BRPI0510136A - steroids with androgenic effect - Google Patents
steroids with androgenic effectInfo
- Publication number
- BRPI0510136A BRPI0510136A BRPI0510136-0A BRPI0510136A BRPI0510136A BR PI0510136 A BRPI0510136 A BR PI0510136A BR PI0510136 A BRPI0510136 A BR PI0510136A BR PI0510136 A BRPI0510136 A BR PI0510136A
- Authority
- BR
- Brazil
- Prior art keywords
- androgenic
- steroids
- effect
- androgenic effect
- steroidal
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0038—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 with an androstane skeleton, including 18- or 19-substituted derivatives, 18-nor derivatives and also derivatives where position 17-beta is substituted by a carbon atom not directly bonded to a further carbon atom and not being part of an amide group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0044—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 with an estrane or gonane skeleton, including 18-substituted derivatives and derivatives where position 17-beta is substituted by a carbon atom not directly bonded to another carbon atom and not being part of an amide group
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Reproductive Health (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
Abstract
PRODROGAS ESTERóIDES COM EFEITO ANDROGêNICO. A presente invenção refere-se a prodrogas esteroidais com efeito androgênico da fórmula geral (I), nas quais o grupo Z está ligado ao esteróide, a composições farmacêuticas, que contêm esses compostos, bem como ao uso dos mesmos para produção de medicamentos com efeito androgênico.STEROID PRODUCTS WITH ANDROGENIC EFFECT. The present invention relates to androgenic steroidal prodrugs of the general formula (I), in which the group Z is attached to the steroid, to pharmaceutical compositions containing such compounds, as well as to their use for the production of medicaments with steroidal effect. androgenic.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE102004025986A DE102004025986A1 (en) | 2004-05-21 | 2004-05-21 | Steroid prodrugs with androgenic effects |
PCT/EP2005/005256 WO2005113575A1 (en) | 2004-05-21 | 2005-05-10 | Steroid prodrugs with androgenic effect |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0510136A true BRPI0510136A (en) | 2007-10-02 |
Family
ID=34968657
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0510136-0A BRPI0510136A (en) | 2004-05-21 | 2005-05-10 | steroids with androgenic effect |
Country Status (22)
Country | Link |
---|---|
EP (1) | EP1747229A1 (en) |
JP (1) | JP2007538026A (en) |
CN (1) | CN1993375A (en) |
AR (1) | AR049547A1 (en) |
AU (1) | AU2005245568A1 (en) |
BR (1) | BRPI0510136A (en) |
CA (1) | CA2564963A1 (en) |
CR (1) | CR8785A (en) |
DE (1) | DE102004025986A1 (en) |
EA (1) | EA200602049A1 (en) |
EC (1) | ECSP067028A (en) |
GT (1) | GT200500122A (en) |
IL (1) | IL179293A0 (en) |
MX (1) | MXPA06013469A (en) |
NO (1) | NO20065885L (en) |
PA (1) | PA8633601A1 (en) |
PE (1) | PE20060271A1 (en) |
SV (1) | SV2006002123A (en) |
TW (1) | TW200613317A (en) |
UY (1) | UY28911A1 (en) |
WO (1) | WO2005113575A1 (en) |
ZA (1) | ZA200610769B (en) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10027887A1 (en) | 2000-05-31 | 2001-12-13 | Jenapharm Gmbh | Compounds with a sulfonamide group and pharmaceutical compositions containing these compounds |
US7534780B2 (en) | 2004-05-21 | 2009-05-19 | Bayer Schering Pharma Aktiengesellschaft | Estradiol prodrugs |
DE102005057224A1 (en) * | 2005-11-29 | 2007-05-31 | Bayer Schering Pharma Ag | New 9-alpha substituted estratriene derivatives esterified with a sulfamoylphenyl-substituted acid residue, are prodrugs useful as carboanhydrase inhibitors for treating estrogen deficiency disorders |
DE102005057408A1 (en) * | 2005-11-30 | 2007-05-31 | Bayer Schering Pharma Ag | New sulfamoylsulfonate prodrugs e.g. useful for protecting red blood cells from attack by parasites or for hormone replacement therapy, female fertility control or treating hormone-associated diseases |
