PA8633801A1 - DERIVATIVES OF SULFAMOYLBENZOATE AND SULFAMOYLAMINOBENZOATE OF ESTRIOL, AND DERIVATIVES OF SULFAMOYLBENZOATE AND SULFAMOYLAMINOBENZOATE OF STETROL - Google Patents

DERIVATIVES OF SULFAMOYLBENZOATE AND SULFAMOYLAMINOBENZOATE OF ESTRIOL, AND DERIVATIVES OF SULFAMOYLBENZOATE AND SULFAMOYLAMINOBENZOATE OF STETROL

Info

Publication number
PA8633801A1
PA8633801A1 PA20058633801A PA8633801A PA8633801A1 PA 8633801 A1 PA8633801 A1 PA 8633801A1 PA 20058633801 A PA20058633801 A PA 20058633801A PA 8633801 A PA8633801 A PA 8633801A PA 8633801 A1 PA8633801 A1 PA 8633801A1
Authority
PA
Panama
Prior art keywords
sulfamoylaminobenzoate
sulfamoylbenzoate
derivatives
stetrol
estriol
Prior art date
Application number
PA20058633801A
Other languages
Spanish (es)
Inventor
Sven Ring
Ralf Wyrwa
Peter Droescher
Walter Elger
Alexander Hillisch
Gudrun Reddersen
Birgitt Schneider
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34969311&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PA8633801(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Ag filed Critical Schering Ag
Publication of PA8633801A1 publication Critical patent/PA8633801A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0072—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26—Androgens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/34—Gestagens

Abstract

PRODROGAS DE ESTRIOL Y ESTETROL DE LA FORMULA GENERAL (I) DONDE EL GRUPO Y ESTA UNIDO AL ESTEROIDE PROCEDIMIENTO PARA SU PREPARACION, COMPOSICIONES FARMACEUTICAS QUE CONTIENEN ESTOS COMPUESTOS Y SU USO PAR PREPARAR MEDICAMENTOS CON EFECTO ESTROGENO.ESTRIOL AND STETROL PRODUCTS OF THE GENERAL FORMULA (I) WHERE THE GROUP IS AND IS JOINED TO THE STEROID PROCEDURE FOR THE PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND THEIR USE TO PREPARE MEDICATIONS WITH STROGEN EFFECT.

PA20058633801A 2004-05-21 2005-05-20 DERIVATIVES OF SULFAMOYLBENZOATE AND SULFAMOYLAMINOBENZOATE OF ESTRIOL, AND DERIVATIVES OF SULFAMOYLBENZOATE AND SULFAMOYLAMINOBENZOATE OF STETROL PA8633801A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102004025985A DE102004025985A1 (en) 2004-05-21 2004-05-21 Estriol and estetrol prodrugs

Publications (1)

Publication Number Publication Date
PA8633801A1 true PA8633801A1 (en) 2006-03-24

Family

ID=34969311

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20058633801A PA8633801A1 (en) 2004-05-21 2005-05-20 DERIVATIVES OF SULFAMOYLBENZOATE AND SULFAMOYLAMINOBENZOATE OF ESTRIOL, AND DERIVATIVES OF SULFAMOYLBENZOATE AND SULFAMOYLAMINOBENZOATE OF STETROL

Country Status (11)

Country Link
EP (1) EP1747231A1 (en)
JP (1) JP2007538027A (en)
AR (1) AR049108A1 (en)
DE (1) DE102004025985A1 (en)
GT (1) GT200500120A (en)
PA (1) PA8633801A1 (en)
PE (1) PE20060314A1 (en)
SV (1) SV2006002122A (en)
TW (1) TW200612962A (en)
UY (1) UY28910A1 (en)
WO (1) WO2005113576A1 (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10027887A1 (en) 2000-05-31 2001-12-13 Jenapharm Gmbh Compounds with a sulfonamide group and pharmaceutical compositions containing these compounds
DE102004025966A1 (en) * 2004-05-21 2005-12-15 Schering Ag Estradiol prodrugs
US7534780B2 (en) 2004-05-21 2009-05-19 Bayer Schering Pharma Aktiengesellschaft Estradiol prodrugs
DE102005057224A1 (en) * 2005-11-29 2007-05-31 Bayer Schering Pharma Ag New 9-alpha substituted estratriene derivatives esterified with a sulfamoylphenyl-substituted acid residue, are prodrugs useful as carboanhydrase inhibitors for treating estrogen deficiency disorders
DE102005057408A1 (en) * 2005-11-30 2007-05-31 Bayer Schering Pharma Ag New sulfamoylsulfonate prodrugs e.g. useful for protecting red blood cells from attack by parasites or for hormone replacement therapy, female fertility control or treating hormone-associated diseases
CN100396693C (en) * 2006-11-08 2008-06-25 浙江大学 Preparation method of 1,4-dipregnene-16-beta-methyl-17-alpha-21-bihydroxy object
CN102079771B (en) * 2010-12-10 2012-10-03 郑州大学 Estrogen amino-acid ester compound with antitumor activity as well as synthetic method thereof

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1238739A (en) * 1958-08-04 1960-08-19 Chimiotherapie Lab Franc Process for the preparation of water-soluble testosterone derivatives
FR8290M (en) * 1968-12-31 1970-11-09 Rech Chimiques Et Ind Mar Lab
US5001234A (en) * 1987-04-16 1991-03-19 The Upjohn Company Cyclic hydrocarbons with an aminoalkyl sidechain
US5116828A (en) * 1989-10-26 1992-05-26 Nippon Zoki Pharmaceutical Co., Ltd. Pharmaceutical composition for treatment of osteoporosis
US5571933A (en) * 1994-11-17 1996-11-05 Duquesne University Of The Holy Ghost Derivatives of estra 1,3,5(10)triene-17-one, 3-amino compounds and their use
DE19712488A1 (en) * 1997-03-25 1998-10-01 Knoell Hans Forschung Ev Steroid sulfamates, processes for their preparation and use thereof
EP1284272A4 (en) * 2000-04-24 2003-09-10 Kyowa Hakko Kogyo Kk Estra-1,3,5(10)-triene derivatives
DE10027887A1 (en) * 2000-05-31 2001-12-13 Jenapharm Gmbh Compounds with a sulfonamide group and pharmaceutical compositions containing these compounds
GB0015876D0 (en) * 2000-06-28 2000-08-23 Novartis Ag Organic compounds
GB0316290D0 (en) * 2003-07-11 2003-08-13 Glaxo Group Ltd Novel compounds
TWI331154B (en) * 2003-11-12 2010-10-01 Solvay Pharm Gmbh Novel 17-hydroxysteroid dehydrogenase type i inhibitors
DE102004025966A1 (en) * 2004-05-21 2005-12-15 Schering Ag Estradiol prodrugs

Also Published As

Publication number Publication date
EP1747231A1 (en) 2007-01-31
AR049108A1 (en) 2006-06-28
WO2005113576A1 (en) 2005-12-01
JP2007538027A (en) 2007-12-27
PE20060314A1 (en) 2006-05-25
SV2006002122A (en) 2006-05-09
TW200612962A (en) 2006-05-01
UY28910A1 (en) 2005-12-30
GT200500120A (en) 2006-01-24
DE102004025985A1 (en) 2005-12-15

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