NZ531700A - 1-Glyoxylamide indolizines for treating cancer - Google Patents

1-Glyoxylamide indolizines for treating cancer

Info

Publication number
NZ531700A
NZ531700A NZ531700A NZ53170002A NZ531700A NZ 531700 A NZ531700 A NZ 531700A NZ 531700 A NZ531700 A NZ 531700A NZ 53170002 A NZ53170002 A NZ 53170002A NZ 531700 A NZ531700 A NZ 531700A
Authority
NZ
New Zealand
Prior art keywords
substituted
group
alkyl
unsubstituted
ring
Prior art date
Application number
NZ531700A
Other languages
English (en)
Inventor
Keizo Koya
Lijun Sun
Mitsunori Ono
Weiwen Ying
Hao Li
Original Assignee
Synta Pharmaceuticals Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synta Pharmaceuticals Corp filed Critical Synta Pharmaceuticals Corp
Publication of NZ531700A publication Critical patent/NZ531700A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NZ531700A 2001-09-13 2002-09-13 1-Glyoxylamide indolizines for treating cancer NZ531700A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32202001P 2001-09-13 2001-09-13
PCT/US2002/029154 WO2003022846A1 (en) 2001-09-13 2002-09-13 1-glyoxlylamide indolizines for treating cancer

Publications (1)

Publication Number Publication Date
NZ531700A true NZ531700A (en) 2006-10-27

Family

ID=23253054

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ531700A NZ531700A (en) 2001-09-13 2002-09-13 1-Glyoxylamide indolizines for treating cancer

Country Status (19)

Country Link
US (2) US6861436B2 (enExample)
EP (1) EP1432709B8 (enExample)
JP (1) JP2005504795A (enExample)
KR (1) KR20040053125A (enExample)
CN (1) CN1568324A (enExample)
AT (1) ATE300542T1 (enExample)
AU (1) AU2002333626B2 (enExample)
BR (1) BR0212794A (enExample)
CA (1) CA2459886A1 (enExample)
DE (1) DE60205265T2 (enExample)
ES (1) ES2245747T3 (enExample)
IL (1) IL160810A0 (enExample)
IS (1) IS7176A (enExample)
MX (1) MXPA04002323A (enExample)
NO (1) NO20041035L (enExample)
NZ (1) NZ531700A (enExample)
PT (1) PT1432709E (enExample)
WO (1) WO2003022846A1 (enExample)
ZA (1) ZA200401996B (enExample)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040116462A1 (en) * 2002-12-12 2004-06-17 Mitsunori Ono Indolizine compounds
PT1432709E (pt) * 2001-09-13 2005-10-31 Synta Pharmaceuticals Corp Indolizinas de 1-glioxilamida para o trtamento do cancro
JP2006504692A (ja) * 2002-09-13 2006-02-09 シンタ ファーマシューティカルズ コーポレーション インドリジンの合成方法
DE10318611A1 (de) 2003-04-24 2004-11-11 Elbion Ag 4-, 6- oder 7-Hydroxyindole mit N-Oxidgruppen und deren Verwendung als Therapeutika
WO2005099824A1 (en) * 2004-03-30 2005-10-27 Synta Pharmaceuticals, Corp. 1-glyoxylamide indolizines for treating lung and ovarian cancer
GB0413605D0 (en) 2004-06-17 2004-07-21 Addex Pharmaceuticals Sa Novel compounds
US20070293456A9 (en) * 2004-12-30 2007-12-20 Anthony Hayford Method for the synthesis of 3-substituted indolizine and benzoindolizine compounds
WO2006128184A2 (en) * 2005-05-20 2006-11-30 Alantos-Pharmaceuticals, Inc. Pyrimidine or triazine fused bicyclic metalloprotease inhibitors
US20070155738A1 (en) 2005-05-20 2007-07-05 Alantos Pharmaceuticals, Inc. Heterobicyclic metalloprotease inhibitors
CA2733247C (en) * 2008-08-14 2018-04-03 Beta Pharma Canada Inc. Heterocyclic amide derivatives as ep4 receptor antagonists
EP4008327A1 (en) 2009-04-29 2022-06-08 Amarin Pharmaceuticals Ireland Limited Pharmaceutical compositions comprising epa and a cardiovascular agent and methods of using the same
AR077428A1 (es) * 2009-07-29 2011-08-24 Sanofi Aventis (aza) indolizinacarboxamidas ciclicas su preparacion y su uso como agentes farmaceuticos
CN113603694B (zh) * 2021-07-16 2022-07-22 浙江工业大学 一种1,2-二酮类化合物及其制备方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2287706A (en) * 1994-03-21 1995-09-27 Fujisawa Pharmaceutical Co Indolizine derivatives
FR2757166B1 (fr) * 1996-12-12 1999-01-29 Rhone Poulenc Rorer Sa Derives du pyrrole, leur preparation et les compositions pharmaceutiques qui les contiennent
WO1998047507A1 (en) * 1997-04-24 1998-10-29 Shionogi & Co., Ltd. Method for the treatment of stroke using n-heterocyclic glyoxylamide compounds
US6472389B1 (en) 1998-05-21 2002-10-29 Shionogi & Co., Ltd. Pyrrolo[1,2-b] pyridazine derivatives having sPLA2 inhibitory effect
CA2346334A1 (en) 1998-10-14 2000-04-20 Shionogi & Co., Ltd. Composition for treating or preventing ischemia reperfusion injury
US6461538B2 (en) * 1999-12-16 2002-10-08 Fuji Photo Film Co., Ltd. Production process for indolizine compounds and their use in organic light-emitting devices
PT1432709E (pt) * 2001-09-13 2005-10-31 Synta Pharmaceuticals Corp Indolizinas de 1-glioxilamida para o trtamento do cancro
US20040116462A1 (en) * 2002-12-12 2004-06-17 Mitsunori Ono Indolizine compounds

Also Published As

Publication number Publication date
IL160810A0 (en) 2004-08-31
CA2459886A1 (en) 2003-03-20
NO20041035L (no) 2004-04-30
AU2002333626B2 (en) 2006-06-29
DE60205265T2 (de) 2006-03-30
KR20040053125A (ko) 2004-06-23
ZA200401996B (en) 2005-05-31
MXPA04002323A (es) 2005-04-08
EP1432709B1 (en) 2005-07-27
EP1432709A1 (en) 2004-06-30
US6861436B2 (en) 2005-03-01
JP2005504795A (ja) 2005-02-17
EP1432709B8 (en) 2005-11-02
IS7176A (is) 2004-03-11
ES2245747T3 (es) 2006-01-16
WO2003022846A1 (en) 2003-03-20
HK1063322A1 (en) 2004-12-24
DE60205265D1 (de) 2005-09-01
PT1432709E (pt) 2005-10-31
BR0212794A (pt) 2004-10-05
CN1568324A (zh) 2005-01-19
ATE300542T1 (de) 2005-08-15
US20030153759A1 (en) 2003-08-14
US20040214850A1 (en) 2004-10-28

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