PA8633601A1 - STEROID PROPHARMS WITH ANDROGENIC ACTION - Google Patents

STEROID PROPHARMS WITH ANDROGENIC ACTION

Info

Publication number
PA8633601A1
PA8633601A1 PA20058633601A PA8633601A PA8633601A1 PA 8633601 A1 PA8633601 A1 PA 8633601A1 PA 20058633601 A PA20058633601 A PA 20058633601A PA 8633601 A PA8633601 A PA 8633601A PA 8633601 A1 PA8633601 A1 PA 8633601A1
Authority
PA
Panama
Prior art keywords
steroid
propharms
androgenic action
androgenic
action
Prior art date
Application number
PA20058633601A
Other languages
Spanish (es)
Inventor
Sven Ring
Ralf Wyrwa
Peter Droescher
Walter Elger
Alexander Hillisch
Birgitt Schneider
Gudrum Reddersen
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of PA8633601A1 publication Critical patent/PA8633601A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0038—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 with an androstane skeleton, including 18- or 19-substituted derivatives, 18-nor derivatives and also derivatives where position 17-beta is substituted by a carbon atom not directly bonded to a further carbon atom and not being part of an amide group
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26—Androgens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0044—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 with an estrane or gonane skeleton, including 18-substituted derivatives and derivatives where position 17-beta is substituted by a carbon atom not directly bonded to another carbon atom and not being part of an amide group

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

PROFARMACOS DE ESTEROIDES CON ACCION ANDROGENICA DE LA FORMULA GENERAL (I), EN LOS CUALES EL GRUPO Z ESTA UNIDO CON EL ESTEROIDE, COMPOSICIONES FARMACEUTICAS, QUE CONTIENEN ESTOS COMPUESTOS, ASI COMO SU USO PARA LA PREPARACION DE MEDICAMENTOS CON ACCION ANDROGENICA.STEROID PROFARMS WITH ANDROGENIC ACTION OF THE GENERAL FORMULA (I), IN WHICH GROUP Z IS JOINED WITH THE STEROID, PHARMACEUTICAL COMPOSITIONS, CONTAINING THESE COMPOUNDS, AS WELL AS THEIR USE FOR THE PREPARATION OF ANDROGENIC DRUGS.

PA20058633601A 2004-05-21 2005-05-20 STEROID PROPHARMS WITH ANDROGENIC ACTION PA8633601A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102004025986A DE102004025986A1 (en) 2004-05-21 2004-05-21 Steroid prodrugs with androgenic effects

Publications (1)

Publication Number Publication Date
PA8633601A1 true PA8633601A1 (en) 2006-07-03

Family

ID=34968657

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20058633601A PA8633601A1 (en) 2004-05-21 2005-05-20 STEROID PROPHARMS WITH ANDROGENIC ACTION

Country Status (22)

Country Link
EP (1) EP1747229A1 (en)
JP (1) JP2007538026A (en)
CN (1) CN1993375A (en)
AR (1) AR049547A1 (en)
AU (1) AU2005245568A1 (en)
BR (1) BRPI0510136A (en)
CA (1) CA2564963A1 (en)
CR (1) CR8785A (en)
DE (1) DE102004025986A1 (en)
EA (1) EA200602049A1 (en)
EC (1) ECSP067028A (en)
GT (1) GT200500122A (en)
IL (1) IL179293A0 (en)
MX (1) MXPA06013469A (en)
NO (1) NO20065885L (en)
PA (1) PA8633601A1 (en)
PE (1) PE20060271A1 (en)
SV (1) SV2006002123A (en)
TW (1) TW200613317A (en)
UY (1) UY28911A1 (en)
WO (1) WO2005113575A1 (en)
ZA (1) ZA200610769B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10027887A1 (en) 2000-05-31 2001-12-13 Jenapharm Gmbh Compounds with a sulfonamide group and pharmaceutical compositions containing these compounds
US7534780B2 (en) 2004-05-21 2009-05-19 Bayer Schering Pharma Aktiengesellschaft Estradiol prodrugs
DE102005057224A1 (en) * 2005-11-29 2007-05-31 Bayer Schering Pharma Ag New 9-alpha substituted estratriene derivatives esterified with a sulfamoylphenyl-substituted acid residue, are prodrugs useful as carboanhydrase inhibitors for treating estrogen deficiency disorders
DE102005057408A1 (en) * 2005-11-30 2007-05-31 Bayer Schering Pharma Ag New sulfamoylsulfonate prodrugs e.g. useful for protecting red blood cells from attack by parasites or for hormone replacement therapy, female fertility control or treating hormone-associated diseases
CN101708338B (en) * 2008-12-26 2014-06-04 中国人民解放军军事医学科学院放射与辐射医学研究所 Prodrug containing sterides structures and high dispersion preparation thereof
CN102964417A (en) * 2012-11-30 2013-03-13 华中药业股份有限公司 Synthetic method of 17-hydroxy tetrahydropyran ether steroid
CN107556258B (en) * 2017-08-22 2021-06-04 湖北江田精密化学有限公司 Preparation method of 4-amino-2-chloro-5 (1H-tetrazolyl-5) benzenesulfonamide
EP3533619A1 (en) * 2018-03-02 2019-09-04 Basf Se Heat sensitive recording material and color developer

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH545316A (en) * 1970-07-17 1973-12-15 Hoffmann La Roche Process for the preparation of acyl derivatives
US5001234A (en) * 1987-04-16 1991-03-19 The Upjohn Company Cyclic hydrocarbons with an aminoalkyl sidechain
US5571933A (en) * 1994-11-17 1996-11-05 Duquesne University Of The Holy Ghost Derivatives of estra 1,3,5(10)triene-17-one, 3-amino compounds and their use
DE19712488A1 (en) * 1997-03-25 1998-10-01 Knoell Hans Forschung Ev Steroid sulfamates, processes for their preparation and use thereof
DE10027887A1 (en) * 2000-05-31 2001-12-13 Jenapharm Gmbh Compounds with a sulfonamide group and pharmaceutical compositions containing these compounds

Also Published As

Publication number Publication date
WO2005113575A1 (en) 2005-12-01
EP1747229A1 (en) 2007-01-31
EA200602049A1 (en) 2007-06-29
AU2005245568A1 (en) 2005-12-01
AR049547A1 (en) 2006-08-16
CN1993375A (en) 2007-07-04
SV2006002123A (en) 2006-02-15
NO20065885L (en) 2006-12-19
GT200500122A (en) 2006-01-24
DE102004025986A1 (en) 2005-12-15
CR8785A (en) 2007-02-05
ZA200610769B (en) 2008-08-27
TW200613317A (en) 2006-05-01
ECSP067028A (en) 2006-12-29
CA2564963A1 (en) 2005-12-01
IL179293A0 (en) 2007-03-08
UY28911A1 (en) 2005-12-30
BRPI0510136A (en) 2007-10-02
JP2007538026A (en) 2007-12-27
MXPA06013469A (en) 2007-01-23
PE20060271A1 (en) 2006-05-25

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