OA00943A - Procédé pour la préparation de dérivés de benzodiazépine. - Google Patents

Procédé pour la préparation de dérivés de benzodiazépine.

Info

Publication number
OA00943A
OA00943A OA51038A OA51038A OA00943A OA 00943 A OA00943 A OA 00943A OA 51038 A OA51038 A OA 51038A OA 51038 A OA51038 A OA 51038A OA 00943 A OA00943 A OA 00943A
Authority
OA
OAPI
Prior art keywords
preparation
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
OA51038A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of OA00943A publication Critical patent/OA00943A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
OA51038A 1963-10-29 1964-12-26 Procédé pour la préparation de dérivés de benzodiazépine. OA00943A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US319673A US3312688A (en) 1963-10-29 1963-10-29 Process for preparing 2-aminobenzodiazepines

Publications (1)

Publication Number Publication Date
OA00943A true OA00943A (fr) 1968-03-22

Family

ID=23243220

Family Applications (1)

Application Number Title Priority Date Filing Date
OA51038A OA00943A (fr) 1963-10-29 1964-12-26 Procédé pour la préparation de dérivés de benzodiazépine.

Country Status (14)

Country Link
US (1) US3312688A (fr)
BE (1) BE654924A (fr)
BR (1) BR6463736D0 (fr)
CH (1) CH443319A (fr)
DE (2) DE1445910A1 (fr)
DK (1) DK114271B (fr)
ES (1) ES305413A1 (fr)
FR (1) FR1442311A (fr)
GB (1) GB1058739A (fr)
IL (1) IL22192A (fr)
NL (3) NL139527B (fr)
NO (1) NO118910B (fr)
OA (1) OA00943A (fr)
SE (2) SE355580B (fr)

Also Published As

Publication number Publication date
IL22192A (en) 1968-01-25
ES305413A1 (es) 1965-05-01
NL6412484A (fr) 1965-05-03
NL139527B (nl) 1973-08-15
BR6463736D0 (pt) 1973-07-17
DE1445910A1 (de) 1969-01-23
DK114271B (da) 1969-06-16
US3312688A (en) 1967-04-04
SE329625B (fr) 1970-10-19
BE654924A (fr) 1965-04-28
NL7115681A (fr) 1972-02-25
SE355580B (fr) 1973-04-30
FR1442311A (fr) 1966-06-17
CH443319A (de) 1967-09-15
NO118910B (fr) 1970-03-02
GB1058739A (en) 1967-02-15
NL7115680A (fr) 1972-02-25
DE1695217A1 (de) 1972-02-17

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