IS7176A - 1-Glýoxlýlamíd-indólízín til meðhöndlunar á krabbameini - Google Patents

1-Glýoxlýlamíd-indólízín til meðhöndlunar á krabbameini

Info

Publication number
IS7176A
IS7176A IS7176A IS7176A IS7176A IS 7176 A IS7176 A IS 7176A IS 7176 A IS7176 A IS 7176A IS 7176 A IS7176 A IS 7176A IS 7176 A IS7176 A IS 7176A
Authority
IS
Iceland
Prior art keywords
substituted
group
unsubstituted
independently
aryl group
Prior art date
Application number
IS7176A
Other languages
English (en)
Inventor
Koya Keizo
Sun Lijun
Ono Mitsunori
Ying Weiwen
Li Hao
Original Assignee
Synta Pharmaceuticals Corp.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synta Pharmaceuticals Corp. filed Critical Synta Pharmaceuticals Corp.
Publication of IS7176A publication Critical patent/IS7176A/is

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IS7176A 2001-09-13 2004-03-11 1-Glýoxlýlamíd-indólízín til meðhöndlunar á krabbameini IS7176A (is)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32202001P 2001-09-13 2001-09-13
PCT/US2002/029154 WO2003022846A1 (en) 2001-09-13 2002-09-13 1-glyoxlylamide indolizines for treating cancer

Publications (1)

Publication Number Publication Date
IS7176A true IS7176A (is) 2004-03-11

Family

ID=23253054

Family Applications (1)

Application Number Title Priority Date Filing Date
IS7176A IS7176A (is) 2001-09-13 2004-03-11 1-Glýoxlýlamíd-indólízín til meðhöndlunar á krabbameini

Country Status (20)

Country Link
US (2) US6861436B2 (is)
EP (1) EP1432709B8 (is)
JP (1) JP2005504795A (is)
KR (1) KR20040053125A (is)
CN (1) CN1568324A (is)
AT (1) ATE300542T1 (is)
AU (1) AU2002333626B2 (is)
BR (1) BR0212794A (is)
CA (1) CA2459886A1 (is)
DE (1) DE60205265T2 (is)
ES (1) ES2245747T3 (is)
HK (1) HK1063322A1 (is)
IL (1) IL160810A0 (is)
IS (1) IS7176A (is)
MX (1) MXPA04002323A (is)
NO (1) NO20041035L (is)
NZ (1) NZ531700A (is)
PT (1) PT1432709E (is)
WO (1) WO2003022846A1 (is)
ZA (1) ZA200401996B (is)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040116462A1 (en) * 2002-12-12 2004-06-17 Mitsunori Ono Indolizine compounds
BR0212794A (pt) * 2001-09-13 2004-10-05 Synta Pharmaceuticals Corp Composto de 1-glioxililamida indolizina e seu uso
WO2004024727A2 (en) * 2002-09-13 2004-03-25 Synta Pharmaceuticals Corp. Synthesis of indolizines
DE10318611A1 (de) 2003-04-24 2004-11-11 Elbion Ag 4-, 6- oder 7-Hydroxyindole mit N-Oxidgruppen und deren Verwendung als Therapeutika
WO2005099824A1 (en) * 2004-03-30 2005-10-27 Synta Pharmaceuticals, Corp. 1-glyoxylamide indolizines for treating lung and ovarian cancer
GB0413605D0 (en) 2004-06-17 2004-07-21 Addex Pharmaceuticals Sa Novel compounds
US20070293456A9 (en) * 2004-12-30 2007-12-20 Anthony Hayford Method for the synthesis of 3-substituted indolizine and benzoindolizine compounds
KR20080087070A (ko) * 2005-05-20 2008-09-30 알란토스 파마슈티컬즈 홀딩, 인코포레이티드 피리미딘 또는 트리아진 융합된 비시클릭 메탈로프로테아제억제제
US20070155738A1 (en) * 2005-05-20 2007-07-05 Alantos Pharmaceuticals, Inc. Heterobicyclic metalloprotease inhibitors
CA2733247C (en) * 2008-08-14 2018-04-03 Beta Pharma Canada Inc. Heterocyclic amide derivatives as ep4 receptor antagonists
NZ624963A (en) 2009-04-29 2016-07-29 Amarin Pharmaceuticals Ie Ltd Pharmaceutical compositions comprising epa and a cardiovascular agent and methods of using the same
AR077428A1 (es) * 2009-07-29 2011-08-24 Sanofi Aventis (aza) indolizinacarboxamidas ciclicas su preparacion y su uso como agentes farmaceuticos
CN113603694B (zh) * 2021-07-16 2022-07-22 浙江工业大学 一种1,2-二酮类化合物及其制备方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2287706A (en) 1994-03-21 1995-09-27 Fujisawa Pharmaceutical Co Indolizine derivatives
FR2757166B1 (fr) * 1996-12-12 1999-01-29 Rhone Poulenc Rorer Sa Derives du pyrrole, leur preparation et les compositions pharmaceutiques qui les contiennent
WO1998047507A1 (en) 1997-04-24 1998-10-29 Shionogi & Co., Ltd. Method for the treatment of stroke using n-heterocyclic glyoxylamide compounds
CA2332528A1 (en) 1998-05-21 1999-11-25 Shionogi & Co., Ltd. Pyrrolo[1,2-b]pyridazine spla2 inhibitory
CA2346334A1 (en) 1998-10-14 2000-04-20 Shionogi & Co., Ltd. Composition for treating or preventing ischemia reperfusion injury
US6461538B2 (en) * 1999-12-16 2002-10-08 Fuji Photo Film Co., Ltd. Production process for indolizine compounds and their use in organic light-emitting devices
BR0212794A (pt) * 2001-09-13 2004-10-05 Synta Pharmaceuticals Corp Composto de 1-glioxililamida indolizina e seu uso
US20040116462A1 (en) * 2002-12-12 2004-06-17 Mitsunori Ono Indolizine compounds

