PH19622A - Spiro-3-hetero-azolones and pharmaceutical composition conaining same - Google Patents

Spiro-3-hetero-azolones and pharmaceutical composition conaining same

Info

Publication number
PH19622A
PH19622A PH29927A PH29927A PH19622A PH 19622 A PH19622 A PH 19622A PH 29927 A PH29927 A PH 29927A PH 29927 A PH29927 A PH 29927A PH 19622 A PH19622 A PH 19622A
Authority
PH
Philippines
Prior art keywords
azolones
conaining
spiro
hetero
same
Prior art date
Application number
PH29927A
Other languages
English (en)
Inventor
Christopher Andrew Lipinski
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of PH19622A publication Critical patent/PH19622A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
PH29927A 1982-12-06 1983-12-05 Spiro-3-hetero-azolones and pharmaceutical composition conaining same PH19622A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US44733782A 1982-12-06 1982-12-06
US06/545,450 US4556670A (en) 1982-12-06 1983-10-28 Spiro-3-hetero-azolones for treatment of diabetic complications

Publications (1)

Publication Number Publication Date
PH19622A true PH19622A (en) 1986-05-30

Family

ID=27034944

Family Applications (1)

Application Number Title Priority Date Filing Date
PH29927A PH19622A (en) 1982-12-06 1983-12-05 Spiro-3-hetero-azolones and pharmaceutical composition conaining same

Country Status (21)

Country Link
US (1) US4556670A (fr)
EP (1) EP0115133B1 (fr)
KR (1) KR860001581B1 (fr)
AU (1) AU545409B2 (fr)
BG (1) BG44708A3 (fr)
CA (1) CA1204763A (fr)
DD (1) DD219482A5 (fr)
DE (1) DE3379043D1 (fr)
DK (1) DK558283A (fr)
ES (1) ES527780A0 (fr)
FI (1) FI80267C (fr)
GR (1) GR78787B (fr)
IE (1) IE56345B1 (fr)
IL (1) IL70379A (fr)
NO (1) NO160001C (fr)
NZ (1) NZ206484A (fr)
PH (1) PH19622A (fr)
PL (1) PL142143B1 (fr)
PT (1) PT77760B (fr)
RO (1) RO88202B (fr)
YU (1) YU43557B (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0159143B1 (fr) * 1984-03-23 1987-12-16 Pfizer Inc. Spiro-indènes et spiro-dihydro-1,2-naphtalènes pour le traitement de complications diabétiques
US4575507A (en) 1985-05-29 1986-03-11 Pfizer Inc. Spiro-imidazolidines as aldose reductase inhibitors and their pharmaceutical use
GB8601100D0 (en) * 1986-01-17 1986-02-19 Cosmas Damian Ltd Drug delivery system
GB2355264A (en) 1999-09-30 2001-04-18 Merck & Co Inc Spirohydantoin derivatives useful as alpha 1a adrenoceptor antagonists
JP2005523314A (ja) 2002-04-18 2005-08-04 ユニバーシティ オブ バージニア パテント ファウンデーション 新規ナトリウムチャンネル遮断化合物
WO2004050039A2 (fr) * 2002-12-04 2004-06-17 Merck & Co., Inc. Urees spirocycliques, compositions les contenant et procedes d'utilisation
JO3501B1 (ar) * 2014-12-22 2020-07-05 Servier Lab مشتقات 5-{(بيبرازين - 1-يل)-3-أوكسو - بروبيل}- إيميدازوليدين-2، 4 - دايون كمثبطات ل adamts لمعالجة هشاشة العظام)

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2872454A (en) * 1959-02-03 Spiro-hydantoins from x-chloro-
GB796069A (en) * 1955-12-23 1958-06-04 Ici Ltd Substituted hydantoins
GB818724A (en) * 1956-10-18 1959-08-19 Ici Ltd Hydantoin derivatives
US3532744A (en) * 1967-07-28 1970-10-06 American Home Prod 1- and 2-amino substituted indane and tetralene carboxylic acids
US3985888A (en) * 1969-07-24 1976-10-12 Richardson-Merrell Inc. Methods of inducing sedation using certain spiroalkanone-imides
US3821383A (en) * 1972-07-10 1974-06-28 Ayerst Mckenna & Harrison Compositions for and a method of treating diabetic complications
US4117230A (en) * 1976-10-18 1978-09-26 Pfizer Inc. Hydantoin derivatives as therapeutic agents
US4130714A (en) * 1977-05-23 1978-12-19 Pfizer Inc. Hydantoin therapeutic agents
US4200642A (en) * 1978-08-21 1980-04-29 Pfizer Inc. Spiro-oxazolidindiones
US4181729A (en) * 1979-03-21 1980-01-01 Pfizer Inc. Phenyl or phenoxy substituted spiro-imidazolidinedione derivatives
US4226875A (en) * 1979-04-02 1980-10-07 Pfizer Inc. Novel spiro-oxazolidinediones
US4307108A (en) * 1979-12-26 1981-12-22 Pfizer Inc. Method for lowering sorbitol levels using spiro-imides
US4248882A (en) * 1980-02-12 1981-02-03 Pfizer Inc. Treating diabetes-associated complications with hydantoin amines
JPS5745185A (en) * 1980-07-21 1982-03-13 Eisai Co Ltd Hydantoin derivative and its preparation

