PE20050360A1 - Inhibidores del proteasoma - Google Patents

Inhibidores del proteasoma

Info

Publication number
PE20050360A1
PE20050360A1 PE2004000784A PE2004000784A PE20050360A1 PE 20050360 A1 PE20050360 A1 PE 20050360A1 PE 2004000784 A PE2004000784 A PE 2004000784A PE 2004000784 A PE2004000784 A PE 2004000784A PE 20050360 A1 PE20050360 A1 PE 20050360A1
Authority
PE
Peru
Prior art keywords
amino
alkyl
methylbutyl
methyl
benzodioxaborol
Prior art date
Application number
PE2004000784A
Other languages
English (en)
Spanish (es)
Inventor
Alberto Bernareggi
Paolo G Cassara
Ernesto Menta
Sankar Chatterjee
Mclaughlin Patricia A Messina
Rafaella Bernardini
Munari Sergio De
Germano D Arasmo
Mohamed Iqbal
Ambrogio Oliva
Edmondo Ferretti
Original Assignee
Cephalon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cephalon Inc filed Critical Cephalon Inc
Publication of PE20050360A1 publication Critical patent/PE20050360A1/es

Links

PE2004000784A 2003-08-14 2004-08-13 Inhibidores del proteasoma PE20050360A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US49576403P 2003-08-14 2003-08-14

Publications (1)

Publication Number Publication Date
PE20050360A1 true PE20050360A1 (es) 2005-06-10

Family

ID=37426112

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2004000784A PE20050360A1 (es) 2003-08-14 2004-08-13 Inhibidores del proteasoma

Country Status (7)

Country Link
CN (1) CN1867572B (ru)
AR (2) AR045381A1 (ru)
MY (1) MY162518A (ru)
PE (1) PE20050360A1 (ru)
TW (1) TWI345465B (ru)
UA (1) UA88771C2 (ru)
ZA (1) ZA200601293B (ru)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105837608B (zh) * 2007-08-06 2018-06-08 米伦纽姆医药公司 蛋白酶体抑制剂及其组合物和用途
GEP20125599B (en) * 2007-08-06 2012-08-10 Millennium Pharm Inc Proteasome inhibitors
CN102961387B (zh) * 2007-08-06 2016-04-27 米伦纽姆医药公司 蛋白酶体抑制剂
DK2730581T3 (en) * 2008-06-17 2016-08-15 Millennium Pharm Inc Boronate Ester Compounds and Pharmaceutical Compositions thereof.
CN101638414B (zh) * 2008-07-30 2014-01-08 江苏先声药物研究有限公司 肽硼酸及其酯类化合物、制备方法及其用途
AR075090A1 (es) * 2008-09-29 2011-03-09 Millennium Pharm Inc Derivados de acido 1-amino-2-ciclobutiletilboronico inhibidores de proteosoma,utiles como agentes anticancerigenos, y composiciones farmaceuticas que los comprenden.
CN101747354B (zh) * 2008-12-04 2014-08-13 江苏先声药物研究有限公司 一类β氨基酸组成的二肽硼酸及其酯类化合物、制备方法及其用途
CA2785300A1 (en) * 2009-12-22 2011-07-21 Cephalon, Inc. Proteasome inhibitors and processes for their preparation, purification and use
CN102892291A (zh) * 2010-03-31 2013-01-23 米伦纽姆医药公司 1-氨基-2-环丙基乙硼酸衍生物
RU2717558C2 (ru) * 2014-10-01 2020-03-24 Мерк Патент Гмбх Производные бороновой кислоты
CN106588965A (zh) 2015-10-15 2017-04-26 北京大学 脲拟肽硼酸化合物及其药物组合物、制备方法和用途
WO2017198194A1 (zh) * 2016-05-19 2017-11-23 成都奥璟生物科技有限公司 一种硼酸和硼酸酯类化合物及其应用
PL3571208T3 (pl) * 2017-01-18 2021-09-20 Principia Biopharma Inc. Inhibitory immunoproteasomu
TW201831191A (zh) * 2017-01-23 2018-09-01 大陸商成都奥璟生物科技有限公司 一種新的硼酸衍生物及其藥物組合物
CN114437119A (zh) * 2020-10-30 2022-05-06 苏州开拓药业股份有限公司 一种c-Myc蛋白抑制剂及其制备方法和用途

Also Published As

Publication number Publication date
AR045381A1 (es) 2005-10-26
TW200529810A (en) 2005-09-16
TWI345465B (en) 2011-07-21
UA88771C2 (ru) 2009-11-25
AR095249A2 (es) 2015-09-30
MY162518A (en) 2017-06-15
CN1867572A (zh) 2006-11-22
ZA200601293B (en) 2009-09-30
CN1867572B (zh) 2012-03-28

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