PE20170447A1 - Metodo para la preparacion de imidazopiridazinas sustituidas - Google Patents
Metodo para la preparacion de imidazopiridazinas sustituidasInfo
- Publication number
- PE20170447A1 PE20170447A1 PE2017000372A PE2017000372A PE20170447A1 PE 20170447 A1 PE20170447 A1 PE 20170447A1 PE 2017000372 A PE2017000372 A PE 2017000372A PE 2017000372 A PE2017000372 A PE 2017000372A PE 20170447 A1 PE20170447 A1 PE 20170447A1
- Authority
- PE
- Peru
- Prior art keywords
- compound
- formula
- preparation
- reacting
- obtaining
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B41/00—Formation or introduction of functional groups containing oxygen
- C07B41/02—Formation or introduction of functional groups containing oxygen of hydroxy or O-metal groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epidemiology (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
SE REFIERE A UN METODO DE PREPARACION DEL COMPUESTO DE FORMULA (I) QUE COMPRENDE: A) HACER REACCIONAR UN COMPUESTO DE FORMULA (II) CON UN COMPUESTO DE FORMULA R1-OH OBTENIENDOSE EL COMPUESTO DE FORMULA (IV); B) HACER REACCIONAR EL COMPUESTO DE FORMULA (IV) CON UN COMPUESTO DE FORMULA R2-Y OBTENIENDOSE EL COMPUESTO DE FORMULA (VI); C) HACER REACCIONAR EL COMPUESTO DE FORMULA (VI) CON UN COMPUESTO DE FORMULA (VII) OBTENIENDOSE EL COMPUESTO DE FORMULA (I); DONDE LG1 ES BROMO; LG2 ES CLORO; LG3 ES IODO; R1 ES FENILO O HETEROARILO OPCIONALMENTE SUSTITUIDOS; R2 ES FENILO OPCIONALMENTE SUSTITUIDO; R3a ES ALQUILO C1-C6 OPCIONALMENTE SUSTITUIDO; R3b ES H O ALQUILO C1-C6 OPCIONALMENTE SUSTITUIDO
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14183029 | 2014-09-01 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PE20170447A1 true PE20170447A1 (es) | 2017-05-18 |
Family
ID=51422014
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PE2017000372A PE20170447A1 (es) | 2014-09-01 | 2015-08-28 | Metodo para la preparacion de imidazopiridazinas sustituidas |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US20170305912A1 (es) |
| EP (1) | EP3189055A1 (es) |
| JP (1) | JP2017525725A (es) |
| KR (1) | KR20170044166A (es) |
| CN (1) | CN106795164A (es) |
| AR (1) | AR101730A1 (es) |
| AU (1) | AU2015311011A1 (es) |
| BR (1) | BR112017003916A2 (es) |
| CA (1) | CA2959224A1 (es) |
| CO (1) | CO2017002070A2 (es) |
| IL (1) | IL250264A0 (es) |
| MX (1) | MX2017002749A (es) |
| PE (1) | PE20170447A1 (es) |
| RU (1) | RU2017110880A (es) |
| SG (1) | SG11201700818XA (es) |
| TW (1) | TW201613927A (es) |
| UY (1) | UY36284A (es) |
| WO (1) | WO2016034507A1 (es) |
| ZA (1) | ZA201702297B (es) |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20070078136A1 (en) | 2005-09-22 | 2007-04-05 | Bristol-Myers Squibb Company | Fused heterocyclic compounds useful as kinase modulators |
| TW201107329A (en) * | 2009-07-30 | 2011-03-01 | Oncotherapy Science Inc | Fused imidazole derivative having ttk inhibitory action |
| TWI541243B (zh) * | 2010-09-10 | 2016-07-11 | 拜耳知識產權公司 | 經取代咪唑并嗒 |
| WO2014020041A1 (en) * | 2012-08-02 | 2014-02-06 | Bayer Pharma Aktiengesellschaft | Combinations for the treatment of cancer |
| WO2014080633A1 (en) | 2012-11-21 | 2014-05-30 | Raqualia Pharma Inc. | Polymorph forms |
| TW201437211A (zh) | 2013-03-01 | 2014-10-01 | Bayer Pharma AG | 經取代咪唑并嗒□ |
| MX2015017245A (es) * | 2013-06-13 | 2016-07-20 | Bayer Pharma AG | Combinacion de un derivado de imidazopiridazina y un agente mitotico para el tratamiento del cancer. |
-
2015
- 2015-08-07 TW TW104125835A patent/TW201613927A/zh unknown
- 2015-08-28 CN CN201580046909.3A patent/CN106795164A/zh active Pending
- 2015-08-28 WO PCT/EP2015/069739 patent/WO2016034507A1/en active Application Filing
- 2015-08-28 AU AU2015311011A patent/AU2015311011A1/en not_active Abandoned
- 2015-08-28 PE PE2017000372A patent/PE20170447A1/es not_active Application Discontinuation
- 2015-08-28 JP JP2017511580A patent/JP2017525725A/ja active Pending
- 2015-08-28 BR BR112017003916-8A patent/BR112017003916A2/pt not_active Application Discontinuation
- 2015-08-28 EP EP15756401.4A patent/EP3189055A1/en not_active Withdrawn
- 2015-08-28 SG SG11201700818XA patent/SG11201700818XA/en unknown
- 2015-08-28 CA CA2959224A patent/CA2959224A1/en not_active Abandoned
- 2015-08-28 RU RU2017110880A patent/RU2017110880A/ru unknown
- 2015-08-28 MX MX2017002749A patent/MX2017002749A/es unknown
- 2015-08-28 US US15/507,716 patent/US20170305912A1/en not_active Abandoned
- 2015-08-28 KR KR1020177007529A patent/KR20170044166A/ko unknown
- 2015-08-31 UY UY0001036284A patent/UY36284A/es not_active Application Discontinuation
- 2015-09-01 AR ARP150102792A patent/AR101730A1/es unknown
-
2017
- 2017-01-24 IL IL250264A patent/IL250264A0/en unknown
- 2017-03-01 CO CONC2017/0002070A patent/CO2017002070A2/es unknown
- 2017-03-31 ZA ZA2017/02297A patent/ZA201702297B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| SG11201700818XA (en) | 2017-03-30 |
| ZA201702297B (en) | 2018-12-19 |
| EP3189055A1 (en) | 2017-07-12 |
| RU2017110880A (ru) | 2018-10-03 |
| US20170305912A1 (en) | 2017-10-26 |
| KR20170044166A (ko) | 2017-04-24 |
| AU2015311011A1 (en) | 2017-02-23 |
| AR101730A1 (es) | 2017-01-11 |
| TW201613927A (en) | 2016-04-16 |
| MX2017002749A (es) | 2017-07-26 |
| CO2017002070A2 (es) | 2017-05-19 |
| CN106795164A (zh) | 2017-05-31 |
| WO2016034507A1 (en) | 2016-03-10 |
| CA2959224A1 (en) | 2016-03-10 |
| JP2017525725A (ja) | 2017-09-07 |
| BR112017003916A2 (pt) | 2018-03-06 |
| IL250264A0 (en) | 2017-03-30 |
| UY36284A (es) | 2016-04-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD | Application declared void or lapsed |