Also Published As

Publication number Publication date
CA1204763A (fr) 1986-05-20
KR860001581B1 (ko) 1986-10-10
PT77760B (en) 1986-05-30
PT77760A (en) 1983-12-01
IL70379A (en) 1988-10-31
IE832854L (en) 1984-06-06
BG44708A3 (fr) 1989-01-16
NO834437L (no) 1984-06-07
YU43557B (en) 1989-08-31
DE3379043D1 (en) 1989-03-02
RO88202B (ro) 1985-12-31
IL70379A0 (en) 1984-03-30
FI80267C (fi) 1990-05-10
NO160001B (no) 1988-11-21
EP0115133A1 (fr) 1984-08-08
NO160001C (no) 1989-03-01
FI834457A0 (fi) 1983-12-05
IE56345B1 (en) 1991-07-03
DD219482A5 (de) 1985-03-06
NZ206484A (en) 1987-07-31
AU2196883A (en) 1984-06-14
GR78787B (fr) 1984-10-02
EP0115133B1 (fr) 1989-01-25
YU237183A (en) 1986-02-28
PL244966A1 (en) 1985-05-21
RO88202A (fr) 1985-12-30
US4556670A (en) 1985-12-03
FI834457A (fi) 1984-06-07
DK558283A (da) 1984-07-11
DK558283D0 (da) 1983-12-05
FI80267B (fi) 1990-01-31
ES8601912A1 (es) 1985-11-16
AU545409B2 (en) 1985-07-11
KR840006975A (ko) 1984-12-04
ES527780A0 (es) 1985-11-16
PL142143B1 (en) 1987-09-30

Similar Documents

Publication Publication Date Title
DE3372705D1 (en) Pharmaceutical composition and its use
DE3376957D1 (en) Pharmaceutical gel composition
PH22863A (en) Pyrrolobenzimidazoles and pharmaceutical composition containing them
EP0138029A3 (en) Pharmaceutical composition
ZA834074B (en) Pharmaceutical composition
PH19849A (en) Steroids and their pharmaceutical composition
GB8314419D0 (en) Polyprenyl compound and pharmaceutical composition
EP0093551A3 (en) Pharmaceutical composition
PH17562A (en) 2-guanidino-4-heteroarylthiazoles and pharmaceutical compositions
PH20168A (en) 7-carboxymethoxyphenylacetamino-3-cephem derivatives and their pharmaceutical compositions
DE3373623D1 (en) Pharmaceutical combination composition and associated method
NZ209095A (en) Piperidinoquinazolines and pharmaceutical compositions
DE3367089D1 (en) 3-phenoxy-1-azetidinecarboxamides and their use and preparation
NZ208244A (en) Phenyl-pyrazol-3-ones and pharmaceutical compositions
PH19622A (en) Spiro-3-hetero-azolones and pharmaceutical composition conaining same
GB8329700D0 (en) Anti-haemophilic pharmaceutical composition
ZA845299B (en) Pharmaceutical compounds and their preparation
NZ205732A (en) Thiatriazine derivatives and pharmaceutical compositions
GB2117757B (en) Alkylspectinomycins and their preparation
PH19896A (en) 4-phenyl-tetrahydro-furano-pyridine and pharmaceutical compositions containing them
GB8328896D0 (en) Pharmaceutical composition
NZ203649A (en) 2-beta-d-ribofuranosylselenazole-4-carboxamide derivatives and pharmaceutical compositions
IL68668A0 (en) Piperidinoquinazolines and pharmaceutical compositions containing them
ZA832811B (en) Azabicyclobenzamides their preparation and their pharmaceutical compositions
ZA834539B (en) Pharmaceutical composition and its preparation and use