Also Published As

Publication number Publication date
PT1432709E (pt) 2005-10-31
US20040214850A1 (en) 2004-10-28
MXPA04002323A (es) 2005-04-08
ZA200401996B (en) 2005-05-31
AU2002333626B2 (en) 2006-06-29
DE60205265D1 (de) 2005-09-01
EP1432709B8 (en) 2005-11-02
KR20040053125A (ko) 2004-06-23
HK1063322A1 (en) 2004-12-24
BR0212794A (pt) 2004-10-05
CA2459886A1 (en) 2003-03-20
EP1432709A1 (en) 2004-06-30
EP1432709B1 (en) 2005-07-27
IL160810A0 (en) 2004-08-31
DE60205265T2 (de) 2006-03-30
CN1568324A (zh) 2005-01-19
JP2005504795A (ja) 2005-02-17
NZ531700A (en) 2006-10-27
US6861436B2 (en) 2005-03-01
NO20041035L (no) 2004-04-30
US20030153759A1 (en) 2003-08-14
WO2003022846A1 (en) 2003-03-20
ATE300542T1 (de) 2005-08-15
ES2245747T3 (es) 2006-01-16

Similar Documents

Publication Publication Date Title
IS7176A (is) 1-Glýoxlýlamíd-indólízín til meðhöndlunar á krabbameini
NO20050418L (no) Kondenserte pyridiner og pyrimidiner med TIE2(TEK) aktivitet
AR043158A1 (es) Compuestos activadores de glucoquinasa de amida tri(ciclo) sustituidos, procedimientos para su preparacion y composiciones farmaceuticas que los contienen
CO5590895A2 (es) Derivados de sulfonamidas, su preparacion y su aplicacion como medicamentos
ATE326454T1 (de) Neue bernsteinsäure derivative als cysteine- protease-inhibitoren
PE20030746A1 (es) DERIVADOS DE PIRIDO [2,1-a] ISOQUINOLINA
CO4970713A1 (es) Derivados de carboxamidotiazoles, su preparacion, composiciones farmaceuticas que los contienen
NO20066015L (no) Fuserte heterosykliske forbindelser
NO20052781L (no) Forbindelser og prosesser
BRPI0506927A (pt) compostos orgánicos
AR054386A1 (es) Moduladores de quinasas con estructuras de alquiloquinolina y alquilquinazolina
CO5690577A2 (es) Derivados de imidazoquinolina como ligandos receptores de adenosina a3
WO2008136444A1 (ja) 縮合複素環誘導体
ES2038678T3 (es) Procedimiento para la preparacion de n-(2-alquil-3-mercapto-glutaril)-alfamino-acidos.
DK471586A (da) 3-vinyl- og 3-ethynyl-beta-carbolinderivater, deres fremstilling og deres anvendelse som laegemiddel
ES2130438T3 (es) Derivados de imidazo(1,2-a)pirazin-4-ona, su preparacion y los medicamentos que les contienen.
CA2461060A1 (en) Method for preparing pyrimidinone compound and pharmaceutically acceptable salts thereof
HUP0201475A2 (hu) Heteroarilamidin-, metilamidin- és guanidinszármazékok, előállításuk és alkalmazásuk, valamint e vegyületeket tartalmazó gyógyászati készítmények
DK118287D0 (da) Heteroaryloxy-beta-carbolinderivater, deres fremstilling og deres anvendelse som laegemiddel
TW200602039A (en) 1-Glyoxylamide indolizines for treating lung and ovarian cancer
DK0712395T3 (da) Fremgangsmåde til fremstilling af fluoralkenylthio-heterocykliske derivater
DK1303512T3 (da) Fremgangsmåde til fremstilling af arylacetylaminothiazoler
ES2058064T3 (es) Derivados de beta-carbolina sustituidos con fenoxi, su preparacion y su utilizacion como medicamentos.
AR043487A1 (es) Heterociclos fusionados de pirimidina y usos de los mismos
AR036735A1 (es) Derivados de 5-metoxi-8-aril-[1,2,4]triazolo[1,5-a]piridina