PE20080887A1 - Composiciones de carbamatos de fenilalquilo - Google Patents
Composiciones de carbamatos de fenilalquiloInfo
- Publication number
- PE20080887A1 PE20080887A1 PE2007001383A PE2007001383A PE20080887A1 PE 20080887 A1 PE20080887 A1 PE 20080887A1 PE 2007001383 A PE2007001383 A PE 2007001383A PE 2007001383 A PE2007001383 A PE 2007001383A PE 20080887 A1 PE20080887 A1 PE 20080887A1
- Authority
- PE
- Peru
- Prior art keywords
- composition
- phenylalkyl carbamate
- refers
- found
- phenyl
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/325—Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A61P25/10—Antiepileptics; Anticonvulsants for petit-mal
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A61P25/12—Antiepileptics; Anticonvulsants for grand-mal
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Epidemiology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Inorganic Chemistry (AREA)
- Physical Education & Sports Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
SE REFIERE A UNA COMPOSICION FARMACEUTICA QUE COMPRENDE: A) UN COMPUESTO CARBAMATO DE FENILALQUILO DE FORMULA (I) DONDE X ES HALOGENO, R1 Y R2 SON CADA UNO H O ALQUILO(C1-C4) OPCIONALMENTE SUSTITUIDO CON FENILO, SIENDO UN COMPUESTO PREFERIDO 2-(2-CLORO-FENIL)-2-HIDROXI-ETIL ESTER DEL ACIDO CARBAMICO Y SE ENCUENTRA EN UNA CANTIDAD DE 75% A 99% DE LA COMPOSICION; B) FOSFATO DE CALCIO DIBASICO DIHIDRATADO QUE REDUCE LA DEGRADACION DEL COMPUESTO CARBAMATO DE FENILALQUILO, PRESENTA UN pH DE 5,0 A 5,8 Y SE ENCUENTRA EN UNA CANTIDAD DE 4% A 40% DE LA COMPOSICION; C) OTROS EXCIPIENTES TALES COMO CELULOSA MICROCRISTALINA, LACTOSA, MANITOL, POLIETILENGLICOL, ESTEARATO DE MAGNESIO, ENTRE OTROS. SE REFIERE TAMBIEN A UN PROCEDIMIENTO DE PREPARACION DE LA COMPOSICION. DICHA COMPOSICION ES UTIL EN EL TRATAMIENTO DE EPILEPSIA, ESPASMO MUSCULAR, ACCIDENTE CEREBROVASCULAR
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US82935506P | 2006-10-13 | 2006-10-13 |
Publications (1)
Publication Number | Publication Date |
---|---|
PE20080887A1 true PE20080887A1 (es) | 2008-06-28 |
Family
ID=39111848
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PE2007001383A PE20080887A1 (es) | 2006-10-13 | 2007-10-12 | Composiciones de carbamatos de fenilalquilo |
Country Status (23)
Country | Link |
---|---|
US (1) | US20080090903A1 (es) |
EP (1) | EP2089002A1 (es) |
JP (1) | JP2010506846A (es) |
KR (1) | KR20090067210A (es) |
CN (1) | CN101663026A (es) |
AR (1) | AR063294A1 (es) |
AU (1) | AU2007313018A1 (es) |
BR (1) | BRPI0719236A2 (es) |
CA (1) | CA2673526A1 (es) |
CL (1) | CL2007002943A1 (es) |
CO (1) | CO6190539A2 (es) |
CR (1) | CR10793A (es) |
EA (1) | EA200970378A1 (es) |
IL (1) | IL198144A0 (es) |
MX (1) | MX2009003929A (es) |
NI (1) | NI200900055A (es) |
NO (1) | NO20091492L (es) |
PE (1) | PE20080887A1 (es) |
SV (1) | SV2009003222A (es) |
TW (1) | TW200831134A (es) |
UY (1) | UY30643A1 (es) |
WO (1) | WO2008048802A1 (es) |
ZA (1) | ZA200903284B (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8263652B2 (en) * | 2007-10-31 | 2012-09-11 | Sk Biopharmaceuticals Co., Ltd. | Stabilized pediatric suspension of carisbamate |
US9018253B2 (en) | 2010-07-02 | 2015-04-28 | Bio-Pharm Solutions Co., Ltd. | Phenylcarbamate compound and muscle relaxant containing the same |
BR112013000050B1 (pt) * | 2010-07-02 | 2021-10-19 | Bio-Pharm Solutions Co., Ltd | Compostos de carbamato de fenila e composição farmacêutica |
