FI98454B - Menetelmä terapeuttisesti aktiivisten 3-indolyylitioasetaattijohdannaisten valmistamiseksi - Google Patents
Menetelmä terapeuttisesti aktiivisten 3-indolyylitioasetaattijohdannaisten valmistamiseksiInfo
- Publication number
- FI98454B FI98454B FI924642A FI924642A FI98454B FI 98454 B FI98454 B FI 98454B FI 924642 A FI924642 A FI 924642A FI 924642 A FI924642 A FI 924642A FI 98454 B FI98454 B FI 98454B
- Authority
- FI
- Finland
- Prior art keywords
- derivatives
- indolylthioacetate
- preparation
- therapeutically active
- directed
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Lubricants (AREA)
- Hard Magnetic Materials (AREA)
- Plural Heterocyclic Compounds (AREA)
- Catalysts (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Polyesters Or Polycarbonates (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US07/514,074 US5051442A (en) | 1990-04-25 | 1990-04-25 | 3-indolyl thioacetate derivatives and NMDA receptor antagonistic use thereof |
US51407490 | 1990-04-25 | ||
PCT/US1991/002179 WO1991016307A1 (en) | 1990-04-25 | 1991-03-28 | 3-indolyl thioacetate derivatives |
US9102179 | 1991-03-28 |
Publications (4)
Publication Number | Publication Date |
---|---|
FI924642A0 FI924642A0 (fi) | 1992-10-14 |
FI924642A FI924642A (fi) | 1992-10-14 |
FI98454B true FI98454B (fi) | 1997-03-14 |
FI98454C FI98454C (fi) | 1997-06-25 |
Family
ID=24045696
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI924642A FI98454C (fi) | 1990-04-25 | 1992-10-14 | Menetelmä terapeuttisesti aktiivisten 3-indolyylitioasetaattijohdannaisten valmistamiseksi |
Country Status (14)
Country | Link |
---|---|
US (1) | US5051442A (fi) |
EP (1) | EP0526478B1 (fi) |
JP (1) | JP3006881B2 (fi) |
KR (1) | KR0178281B1 (fi) |
AT (1) | ATE119882T1 (fi) |
AU (1) | AU646251B2 (fi) |
CA (1) | CA2081330C (fi) |
DE (1) | DE69108234T2 (fi) |
DK (1) | DK0526478T3 (fi) |
ES (1) | ES2072607T3 (fi) |
FI (1) | FI98454C (fi) |
HU (1) | HU213205B (fi) |
NO (1) | NO178857C (fi) |
WO (1) | WO1991016307A1 (fi) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5189054A (en) * | 1990-11-02 | 1993-02-23 | Merrell Dow Pharmaceuticals Inc. | 3-amidoindolyl derivatives and pharmaceutical compositions thereof |
US5318985A (en) * | 1991-12-20 | 1994-06-07 | Merrell Dow Pharmaceuticals Inc. | Potentiation of NMDA antagonists |
US5321012A (en) * | 1993-01-28 | 1994-06-14 | Virginia Commonwealth University Medical College | Inhibiting the development of tolerance to and/or dependence on a narcotic addictive substance |
USRE39300E1 (en) | 1993-01-28 | 2006-09-19 | Virginia Commonwealth University Medical College Of Virginia | Inhibiting the development of tolerance to and/or dependence on an addictive substance |
GB9311948D0 (en) * | 1993-06-10 | 1993-07-28 | Zeneca Ltd | Substituted nitrogen heterocycles |
US5424329A (en) * | 1993-08-18 | 1995-06-13 | Warner-Lambert Company | Indole-2-carboxamides as inhibitors of cell adhesion |
US5801168A (en) * | 1994-06-09 | 1998-09-01 | Zeneca Limited | Substituted nitrogen heterocycles |
ATE206701T1 (de) * | 1996-04-19 | 2001-10-15 | American Home Prod | Östrogene verbindungen |
US6069153A (en) * | 1998-05-12 | 2000-05-30 | American Home Products Corporation | Indenoindoles and benzocarbazoles as estrogenic agents |
