OA11045A - Conformationally constrained lh-rh analogues theiruses and pharmaceutical commpositions containing them - Google Patents

Conformationally constrained lh-rh analogues theiruses and pharmaceutical commpositions containing them Download PDF

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Publication number
OA11045A
OA11045A OA9900098A OA9900098A OA11045A OA 11045 A OA11045 A OA 11045A OA 9900098 A OA9900098 A OA 9900098A OA 9900098 A OA9900098 A OA 9900098A OA 11045 A OA11045 A OA 11045A
Authority
OA
OAPI
Prior art keywords
peptide
spl
formula
pro
ser
Prior art date
Application number
OA9900098A
Other languages
English (en)
Inventor
Remi Delansorne
Jacques Paris
Original Assignee
Theramex
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Theramex filed Critical Theramex
Publication of OA11045A publication Critical patent/OA11045A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/23Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10STECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00Peptide or protein sequence
    • Y10S930/01Peptide or protein sequence
    • Y10S930/13Luteinizing hormone-releasing hormone; related peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Endocrinology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Gynecology & Obstetrics (AREA)
  • Reproductive Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Steroid Compounds (AREA)
OA9900098A 1996-11-14 1999-05-12 Conformationally constrained lh-rh analogues theiruses and pharmaceutical commpositions containing them OA11045A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP96402441A EP0842946A1 (de) 1996-11-14 1996-11-14 LHRH Analoge mit starrer Konformation, deren Verwendungen und pharmazeutische Zusammensetzungen

Publications (1)

Publication Number Publication Date
OA11045A true OA11045A (en) 2003-03-07

Family

ID=8225315

Family Applications (1)

Application Number Title Priority Date Filing Date
OA9900098A OA11045A (en) 1996-11-14 1999-05-12 Conformationally constrained lh-rh analogues theiruses and pharmaceutical commpositions containing them

Country Status (28)

Country Link
US (1) US6153587A (de)
EP (2) EP0842946A1 (de)
JP (1) JP2001503444A (de)
KR (1) KR20000068975A (de)
CN (1) CN1237979A (de)
AP (1) AP9901529A0 (de)
AT (1) ATE196914T1 (de)
AU (1) AU5481798A (de)
BR (1) BR9713060A (de)
CA (1) CA2270158A1 (de)
CO (1) CO4930283A1 (de)
CZ (1) CZ172899A3 (de)
DE (1) DE69703308D1 (de)
EE (1) EE9900174A (de)
HU (1) HUP0000249A3 (de)
ID (1) ID21990A (de)
IL (1) IL129821A0 (de)
JO (1) JO1999B1 (de)
MA (1) MA26447A1 (de)
NO (1) NO992298L (de)
NZ (1) NZ335454A (de)
OA (1) OA11045A (de)
PE (1) PE16899A1 (de)
PL (1) PL333358A1 (de)
TN (1) TNSN97173A1 (de)
TR (1) TR199901054T2 (de)
WO (1) WO1998021229A1 (de)
ZA (1) ZA9710254B (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5677184A (en) * 1994-04-19 1997-10-14 Takeda Chemical Industries, Ltd. CHO cells that express human LH-RH receptor
EP0842946A1 (de) * 1996-11-14 1998-05-20 Laboratoire Theramex S.A. LHRH Analoge mit starrer Konformation, deren Verwendungen und pharmazeutische Zusammensetzungen
EP0882736A1 (de) * 1997-06-02 1998-12-09 Laboratoire Theramex S.A. Peptidanaloge des LH-RH, ihre Verwendungen und die sie enthaltenden pharmazeutischen Zusammensetzungen
EP0998940A1 (de) * 1998-09-30 2000-05-10 Laboratoire Theramex Pharmazeutische zusammensetzung basierend auf alpha-cyclodextrin für die orale verabreichung von LH-RH analogen
CN1261449C (zh) * 1999-04-26 2006-06-28 味之素株式会社 促黑素细胞激素抑制剂
US8821943B2 (en) * 2006-09-12 2014-09-02 Board Of Regents Of The University Of Nebraska Methods and compositions for targeted delivery of therapeutic agents
EP4225771A4 (de) * 2020-10-08 2025-01-01 Dignify Therapeutics, LLC Zusammensetzungen zur induzierung von urinentleerung und -defäkation

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4377515A (en) * 1979-10-01 1983-03-22 Merck & Co., Inc. Long lasting agonists and antagonists of LH-RH
US5110904A (en) * 1989-08-07 1992-05-05 Abbott Laboratories Lhrh analogs
EP0842946A1 (de) * 1996-11-14 1998-05-20 Laboratoire Theramex S.A. LHRH Analoge mit starrer Konformation, deren Verwendungen und pharmazeutische Zusammensetzungen

Also Published As

Publication number Publication date
MA26447A1 (fr) 2004-12-20
JO1999B1 (en) 1999-05-15
CN1237979A (zh) 1999-12-08
NZ335454A (en) 2000-10-27
BR9713060A (pt) 2000-04-11
WO1998021229A1 (en) 1998-05-22
TR199901054T2 (xx) 1999-07-21
AP9901529A0 (en) 1999-06-30
CA2270158A1 (en) 1998-05-22
ATE196914T1 (de) 2000-10-15
PL333358A1 (en) 1999-12-06
US6153587A (en) 2000-11-28
NO992298L (no) 1999-07-08
HUP0000249A3 (en) 2000-11-28
CO4930283A1 (es) 2000-06-27
TNSN97173A1 (fr) 2005-03-15
KR20000068975A (ko) 2000-11-25
PE16899A1 (es) 1999-02-19
ID21990A (id) 1999-08-19
EP0842946A1 (de) 1998-05-20
HUP0000249A2 (en) 2000-07-28
AU5481798A (en) 1998-06-03
EE9900174A (et) 1999-12-15
IL129821A0 (en) 2000-02-29
ZA9710254B (en) 1998-05-28
CZ172899A3 (cs) 1999-08-11
EP0937101A1 (de) 1999-08-25
NO992298D0 (no) 1999-05-12
JP2001503444A (ja) 2001-03-13
EP0937101B1 (de) 2000-10-11
DE69703308D1 (de) 2000-11-16

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