OA06083A - Nouvelles pipérazines disubstituées, leurs procédés de préparation et les compositions pharmaceutiques les renfermant. - Google Patents

Nouvelles pipérazines disubstituées, leurs procédés de préparation et les compositions pharmaceutiques les renfermant.

Info

Publication number
OA06083A
OA06083A OA56649A OA56649A OA06083A OA 06083 A OA06083 A OA 06083A OA 56649 A OA56649 A OA 56649A OA 56649 A OA56649 A OA 56649A OA 06083 A OA06083 A OA 06083A
Authority
OA
OAPI
Prior art keywords
pharmaceutical compositions
compositions containing
preparation processes
disubstituted piperazines
new disubstituted
Prior art date
Application number
OA56649A
Other languages
English (en)
French (fr)
Inventor
Gilbert Regnier
Roger Canevari
Michel Laubie Et Jean Poignant
Original Assignee
Science Union & Cie Ste Franca
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Science Union & Cie Ste Franca filed Critical Science Union & Cie Ste Franca
Publication of OA06083A publication Critical patent/OA06083A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D327/00Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D327/02Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms one oxygen atom and one sulfur atom
    • C07D327/04Five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
OA56649A 1977-11-09 1978-11-02 Nouvelles pipérazines disubstituées, leurs procédés de préparation et les compositions pharmaceutiques les renfermant. OA06083A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4664677 1977-11-09

Publications (1)

Publication Number Publication Date
OA06083A true OA06083A (fr) 1981-06-30

Family

ID=10442057

Family Applications (1)

Application Number Title Priority Date Filing Date
OA56649A OA06083A (fr) 1977-11-09 1978-11-02 Nouvelles pipérazines disubstituées, leurs procédés de préparation et les compositions pharmaceutiques les renfermant.

Country Status (14)

Country Link
US (1) US4260610A (de)
JP (1) JPS5481284A (de)
AR (3) AR220730A1 (de)
AU (1) AU4140778A (de)
BE (1) BE871857A (de)
CA (1) CA1117944A (de)
DE (1) DE2848139A1 (de)
ES (1) ES474896A1 (de)
FR (1) FR2408605A1 (de)
IL (1) IL55894A (de)
IT (1) IT1109266B (de)
NL (1) NL7811135A (de)
OA (1) OA06083A (de)
ZA (1) ZA786262B (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3321969A1 (de) * 1983-06-18 1984-12-20 Troponwerke GmbH & Co KG, 5000 Köln 2-pyrimidinyl-1-piperazin-derivate, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
DE3902316A1 (de) * 1989-01-26 1990-08-02 Lentia Gmbh Neue piperazinylalkyl-3(2h)-pyridazinone, verfahren zu ihrer herstellung und ihre verwendung als blutdrucksenkende mittel
US4988699A (en) * 1989-03-14 1991-01-29 Warner-Lambert Company Substituted tetrahydrobenzothiazoles as dopaminergic agents
US4954503A (en) * 1989-09-11 1990-09-04 Hoechst-Roussel Pharmaceuticals, Inc. 3-(1-substituted-4-piperazinyl)-1H-indazoles
FR2671350A1 (fr) * 1991-01-08 1992-07-10 Adir Nouveaux derives de benzisoxazole et de benzisothiazole, leur procede de preparation, et les compositions pharmaceutiques les renfermant.
US5859246A (en) 1997-01-30 1999-01-12 Neurogen Corporation 1-phenyl-4-benzylpiperazines: dopamine receptor subtype specific ligands
RU2576037C1 (ru) * 2014-11-28 2016-02-27 Закрытое акционерное общество "Исследовательский институт Химического разнообразия" ЗАО "ИИХР" Замещенные 4-{ [4-(3,3-диоксидо-1,3-бензоксатиол-6-ил)арилокси]метил} пиперидины как агонисты рецепторов gpr119, фармацевтическая композиция, способы их получения и применения
JP2019517563A (ja) * 2016-06-09 2019-06-24 プラマーナ ファーマシューティカルズ インコーポレイテッド ベンゾ[d][1,3]オキサチオール、ベンゾ[d][1,3]オキサチオール3−オキシドまたはベンゾ[d][1,3]オキサチオール3,3−ジオキシドを含有する化合物およびGタンパク質共役型受容体119のアゴニストとしてのその方法/使用
US11358956B2 (en) 2017-11-30 2022-06-14 Pramana Pharmaceuticals Inc. Compounds containing polysubstituted benzo[d][1,3]oxathiole, benzo[d][1,3]oxathiole 3-oxide or benzo[d][1,3]oxathiole 3,3-dioxide and methods/uses thereof as agonists of G protein-coupled receptor 119

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2459367A (en) * 1947-11-12 1949-01-18 American Cyanamid Co 1,4-di (heterocyclic substituted) piperazines
US2561036A (en) * 1948-06-07 1951-07-17 Noel S Sodders Thread-cutting sheet metal nut
NL127996C (de) * 1963-11-19
DE1595923A1 (de) * 1965-02-20 1969-11-27 Merck Ag E 1-Aralkyl-4-(thiazolyl-2)-piperazine und Verfahren zu ihrer Herstellung
GB1187680A (en) * 1967-11-15 1970-04-15 Science Union & Cie New Heterocyclic Substituted Piperazines
GB1407552A (en) * 1973-04-02 1975-09-24 Science Union & Cie Disubstituted piperazines processes for their preparation and pharmaceutical compositions containing them
GB1432660A (en) * 1973-10-30 1976-04-22 Science Union & Cie Piperazine derivatives processes for their preparation and and pharamacueitcal compositions containing them

Also Published As

Publication number Publication date
CA1117944A (fr) 1982-02-09
FR2408605B1 (de) 1982-02-05
JPS6136755B2 (de) 1986-08-20
AR220794A1 (es) 1980-11-28
DE2848139A1 (de) 1979-05-10
US4260610A (en) 1981-04-07
AR220793A1 (es) 1980-11-28
IT7851814A0 (it) 1978-11-08
AU4140778A (en) 1979-05-17
NL7811135A (nl) 1979-05-11
FR2408605A1 (fr) 1979-06-08
IL55894A (en) 1981-09-13
BE871857A (fr) 1979-05-08
JPS5481284A (en) 1979-06-28
ZA786262B (en) 1979-10-31
IT1109266B (it) 1985-12-16
ES474896A1 (es) 1979-03-16
IL55894A0 (en) 1979-01-31
AR220730A1 (es) 1980-11-28

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