OA12893A - Broadspectrum 2-Amino-Benzothiazole Sulfonamide HIV Protease Inhibitors. - Google Patents
Broadspectrum 2-Amino-Benzothiazole Sulfonamide HIV Protease Inhibitors. Download PDFInfo
- Publication number
- OA12893A OA12893A OA1200500026A OA1200500026A OA12893A OA 12893 A OA12893 A OA 12893A OA 1200500026 A OA1200500026 A OA 1200500026A OA 1200500026 A OA1200500026 A OA 1200500026A OA 12893 A OA12893 A OA 12893A
- Authority
- OA
- OAPI
- Prior art keywords
- amino
- benzyl
- sulfonyl
- hydroxy
- isobutyl
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP02078231 | 2002-08-02 | ||
US42786202P | 2002-11-20 | 2002-11-20 |
Publications (1)
Publication Number | Publication Date |
---|---|
OA12893A true OA12893A (en) | 2006-10-13 |
Family
ID=38068099
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
OA1200500026A OA12893A (en) | 2002-08-02 | 2003-08-04 | Broadspectrum 2-Amino-Benzothiazole Sulfonamide HIV Protease Inhibitors. |
Country Status (5)
Country | Link |
---|---|
JP (1) | JP4879484B2 (ja) |
KR (1) | KR101327772B1 (ja) |
CN (1) | CN101445493A (ja) |
OA (1) | OA12893A (ja) |
ZA (1) | ZA200500926B (ja) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
UA103013C2 (uk) * | 2007-12-06 | 2013-09-10 | Тиботек Фармасьютикелз | Амідні сполуки як активатори противірусних препаратів |
KR20140027295A (ko) * | 2011-04-21 | 2014-03-06 | 길리애드 사이언시즈, 인코포레이티드 | 벤조티아졸 화합물 및 이들의 약학적 용도 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0715618B1 (en) * | 1993-08-24 | 1998-12-16 | G.D. Searle & Co. | Hydroxyethylamino sulphonamides useful as retroviral protease inhibitors |
US5756533A (en) * | 1995-03-10 | 1998-05-26 | G.D. Searle & Co. | Amino acid hydroxyethylamino sulfonamide retroviral protease inhibitors |
AU7722296A (en) * | 1995-11-15 | 1997-06-05 | G.D. Searle & Co. | Substituted sulfonylalkanoylamino hydroxyethylamino sulfonamide retroviral protease inhibitors |
AU4828199A (en) * | 1998-06-23 | 2000-01-10 | Board Of Trustees Of The University Of Illinois, The | Multi-drug resistant retroviral protease inhibitors and associated methods |
DK1222192T3 (da) * | 1999-10-06 | 2008-10-20 | Tibotec Pharm Ltd | Hexahydrofuro-2,3-b furan-3-yl-N-3-(1,3-benzodioxol-5-ylsulfonyl)(isobutyl)amino-1-benzyl-2-hydroxypropyl-carbamat som retroviral proteaseinhibitor |
CN100369904C (zh) * | 2001-02-14 | 2008-02-20 | 泰博特克药品有限公司 | 2-(取代-氨基)-苯并噻唑磺酰胺hiv蛋白酶抑制剂 |
-
2003
- 2003-08-04 OA OA1200500026A patent/OA12893A/en unknown
- 2003-08-04 CN CN 200810170597 patent/CN101445493A/zh active Pending
- 2003-08-04 JP JP2004526916A patent/JP4879484B2/ja not_active Expired - Fee Related
- 2003-08-04 KR KR1020107026841A patent/KR101327772B1/ko active IP Right Grant
-
2006
- 2006-01-16 ZA ZA200500926A patent/ZA200500926B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
JP4879484B2 (ja) | 2012-02-22 |
KR20100137584A (ko) | 2010-12-30 |
KR101327772B1 (ko) | 2013-11-11 |
JP2006503815A (ja) | 2006-02-02 |
ZA200500926B (en) | 2006-03-29 |
CN101445493A (zh) | 2009-06-03 |
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