CN101708338B (en) * | 2008-12-26 | 2014-06-04 | 中国人民解放军军事医学科学院放射与辐射医学研究所 | Prodrug containing sterides structures and high dispersion preparation thereof |
CN102964417A (en) * | 2012-11-30 | 2013-03-13 | 华中药业股份有限公司 | Synthetic method of 17-hydroxy tetrahydropyran ether steroid |
CN107556258B (en) * | 2017-08-22 | 2021-06-04 | 湖北江田精密化学有限公司 | Preparation method of 4-amino-2-chloro-5 (1H-tetrazolyl-5) benzenesulfonamide |
EP3533619A1 (en) * | 2018-03-02 | 2019-09-04 | Basf Se | Heat sensitive recording material and color developer |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH545316A (en) * | 1970-07-17 | 1973-12-15 | Hoffmann La Roche | Process for the preparation of acyl derivatives |
US5001234A (en) * | 1987-04-16 | 1991-03-19 | The Upjohn Company | Cyclic hydrocarbons with an aminoalkyl sidechain |
US5571933A (en) * | 1994-11-17 | 1996-11-05 | Duquesne University Of The Holy Ghost | Derivatives of estra 1,3,5(10)triene-17-one, 3-amino compounds and their use |
DE19712488A1 (en) * | 1997-03-25 | 1998-10-01 | Knoell Hans Forschung Ev | Steroid sulfamates, processes for their preparation and use thereof |
DE10027887A1 (en) * | 2000-05-31 | 2001-12-13 | Jenapharm Gmbh | Compounds with a sulfonamide group and pharmaceutical compositions containing these compounds |
-
2004
- 2004-05-21 DE DE102004025986A patent/DE102004025986A1/en not_active Ceased
-
2005
- 2005-05-10 EP EP05742657A patent/EP1747229A1/en not_active Withdrawn
- 2005-05-10 BR BRPI0510136-0A patent/BRPI0510136A/en not_active Application Discontinuation
- 2005-05-10 WO PCT/EP2005/005256 patent/WO2005113575A1/en active Application Filing
- 2005-05-10 JP JP2007517047A patent/JP2007538026A/en active Pending
- 2005-05-10 MX MXPA06013469A patent/MXPA06013469A/en not_active Application Discontinuation
- 2005-05-10 EA EA200602049A patent/EA200602049A1/en unknown
- 2005-05-10 CA CA002564963A patent/CA2564963A1/en not_active Abandoned
- 2005-05-10 CN CNA200580016339XA patent/CN1993375A/en active Pending
- 2005-05-10 AU AU2005245568A patent/AU2005245568A1/en not_active Abandoned
- 2005-05-20 AR ARP050102084A patent/AR049547A1/en not_active Application Discontinuation
- 2005-05-20 PE PE2005000556A patent/PE20060271A1/en not_active Application Discontinuation
- 2005-05-20 GT GT200500122A patent/GT200500122A/en unknown
- 2005-05-20 TW TW094116504A patent/TW200613317A/en unknown
- 2005-05-20 UY UY28911A patent/UY28911A1/en not_active Application Discontinuation
- 2005-05-20 PA PA20058633601A patent/PA8633601A1/en unknown
- 2005-05-23 SV SV2005002123A patent/SV2006002123A/en not_active Application Discontinuation
-
2006
- 2006-11-15 IL IL179293A patent/IL179293A0/en unknown
- 2006-11-27 EC EC2006007028A patent/ECSP067028A/en unknown
- 2006-12-05 CR CR8785A patent/CR8785A/en not_active Application Discontinuation
- 2006-12-19 NO NO20065885A patent/NO20065885L/en unknown
- 2006-12-20 ZA ZA200610769A patent/ZA200610769B/en unknown
Also Published As
Publication number | Publication date |
---|---|
CA2564963A1 (en) | 2005-12-01 |
SV2006002123A (en) | 2006-02-15 |
CN1993375A (en) | 2007-07-04 |
MXPA06013469A (en) | 2007-01-23 |
EP1747229A1 (en) | 2007-01-31 |
ZA200610769B (en) | 2008-08-27 |
JP2007538026A (en) | 2007-12-27 |
AR049547A1 (en) | 2006-08-16 |
CR8785A (en) | 2007-02-05 |
DE102004025986A1 (en) | 2005-12-15 |
NO20065885L (en) | 2006-12-19 |
AU2005245568A1 (en) | 2005-12-01 |
ECSP067028A (en) | 2006-12-29 |
PA8633601A1 (en) | 2006-07-03 |
IL179293A0 (en) | 2007-03-08 |
WO2005113575A1 (en) | 2005-12-01 |
PE20060271A1 (en) | 2006-05-25 |
GT200500122A (en) | 2006-01-24 |
TW200613317A (en) | 2006-05-01 |
UY28911A1 (en) | 2005-12-30 |
EA200602049A1 (en) | 2007-06-29 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] |