US8609849B1 (en) | 2010-11-30 | 2013-12-17 | Fox Chase Chemical Diversity Center, Inc. | Hydroxylated sulfamides exhibiting neuroprotective action and their method of use |
CN104870421A (zh) | 2011-12-27 | 2015-08-26 | 比皮艾思药物研发有限公司 | 用于预防或治疗als的苯基氨基甲酸酯化合物 |
WO2014097137A2 (en) * | 2012-12-18 | 2014-06-26 | Mahesh Kandula | Compositions and methods for the treatment of seizures and neurologic diseases |
KR101717872B1 (ko) * | 2013-03-12 | 2017-03-17 | (주)바이오팜솔루션즈 | 소아 간질 및 간질-관련 증후군의 예방 또는 치료용 페닐카바메이트 화합물 |
CN105209430B (zh) * | 2013-03-12 | 2019-09-13 | 比皮艾思药物研发有限公司 | 苯基氨基甲酸酯化合物及包含其的神经保护组合物 |
KR102213484B1 (ko) * | 2016-02-29 | 2021-02-08 | (주)바이오팜솔루션즈 | 카바메이트 유도체 화합물, 이의 제조 방법 및 용도 |
KR102121680B1 (ko) * | 2016-02-29 | 2020-06-10 | (주)바이오팜솔루션즈 | 설파메이트 유도체 화합물, 이의 제조 방법 및 용도 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3265728A (en) * | 1962-07-18 | 1966-08-09 | Armour Pharma | Substituted phenethyl carbamates |
US5698588A (en) * | 1996-01-16 | 1997-12-16 | Yukong Limited | Halogen substituted carbamate compounds from 2-phenyl-1,2-ethanediol |
US20010034365A1 (en) * | 1996-01-16 | 2001-10-25 | Choi Yong Moon | Halogen substituted carbamate compounds from 2-phenyl-1,2-ethanediol |
FR2758459B1 (fr) * | 1997-01-17 | 1999-05-07 | Pharma Pass | Composition pharmaceutique de fenofibrate presentant une biodisponibilite elevee et son procede de preparation |
US20020147229A1 (en) * | 2000-08-17 | 2002-10-10 | Allerton Charlotte Moira Norfor | Pharmaceuticals |
BR0213634A (pt) * | 2001-10-08 | 2004-11-30 | Sun Pharmaceutical Ind Ltd | Sistema de liberação de droga com ação retardada para um agente antiespasmódico |
-
2007
- 2007-10-08 EA EA200970378A patent/EA200970378A1/ru unknown
- 2007-10-08 EP EP07843959A patent/EP2089002A1/en not_active Withdrawn
- 2007-10-08 JP JP2009532515A patent/JP2010506846A/ja active Pending
- 2007-10-08 CA CA002673526A patent/CA2673526A1/en not_active Abandoned
- 2007-10-08 US US11/868,588 patent/US20080090903A1/en not_active Abandoned
- 2007-10-08 MX MX2009003929A patent/MX2009003929A/es unknown
- 2007-10-08 BR BRPI0719236-3A patent/BRPI0719236A2/pt not_active IP Right Cessation
- 2007-10-08 CN CN200780045911A patent/CN101663026A/zh active Pending
- 2007-10-08 KR KR1020097009746A patent/KR20090067210A/ko not_active Application Discontinuation
- 2007-10-08 AU AU2007313018A patent/AU2007313018A1/en not_active Abandoned
- 2007-10-08 WO PCT/US2007/080677 patent/WO2008048802A1/en active Application Filing
- 2007-10-12 PE PE2007001383A patent/PE20080887A1/es not_active Application Discontinuation
- 2007-10-12 TW TW096138084A patent/TW200831134A/zh unknown
- 2007-10-12 AR ARP070104554A patent/AR063294A1/es not_active Application Discontinuation
- 2007-10-12 UY UY30643A patent/UY30643A1/es unknown
- 2007-10-12 CL CL200702943A patent/CL2007002943A1/es unknown
-
2009
- 2009-04-13 NI NI200900055A patent/NI200900055A/es unknown
- 2009-04-14 SV SV2009003222A patent/SV2009003222A/es unknown
- 2009-04-14 CO CO09037411A patent/CO6190539A2/es not_active Application Discontinuation
- 2009-04-16 NO NO20091492A patent/NO20091492L/no not_active Application Discontinuation
- 2009-04-16 IL IL198144A patent/IL198144A0/en unknown
- 2009-05-12 ZA ZA200903284A patent/ZA200903284B/xx unknown
- 2009-05-13 CR CR10793A patent/CR10793A/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
CA2673526A1 (en) | 2008-04-24 |
