 - Sposób otrzymywania arypiprazolu - Google Patents

Sposób otrzymywania arypiprazolu

Info

Publication number
PL1844036T3
PL1844036T3 PL06704096T PL06704096T PL1844036T3 PL 1844036 T3 PL1844036 T3 PL 1844036T3 PL 06704096 T PL06704096 T PL 06704096T PL 06704096 T PL06704096 T PL 06704096T PL 1844036 T3 PL1844036 T3 PL 1844036T3
Authority
PL
Poland
Prior art keywords
aripiprazole
preparation
Prior art date
Application number
PL06704096T
Other languages
English (en)
Inventor
Johannes Ludescher
Hubert Sturm
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP05001639A external-priority patent/EP1686126A1/en
Priority claimed from EP05001638A external-priority patent/EP1686117A1/en
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of PL1844036T3 publication Critical patent/PL1844036T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • C07D215/22—Oxygen atoms attached in position 2 or 4
    • C07D215/227—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
PL06704096T 2005-01-27 2006-01-27 Sposób otrzymywania arypiprazolu PL1844036T3 (pl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP05001639A EP1686126A1 (en) 2005-01-27 2005-01-27 Salts of aripiprazole
EP05001638A EP1686117A1 (en) 2005-01-27 2005-01-27 Polymorph and solvates of aripiprazole
EP06704096.4A EP1844036B1 (en) 2005-01-27 2006-01-27 Process for the preparation of aripiprazole
PCT/EP2006/000726 WO2006079549A1 (en) 2005-01-27 2006-01-27 Salts of aripiprazole

Publications (1)

Publication Number Publication Date
PL1844036T3 true PL1844036T3 (pl) 2016-02-29

Family

ID=36218176

Family Applications (1)

Application Number Title Priority Date Filing Date
PL06704096T PL1844036T3 (pl) 2005-01-27 2006-01-27 Sposób otrzymywania arypiprazolu

Country Status (10)

Country Link
US (1) US7884205B2 (pl)
EP (3) EP2093217B1 (pl)
JP (1) JP5426828B2 (pl)
CN (1) CN101107242B (pl)
AU (2) AU2006208628B2 (pl)
CA (1) CA2594690C (pl)
ES (1) ES2550359T3 (pl)
PL (1) PL1844036T3 (pl)
SI (1) SI1844036T1 (pl)
WO (1) WO2006079549A1 (pl)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7714129B2 (en) 2003-12-16 2010-05-11 Teva Pharmaceutical Industries Ltd. Methods of preparing anhydrous aripiprazole form II
EP1686117A1 (en) * 2005-01-27 2006-08-02 Sandoz AG Polymorph and solvates of aripiprazole
CZ300352B6 (cs) * 2005-02-15 2009-04-29 Zentiva, A. S. Zpusob prípravy fosforecnanu aripiprazolu
CZ300456B6 (cs) * 2005-02-15 2009-05-27 Zentiva, A. S. Zpusob prípravy vinanu aripiprazolu v krystalické forme
HUP0500683A3 (en) * 2005-07-14 2009-03-30 Egis Gyogyszergyar Nyilvanosan New arylpiprazole salts for producing pharmaceutical composition
US20060223820A1 (en) * 2006-03-21 2006-10-05 Chemagis Ltd. Crystalline aripiprazole salts and processes for preparation and purification thereof
EP1880714A1 (en) * 2006-07-20 2008-01-23 Helm AG Amorphous Aripiprazole and Process for the Preparation thereof
US7799790B2 (en) 2006-07-20 2010-09-21 Helm Ag Amorphous aripiprazole and process for the preparation thereof
WO2008026220A1 (en) * 2006-08-28 2008-03-06 Lupin Limited A process for purification of 7-(4-bromobutoxy)-3,4 dihydrocarbostyril, an intermediate for manufacture of aripirazole
EP2233471A1 (en) * 2009-02-06 2010-09-29 Adamed Sp. z o.o. A salt of 7-{4-[4-(2,3-dichlorophenyl)-1-piperazinyl]butoxy}-3,4.dihydro-2(1h)-quinolinone with 5-sulfosalicylic acid and its preparation process
JP5664871B2 (ja) * 2009-06-19 2015-02-04 株式会社 メドレックス アリピプラゾールと有機酸を有効成分とする外用剤組成物
CN102106826B (zh) * 2009-12-29 2013-06-05 上海中西制药有限公司 一种阿立哌唑固体制剂及其制备方法
CN102863377A (zh) * 2012-08-17 2013-01-09 南京正大天晴制药有限公司 一种制备高纯度阿立哌唑的方法
CN108069900B (zh) * 2016-11-08 2022-09-23 齐鲁制药有限公司 阿立哌唑盐酸盐的制备方法和用途
CN111909086B (zh) * 2020-05-05 2022-05-20 天津大学 阿立哌唑-乙酰水杨酸盐及制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS54130587A (en) 1978-03-30 1979-10-09 Otsuka Pharmaceut Co Ltd Carbostyryl derivative
US5006528A (en) * 1988-10-31 1991-04-09 Otsuka Pharmaceutical Co., Ltd. Carbostyril derivatives
JP2608788B2 (ja) * 1988-10-31 1997-05-14 大塚製薬 株式会社 精神分裂病治療剤
AR033485A1 (es) 2001-09-25 2003-12-26 Otsuka Pharma Co Ltd Sustancia medicinal de aripiprazol de baja higroscopicidad y proceso para la preparacion de la misma
WO2004083183A1 (en) * 2003-03-21 2004-09-30 Hetero Drugs Limited Novel crystalline forms of aripiprazole
EP1618103A2 (en) 2003-04-25 2006-01-25 Cadila Healthcare Ltd. Polymorphs of aripiprazole
CA2428237C (en) * 2003-05-08 2010-07-20 Delmar Chemicals Inc. Process for the preparation of carbostyril derivatives
WO2005009990A1 (en) * 2003-07-25 2005-02-03 Hetero Drugs Limited Aripiprazole crystalline forms
WO2006030446A1 (en) 2004-09-13 2006-03-23 Matrix Laboratories Ltd Process for the preparation of polymorphs, solvates of aripiprazole using aripiprazole acid salts

