PA8657701A1 - Derivado de quinolina, su uso, preparacion y medicamento que lo contiene - Google Patents

Derivado de quinolina, su uso, preparacion y medicamento que lo contiene

Info

Publication number
PA8657701A1
PA8657701A1 PA20058657701A PA8657701A PA8657701A1 PA 8657701 A1 PA8657701 A1 PA 8657701A1 PA 20058657701 A PA20058657701 A PA 20058657701A PA 8657701 A PA8657701 A PA 8657701A PA 8657701 A1 PA8657701 A1 PA 8657701A1
Authority
PA
Panama
Prior art keywords
preparation
derivative
quinolina
product containing
medicinal product
Prior art date
Application number
PA20058657701A
Other languages
English (en)
Inventor
Estefan Jaroch
Benjamin Bader
Roman Hillig
Wolfgang Schwede
Dieter Zopf
Laak Antonius Ter
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of PA8657701A1 publication Critical patent/PA8657701A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62Benzothiazoles
    • C07D277/64Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Abstract

LA PRESENTE INVENCION SE REFIERE A UN DERIVADO DE QUINOLINA DE LA FORMULA GENERAL A EN LA QUE R1,R2,R3,X,Y,Z Y A SE INDICAN EN LA DESCRIPCION Y EN LAS REIVINDICACIONES, AL USO DE LOS COMPUESTOS LA FORMULA GENERAL A PARA EL TRATAMIENTO DE DIVERSAS ENFERMEDADES, ASI COMO A LA PREPARACION DE COMPUESTOS LA FORMULA GENERAL A.
PA20058657701A 2004-12-22 2005-12-22 Derivado de quinolina, su uso, preparacion y medicamento que lo contiene PA8657701A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102004063223A DE102004063223A1 (de) 2004-12-22 2004-12-22 Chinolinderivat, dessen Verwendung, Herstellung und dieses enthaltendes Arzneimittel

Publications (1)

Publication Number Publication Date
PA8657701A1 true PA8657701A1 (es) 2006-09-08

Family

ID=36599298

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20058657701A PA8657701A1 (es) 2004-12-22 2005-12-22 Derivado de quinolina, su uso, preparacion y medicamento que lo contiene

Country Status (7)

Country Link
CN (1) CN101087788A (es)
AR (1) AR052544A1 (es)
DE (1) DE102004063223A1 (es)
GT (1) GT200500381A (es)
PA (1) PA8657701A1 (es)
SV (1) SV2007002357A (es)
UY (1) UY29308A1 (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103382206B (zh) * 2012-05-04 2016-09-28 上海恒瑞医药有限公司 喹啉或喹唑啉类衍生物、其制备方法及其在医药上的应用
CN106565823B (zh) * 2016-11-10 2020-09-11 珠海诺贝尔国际生物医药研究院有限公司 一种Eph受体小分子抑制剂及其制备方法
WO2019233458A1 (zh) * 2018-06-08 2019-12-12 江苏威凯尔医药科技有限公司 Vegfr抑制剂及其制备方法和应用
CN110577546B (zh) * 2018-06-08 2021-09-07 江苏威凯尔医药科技有限公司 Vegfr抑制剂及其制备方法和应用
CN113061142A (zh) * 2020-01-02 2021-07-02 爱科诺生物医药股份有限公司 一类具有程序性细胞坏死通路抑制活性的杂环化合物及其应用
CN113150009B (zh) * 2020-01-07 2023-05-23 爱科诺生物医药(香港)有限公司 一类具有程序性细胞坏死通路抑制活性的杂环化合物及其应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3919238A (en) * 1973-06-06 1975-11-11 Morton Norwich Products Inc 9-(Substituted amino)imidazo(4,5-f) quinolines
CA1263378A (en) * 1985-01-08 1989-11-28 Robert James Alaimo Imidazo¬4,5-f|quinolines useful as immunomodulating agents
EP0597003A1 (en) * 1991-08-02 1994-05-18 Pfizer Inc. Quinoline derivatives as immunostimulants

Also Published As

Publication number Publication date
DE102004063223A1 (de) 2006-07-13
UY29308A1 (es) 2006-06-30
SV2007002357A (es) 2007-02-16
GT200500381A (es) 2006-08-03
CN101087788A (zh) 2007-12-12
AR052544A1 (es) 2007-03-21

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