NO924126D0 - 3-indolylthioacetatderivater - Google Patents
3-indolylthioacetatderivaterInfo
- Publication number
- NO924126D0 NO924126D0 NO1992924126A NO924126A NO924126D0 NO 924126 D0 NO924126 D0 NO 924126D0 NO 1992924126 A NO1992924126 A NO 1992924126A NO 924126 A NO924126 A NO 924126A NO 924126 D0 NO924126 D0 NO 924126D0
- Authority
- NO
- Norway
- Prior art keywords
- indolylthioacetatderivater
- directed
- present
- new class
- nmda antagonists
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US07/514,074 US5051442A (en) | 1990-04-25 | 1990-04-25 | 3-indolyl thioacetate derivatives and NMDA receptor antagonistic use thereof |
PCT/US1991/002179 WO1991016307A1 (en) | 1990-04-25 | 1991-03-28 | 3-indolyl thioacetate derivatives |
Publications (4)
Publication Number | Publication Date |
---|---|
NO924126D0 true NO924126D0 (no) | 1992-10-23 |
NO924126L NO924126L (no) | 1992-10-23 |
NO178857B NO178857B (no) | 1996-03-11 |
NO178857C NO178857C (no) | 1996-06-19 |
Family
ID=24045696
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO924126A NO178857C (no) | 1990-04-25 | 1992-10-23 | Analogifremgangsmåte for fremstilling av terapeutisk aktive 3-indolylthioacetatderivater |
Country Status (14)
Country | Link |
---|---|
US (1) | US5051442A (no) |
EP (1) | EP0526478B1 (no) |
JP (1) | JP3006881B2 (no) |
KR (1) | KR0178281B1 (no) |
AT (1) | ATE119882T1 (no) |
AU (1) | AU646251B2 (no) |
CA (1) | CA2081330C (no) |
DE (1) | DE69108234T2 (no) |
DK (1) | DK0526478T3 (no) |
ES (1) | ES2072607T3 (no) |
FI (1) | FI98454C (no) |
HU (1) | HU213205B (no) |
NO (1) | NO178857C (no) |
WO (1) | WO1991016307A1 (no) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5189054A (en) * | 1990-11-02 | 1993-02-23 | Merrell Dow Pharmaceuticals Inc. | 3-amidoindolyl derivatives and pharmaceutical compositions thereof |
US5318985A (en) * | 1991-12-20 | 1994-06-07 | Merrell Dow Pharmaceuticals Inc. | Potentiation of NMDA antagonists |
USRE39300E1 (en) | 1993-01-28 | 2006-09-19 | Virginia Commonwealth University Medical College Of Virginia | Inhibiting the development of tolerance to and/or dependence on an addictive substance |
US5321012A (en) * | 1993-01-28 | 1994-06-14 | Virginia Commonwealth University Medical College | Inhibiting the development of tolerance to and/or dependence on a narcotic addictive substance |
GB9311948D0 (en) * | 1993-06-10 | 1993-07-28 | Zeneca Ltd | Substituted nitrogen heterocycles |
US5424329A (en) * | 1993-08-18 | 1995-06-13 | Warner-Lambert Company | Indole-2-carboxamides as inhibitors of cell adhesion |
US5801168A (en) * | 1994-06-09 | 1998-09-01 | Zeneca Limited | Substituted nitrogen heterocycles |
SK281737B6 (sk) * | 1996-04-19 | 2001-07-10 | American Home Products Corporation | 2-fenylindolové zlúčeniny, farmaceutický prostriedok s ich obsahom a ich použitie |
US6069153A (en) * | 1998-05-12 | 2000-05-30 | American Home Products Corporation | Indenoindoles and benzocarbazoles as estrogenic agents |
US6479535B1 (en) | 1998-05-15 | 2002-11-12 | Wyeth | 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indole and estrogen formulations |