US6479535B1 (en) | 1998-05-15 | 2002-11-12 | Wyeth | 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indole and estrogen formulations |
US6159959A (en) * | 1999-05-06 | 2000-12-12 | American Home Products Corporation | Combined estrogen and antiestrogen therapy |
AR081930A1 (es) | 2010-06-16 | 2012-10-31 | Ardea Biosciences Inc | Compuestos de tioacetato |
BR112012032193A2 (pt) | 2010-06-16 | 2019-09-24 | Ardea Biosciences Inc | composto, composiçoes e métodos de uso de feniltioacetato |
SG11201402016PA (en) | 2011-11-03 | 2014-05-29 | Ardea Biosciences Inc | 3,4-di-substituted pyridine compound, methods of using and compositions comprising the same |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4675332A (en) * | 1984-12-10 | 1987-06-23 | Warner-Lambert Company | Acidic tetrazolyl substituted indole compounds and their use as antiallergy agents |
IL84796A (en) * | 1986-12-17 | 1992-03-29 | Merck Frosst Canada Inc | Substituted n-benzyl-indoles and pharmaceutical compositions containing them |
US4960786A (en) * | 1989-04-24 | 1990-10-02 | Merrell Dow Pharmaceuticals Inc. | Excitatory amino acid antagonists |
PT93943A (pt) * | 1989-05-05 | 1991-02-08 | Searle & Co | Processo para a preparacao de composicoes contendo compostos indole-2-carboxilato para tratamento de perturbacoes do snc |
-
1990
- 1990-04-25 US US07/514,074 patent/US5051442A/en not_active Expired - Fee Related
-
1991
- 1991-03-28 DE DE69108234T patent/DE69108234T2/de not_active Expired - Fee Related
- 1991-03-28 DK DK91907138.1T patent/DK0526478T3/da active
- 1991-03-28 ES ES91907138T patent/ES2072607T3/es not_active Expired - Lifetime
- 1991-03-28 CA CA002081330A patent/CA2081330C/en not_active Expired - Fee Related
- 1991-03-28 WO PCT/US1991/002179 patent/WO1991016307A1/en active IP Right Grant
- 1991-03-28 AU AU76500/91A patent/AU646251B2/en not_active Ceased
- 1991-03-28 AT AT91907138T patent/ATE119882T1/de not_active IP Right Cessation
- 1991-03-28 KR KR1019920702634A patent/KR0178281B1/ko not_active IP Right Cessation
- 1991-03-28 JP JP3507419A patent/JP3006881B2/ja not_active Expired - Fee Related
- 1991-03-28 HU HU9203336A patent/HU213205B/hu not_active IP Right Cessation
- 1991-03-28 EP EP91907138A patent/EP0526478B1/en not_active Expired - Lifetime
-
1992
- 1992-10-14 FI FI924642A patent/FI98454C/fi active
- 1992-10-23 NO NO924126A patent/NO178857C/no not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
US5051442A (en) | 1991-09-24 |
CA2081330A1 (en) | 1991-10-26 |
FI924642A0 (fi) | 1992-10-14 |
DE69108234D1 (en) | 1995-04-20 |
JP3006881B2 (ja) | 2000-02-07 |
NO178857C (no) | 1996-06-19 |
FI98454C (fi) | 1997-06-25 |
EP0526478A1 (en) | 1993-02-10 |
HUT64744A (en) | 1994-02-28 |
ES2072607T3 (es) | 1995-07-16 |
CA2081330C (en) | 2002-02-05 |
KR0178281B1 (ko) | 1999-03-20 |
AU646251B2 (en) | 1994-02-17 |
JPH07500567A (ja) | 1995-01-19 |
NO178857B (no) | 1996-03-11 |
FI924642A (fi) | 1992-10-14 |
WO1991016307A1 (en) | 1991-10-31 |
DK0526478T3 (da) | 1995-05-29 |
EP0526478B1 (en) | 1995-03-15 |
HU213205B (en) | 1997-03-28 |
NO924126L (no) | 1992-10-23 |
AU7650091A (en) | 1991-11-11 |
HU9203336D0 (en) | 1993-01-28 |
KR937000438A (ko) | 1993-03-15 |
ATE119882T1 (de) | 1995-04-15 |
DE69108234T2 (de) | 1995-08-24 |
NO924126D0 (no) | 1992-10-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
BB | Publication of examined application |