UY30643A1 (es) | 2008-05-02 |
CN101663026A (zh) | 2010-03-03 |
NI200900055A (es) | 2010-02-01 |
BRPI0719236A2 (pt) | 2014-07-08 |
CO6190539A2 (es) | 2010-08-19 |
AU2007313018A1 (en) | 2008-04-24 |
TW200831134A (en) | 2008-08-01 |
IL198144A0 (en) | 2009-12-24 |
JP2010506846A (ja) | 2010-03-04 |
AR063294A1 (es) | 2009-01-21 |
EA200970378A1 (ru) | 2009-10-30 |
KR20090067210A (ko) | 2009-06-24 |
EP2089002A1 (en) | 2009-08-19 |
US20080090903A1 (en) | 2008-04-17 |
MX2009003929A (es) | 2009-06-26 |
NO20091492L (no) | 2009-07-09 |
WO2008048802A1 (en) | 2008-04-24 |
CR10793A (es) | 2009-09-29 |
CL2007002943A1 (es) | 2008-04-18 |
SV2009003222A (es) | 2009-10-15 |
ZA200903284B (en) | 2010-07-28 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
PE20080887A1 (es) | Composiciones de carbamatos de fenilalquilo | |
AR047993A1 (es) | Composicion farmaceutica que comprende pimobendano | |
ATE499940T1 (de) | Carbonat- und carbamat-prodrugs von thiazolo ä4,5-dü-pyrimidinen | |
PE20090649A1 (es) | DERIVADOS DE PIRAZOL COMO INHIBIDORES DE LA ENZIMA 11ßHSD1 | |
EA201070597A1 (ru) | Антибактериальные аналоги аминогликозида | |
PE20201500A1 (es) | Inhibidores de glicolato oxidasa para el tratamiento de enfermedades | |
PE20060176A1 (es) | Antagonistas de cgrp seleccionados, procedimientos para su preparacion, y su empleo como medicamentos | |
AR077252A1 (es) | Enantiomeros de compuestos de espirooxindol y sus usos como agentes terapeuticos | |
PE20120028A1 (es) | Nueva composicion a base de acido gamma-hidroxibutirico | |
ECSP088765A (es) | Aminotetrahidropiranos como inhibidores de dipeptidil peptidasa-iv para el tratamiento o prevención de diabetes | |
PE20080832A1 (es) | Compuestos de n-metilaminometil isoindol y composiciones que los comprenden | |
EA201171109A1 (ru) | Новая композиция замедленного высвобождения соединений, выбранных из класса миорелаксантов центрального действия | |
UA86614C2 (ru) | Соединение, которое имеет активность ингибитора киназ, фармацевтическая композиция, которая включает указанное соединение, и их применение для приготовления лекарственного препарата | |
NZ591810A (en) | Pharmaceutical compositions and related methods of delivery the composition comprises a medium chain fatty acid | |
BRPI0608097A2 (pt) | composto ou enanciÈmeros, diastereÈmeros, sais, solvatos e n-óxidos do mesmo, composição farmacêutica, e,uso de uma quantidade eficaz de um composto | |
UY32547A (es) | Piperidinas sustituidas como antagonistas de ccr3 | |
MX2011013201A (es) | Composiciones para tratar adiccion a drogas y para mejorar comportamiento relacionado a la adiccion. | |
NZ619076A (en) | Isoxazolines as inhibitors of fatty acid amide hydrolase | |
BR112014015568A8 (pt) | compostos carbamato de fenila para uso em prevenção ou tratamento de epilepsia | |
AR083879A1 (es) | Analogos de aminoglicosidos antibacterianos, metodos de preparacion y uso como agentes terapeuticos | |
NO20051896L (no) | Farmasoytisk sammensetning som fast doseringsform samt fremgangsmate for fremstilling derav | |
ITBO20110012A1 (it) | Composizioni farmaceutiche comprendenti rifaximina e loro uso. | |
BRPI0506493A (pt) | combinações terapêuticas | |
MX2009003926A (es) | Composiciones de fenilalquilamino-carbamato. | |
BR112012025590A2 (pt) | análogos de pirimidinilpiperidiniloxipiridinona como moduladores de gpr119 |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC | Refusal |