PA8629401A1 - D-HOMO-17-CHLORINE-16 (17) ENO STEROIDS - Google Patents

D-HOMO-17-CHLORINE-16 (17) ENO STEROIDS

Info

Publication number
PA8629401A1
PA8629401A1 PA20058629401A PA8629401A PA8629401A1 PA 8629401 A1 PA8629401 A1 PA 8629401A1 PA 20058629401 A PA20058629401 A PA 20058629401A PA 8629401 A PA8629401 A PA 8629401A PA 8629401 A1 PA8629401 A1 PA 8629401A1
Authority
PA
Panama
Prior art keywords
steroids
homo
chlorine
eno
compounds
Prior art date
Application number
PA20058629401A
Other languages
Spanish (es)
Inventor
Guenter Kaufmann
Sven Ring
Ralf Wyrwa
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of PA8629401A1 publication Critical patent/PA8629401A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J63/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J63/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C07J63/008Expansion of ring D by one atom, e.g. D homo steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26Androgens

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

D-HOMO-17-CLORO-16(17)-EN ESTEROIDES DE LA FORMULA I CON ACTIVIDAD ANDROGENA, PROCEDIMIENTO PARA SU PREPARACION Y COMPOSICIONES FARMACEUTICAS QUE CONTIENEN ESTOS COMPUESTOS Y SU USO PARA PREPARAR MEDICAMENTOS.D-HOMO-17-CHLORINE-16 (17) - IN FORMULA STEROIDS WITH ANDROGEN ACTIVITY, PROCEDURE FOR THE PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND THEIR USE TO PREPARE MEDICATIONS.

PA20058629401A 2004-04-08 2005-04-08 D-HOMO-17-CHLORINE-16 (17) ENO STEROIDS PA8629401A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102004018441A DE102004018441B4 (en) 2004-04-08 2004-04-08 D-homo-17-chloro-16 (17) and steroids

Publications (1)

Publication Number Publication Date
PA8629401A1 true PA8629401A1 (en) 2006-07-03

Family

ID=34966688

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20058629401A PA8629401A1 (en) 2004-04-08 2005-04-08 D-HOMO-17-CHLORINE-16 (17) ENO STEROIDS

Country Status (18)

Country Link
EP (1) EP1735331A1 (en)
KR (1) KR20070007910A (en)
CN (1) CN1997659A (en)
AR (1) AR048536A1 (en)
AU (1) AU2005231970A1 (en)
CA (1) CA2563541A1 (en)
CR (1) CR8736A (en)
DE (1) DE102004018441B4 (en)
EA (1) EA200601842A1 (en)
EC (1) ECSP066973A (en)
GT (1) GT200500084A (en)
MX (1) MXPA06012849A (en)
NO (1) NO20065126L (en)
PA (1) PA8629401A1 (en)
SV (1) SV2005002076A (en)
TW (1) TW200603812A (en)
WO (1) WO2005097819A1 (en)
ZA (1) ZA200609275B (en)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4788218A (en) * 1984-05-21 1988-11-29 Sri International 17 a β-hydroxy-7 α-methyl-d-homo-19-norandrost-4,16-diene-3-one and the 17-esters thereof: methods of preparation and uses
DE4042005A1 (en) * 1990-12-22 1992-06-25 Schering Ag D-HOMO- (16-EN) -11 (BETA) -ARYL-4-ESTRENE
DK0640294T4 (en) * 1993-08-21 2000-04-03 Nestle Sa Preparation of a spice
DE10151365A1 (en) * 2001-10-17 2003-04-30 Schering Ag New 17-chloro-D-homosteroids, useful as estrogen receptor ligands for female or male contraception or treating benign or malignant proliferative diseases of the ovary

Also Published As

Publication number Publication date
TW200603812A (en) 2006-02-01
CR8736A (en) 2007-08-28
AR048536A1 (en) 2006-05-03
WO2005097819A1 (en) 2005-10-20
EA200601842A1 (en) 2007-04-27
DE102004018441B4 (en) 2007-12-20
CA2563541A1 (en) 2005-10-20
DE102004018441A1 (en) 2005-11-03
EP1735331A1 (en) 2006-12-27
MXPA06012849A (en) 2007-01-26
NO20065126L (en) 2007-01-04
SV2005002076A (en) 2005-12-06
AU2005231970A1 (en) 2005-10-20
CN1997659A (en) 2007-07-11
GT200500084A (en) 2006-03-24
KR20070007910A (en) 2007-01-16
ECSP066973A (en) 2006-12-29
ZA200609275B (en) 2009-08-26

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