US6159959A (en) * | 1999-05-06 | 2000-12-12 | American Home Products Corporation | Combined estrogen and antiestrogen therapy |
AR081930A1 (es) | 2010-06-16 | 2012-10-31 | Ardea Biosciences Inc | Compuestos de tioacetato |
JP5709146B2 (ja) | 2010-06-16 | 2015-04-30 | アルデア バイオサイエンシーズ インク. | フェニルチオ酢酸化合物、組成物、および、その使用方法 |
UA114304C2 (uk) | 2011-11-03 | 2017-05-25 | Ардеа Біосайєнсіс, Інк. | Спосіб зниження сироваткових рівнів сечової кислоти у людини |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4675332A (en) * | 1984-12-10 | 1987-06-23 | Warner-Lambert Company | Acidic tetrazolyl substituted indole compounds and their use as antiallergy agents |
NZ222878A (en) * | 1986-12-17 | 1991-02-26 | Merck Frosst Canada Inc | 3-hetero-substituted-n-benzyl-indole derivatives, and pharmaceutical compositions |
US4960786A (en) * | 1989-04-24 | 1990-10-02 | Merrell Dow Pharmaceuticals Inc. | Excitatory amino acid antagonists |
JPH0347123A (ja) * | 1989-05-05 | 1991-02-28 | G D Searle & Co | インドール―2―カルボキシレート化合物類を含有するcns疾患治療用組成物 |
-
1990
- 1990-04-25 US US07/514,074 patent/US5051442A/en not_active Expired - Fee Related
-
1991
- 1991-03-28 DE DE69108234T patent/DE69108234T2/de not_active Expired - Fee Related
- 1991-03-28 EP EP91907138A patent/EP0526478B1/en not_active Expired - Lifetime
- 1991-03-28 KR KR1019920702634A patent/KR0178281B1/ko not_active IP Right Cessation
- 1991-03-28 CA CA002081330A patent/CA2081330C/en not_active Expired - Fee Related
- 1991-03-28 AU AU76500/91A patent/AU646251B2/en not_active Ceased
- 1991-03-28 DK DK91907138.1T patent/DK0526478T3/da active
- 1991-03-28 JP JP3507419A patent/JP3006881B2/ja not_active Expired - Fee Related
- 1991-03-28 ES ES91907138T patent/ES2072607T3/es not_active Expired - Lifetime
- 1991-03-28 WO PCT/US1991/002179 patent/WO1991016307A1/en active IP Right Grant
- 1991-03-28 HU HU9203336A patent/HU213205B/hu not_active IP Right Cessation
- 1991-03-28 AT AT91907138T patent/ATE119882T1/de not_active IP Right Cessation
-
1992
- 1992-10-14 FI FI924642A patent/FI98454C/fi active
- 1992-10-23 NO NO924126A patent/NO178857C/no not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
FI98454B (fi) | 1997-03-14 |
HU9203336D0 (en) | 1993-01-28 |
ES2072607T3 (es) | 1995-07-16 |
US5051442A (en) | 1991-09-24 |
AU7650091A (en) | 1991-11-11 |
DE69108234T2 (de) | 1995-08-24 |
HUT64744A (en) | 1994-02-28 |
DK0526478T3 (da) | 1995-05-29 |
CA2081330A1 (en) | 1991-10-26 |
CA2081330C (en) | 2002-02-05 |
KR0178281B1 (ko) | 1999-03-20 |
WO1991016307A1 (en) | 1991-10-31 |
KR937000438A (ko) | 1993-03-15 |
FI924642A (fi) | 1992-10-14 |
ATE119882T1 (de) | 1995-04-15 |
EP0526478B1 (en) | 1995-03-15 |
NO924126L (no) | 1992-10-23 |
FI924642A0 (fi) | 1992-10-14 |
JP3006881B2 (ja) | 2000-02-07 |
FI98454C (fi) | 1997-06-25 |
HU213205B (en) | 1997-03-28 |
NO178857C (no) | 1996-06-19 |
NO178857B (no) | 1996-03-11 |
EP0526478A1 (en) | 1993-02-10 |
AU646251B2 (en) | 1994-02-17 |
DE69108234D1 (en) | 1995-04-20 |
JPH07500567A (ja) | 1995-01-19 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM1K | Lapsed by not paying the annual fees |
Free format text: LAPSED IN SEPTEMBER 2003 |