Also Published As

Publication number Publication date
CA2594690A1 (en) 2006-08-03
WO2006079549A1 (en) 2006-08-03
CA2594690C (en) 2013-08-27
SI1844036T1 (sl) 2015-12-31
JP2008536798A (ja) 2008-09-11
US7884205B2 (en) 2011-02-08
ES2550359T3 (es) 2015-11-06
EP2093217B1 (en) 2014-03-12
EP1844036B1 (en) 2015-09-23
CN101107242B (zh) 2011-08-10
CN101107242A (zh) 2008-01-16
EP1844016A1 (en) 2007-10-17
EP1844036A1 (en) 2007-10-17
JP5426828B2 (ja) 2014-02-26
AU2010241386B2 (en) 2013-07-11
US20080287677A1 (en) 2008-11-20
AU2006208628B2 (en) 2010-08-12
AU2010241386B9 (en) 2013-07-25
AU2006208628A1 (en) 2006-08-03
AU2010241386A1 (en) 2010-12-02
EP2093217A1 (en) 2009-08-26

Similar Documents

Publication Publication Date Title
PL1844036T3 (pl) Sposób otrzymywania arypiprazolu
IL188330A0 (en) Processes for the preparation of
DK3872059T3 (en) Process for the preparation of 2,3,3,3 tetrahydrofluoropropene
PT2308825E (pt) Processo para a preparação de um intermediário para a azoxistrobina
EP1893570A4 (en) IMPROVED PROCESS FOR THE PREPARATION OF EZETIMIBE
ZA200903533B (en) Process for the preparation of rosuvastatin
EP1940793A4 (en) METHOD FOR PRODUCING MONTELUCASTS
ZA200804264B (en) Process for the preparation of ferri-succinylcasein
SI2093217T1 (sl) Postopek za pripravo oblike X aripiprazola
EG25547A (en) Process for the preparation of amines
ZA200601910B (en) Process for the preparation of organosilances
IL184715A0 (en) Process for the preparation of intermediates
EP2024369A4 (en) NEW PROCESS FOR THE PREPARATION OF SILDENAFIL CITRATE
IL213474A0 (en) Processes for the preparation of cyclopropyl-amide derivatives
TWI365869B (en) Process for the preparation of phenol
EP1996192A4 (en) PROCESS FOR PREPARING 3,4-SUBSTITUTED THIAZOLIDIN-2-ONES IN 3,4
EP1917231A4 (en) PROCESS FOR THE PREPARATION OF BROMOPICRIN
HUP0401379A3 (en) Process for the preparation of risperidon
IL178960A0 (en) Process for the preparation of pyridin-2-ylmethylsulphinyl-1h-benzimidazol compounds
HU0500570D0 (en) Process for the preparation of (s)-(-)-amlodipine
EP1915380A4 (en) PROCESS FOR THE SYNTHESIS OF N, N'-DISUBSTITUTED OXABISPIDINES
HUP0501046A2 (en) Process for the preparation of olanzapine
HU0500126D0 (en) New compounds and process for their preparation
SI1732916T1 (sl) Postopek za pripravo alkoksikarbonilmetoksi-ciklopentanov
HK1112242A1 (en) Process for the preparation of precursors of 5-alkylthioalkylamino-1- phenyl-pyrazoles 5-