BR9713060A - Análogos de lh-rh estruturalmente submetidos, os seus usos e as composições farmacêuticas contendo-os. - Google Patents

Análogos de lh-rh estruturalmente submetidos, os seus usos e as composições farmacêuticas contendo-os.

Info

Publication number
BR9713060A
BR9713060A BR9713060-5A BR9713060A BR9713060A BR 9713060 A BR9713060 A BR 9713060A BR 9713060 A BR9713060 A BR 9713060A BR 9713060 A BR9713060 A BR 9713060A
Authority
BR
Brazil
Prior art keywords
pharmaceutical compositions
compositions containing
analogs
structurally
subjected
Prior art date
Application number
BR9713060-5A
Other languages
English (en)
Inventor
Remi Delansorne
Jacques Paris
Original Assignee
Theramex
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Theramex filed Critical Theramex
Publication of BR9713060A publication Critical patent/BR9713060A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/23Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10STECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00Peptide or protein sequence
    • Y10S930/01Peptide or protein sequence
    • Y10S930/13Luteinizing hormone-releasing hormone; related peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Endocrinology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Gynecology & Obstetrics (AREA)
  • Reproductive Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Steroid Compounds (AREA)

Abstract

Patente de Invenção para "ANáLOGOS DE LH-RH ESTRUTURALMENTE SUBMETIDOS, OS SEUS USOS E AS COMPOSIçõES FARMACêUTICAS CONTENDO-OS". A invenção refere-se aos peptídios análogos LH-RH com excelente afinidade aos receptores LH-RH, de fórmula: V-W-X-SPL-Y-Pro-Z onde V, W, X, SPL, Y e Z são tal como definidos nas especificações. A invenção ainda refere-se aos usos dos peptídios análogos e às composições farmacêuticas contendo-os.
BR9713060-5A 1996-11-14 1997-11-12 Análogos de lh-rh estruturalmente submetidos, os seus usos e as composições farmacêuticas contendo-os. BR9713060A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP96402441A EP0842946A1 (en) 1996-11-14 1996-11-14 Conformationally constrained LH-RH analogues, their uses and pharmaceutical compositions containing them
PCT/EP1997/006322 WO1998021229A1 (en) 1996-11-14 1997-11-12 Conformationally constrained lh-rh analogues, their uses and pharmaceutical compositions containing them

Publications (1)

Publication Number Publication Date
BR9713060A true BR9713060A (pt) 2000-04-11

Family

ID=8225315

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9713060-5A BR9713060A (pt) 1996-11-14 1997-11-12 Análogos de lh-rh estruturalmente submetidos, os seus usos e as composições farmacêuticas contendo-os.

Country Status (28)

Country Link
US (1) US6153587A (pt)
EP (2) EP0842946A1 (pt)
JP (1) JP2001503444A (pt)
KR (1) KR20000068975A (pt)
CN (1) CN1237979A (pt)
AP (1) AP9901529A0 (pt)
AT (1) ATE196914T1 (pt)
AU (1) AU5481798A (pt)
BR (1) BR9713060A (pt)
CA (1) CA2270158A1 (pt)
CO (1) CO4930283A1 (pt)
CZ (1) CZ172899A3 (pt)
DE (1) DE69703308D1 (pt)
EE (1) EE9900174A (pt)
HU (1) HUP0000249A3 (pt)
ID (1) ID21990A (pt)
IL (1) IL129821A0 (pt)
JO (1) JO1999B1 (pt)
MA (1) MA26447A1 (pt)
NO (1) NO992298L (pt)
NZ (1) NZ335454A (pt)
OA (1) OA11045A (pt)
PE (1) PE16899A1 (pt)
PL (1) PL333358A1 (pt)
TN (1) TNSN97173A1 (pt)
TR (1) TR199901054T2 (pt)
WO (1) WO1998021229A1 (pt)
ZA (1) ZA9710254B (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5677184A (en) * 1994-04-19 1997-10-14 Takeda Chemical Industries, Ltd. CHO cells that express human LH-RH receptor
EP0842946A1 (en) * 1996-11-14 1998-05-20 Laboratoire Theramex S.A. Conformationally constrained LH-RH analogues, their uses and pharmaceutical compositions containing them
EP0882736A1 (en) * 1997-06-02 1998-12-09 Laboratoire Theramex S.A. LH-RH peptide analogues, their uses and pharmaceutical compositions containing them
EP0998940A1 (en) * 1998-09-30 2000-05-10 Laboratoire Theramex Pharmaceutical compositions based on alpha-cyclodextrin for the oral administration of LH-RH analogues
KR100679878B1 (ko) * 1999-04-26 2007-02-07 아지노모토 가부시키가이샤 멜라노사이트-자극 호르몬 억제제
WO2008033924A2 (en) * 2006-09-12 2008-03-20 Board Of Regents Of The University Of Nebraska Methods and compositions for targeted delivery of therapeutic agents
AU2021358995A1 (en) * 2020-10-08 2023-06-08 Dignify Therapeutics, Llc Compositions for inducing urinary voiding and defecation

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4377515A (en) * 1979-10-01 1983-03-22 Merck & Co., Inc. Long lasting agonists and antagonists of LH-RH
US5110904A (en) * 1989-08-07 1992-05-05 Abbott Laboratories Lhrh analogs
EP0842946A1 (en) * 1996-11-14 1998-05-20 Laboratoire Theramex S.A. Conformationally constrained LH-RH analogues, their uses and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
MA26447A1 (fr) 2004-12-20
TNSN97173A1 (fr) 2005-03-15
NO992298L (no) 1999-07-08
HUP0000249A2 (en) 2000-07-28
KR20000068975A (ko) 2000-11-25
EP0937101A1 (en) 1999-08-25
CA2270158A1 (en) 1998-05-22
PE16899A1 (es) 1999-02-19
CN1237979A (zh) 1999-12-08
WO1998021229A1 (en) 1998-05-22
HUP0000249A3 (en) 2000-11-28
DE69703308D1 (de) 2000-11-16
IL129821A0 (en) 2000-02-29
CZ172899A3 (cs) 1999-08-11
ID21990A (id) 1999-08-19
ATE196914T1 (de) 2000-10-15
EE9900174A (et) 1999-12-15
ZA9710254B (en) 1998-05-28
AU5481798A (en) 1998-06-03
EP0937101B1 (en) 2000-10-11
EP0842946A1 (en) 1998-05-20
US6153587A (en) 2000-11-28
OA11045A (en) 2003-03-07
JO1999B1 (en) 1999-05-15
TR199901054T2 (xx) 1999-07-21
CO4930283A1 (es) 2000-06-27
NZ335454A (en) 2000-10-27
PL333358A1 (en) 1999-12-06
NO992298D0 (no) 1999-05-12
AP9901529A0 (en) 1999-06-30
JP2001503444A (ja) 2001-03-13

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 5A, 6A, 7A, 8A E 9A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1894 DE 24/04/2007.