NO914102D0 - Fremgangsmaate for fremstilling av 5,11-dihydro-6h-dipyrido(3,2-b:2',3'-e)(1,4)diazepiner - Google Patents

Fremgangsmaate for fremstilling av 5,11-dihydro-6h-dipyrido(3,2-b:2',3'-e)(1,4)diazepiner

Info

Publication number
NO914102D0
NO914102D0 NO914102A NO914102A NO914102D0 NO 914102 D0 NO914102 D0 NO 914102D0 NO 914102 A NO914102 A NO 914102A NO 914102 A NO914102 A NO 914102A NO 914102 D0 NO914102 D0 NO 914102D0
Authority
NO
Norway
Prior art keywords
dipyrido
diazepines
dihydro
preparing
procedure
Prior art date
Application number
NO914102A
Other languages
English (en)
Other versions
NO914102L (no
Inventor
Karl G Grozinger
Karl D Hargrave
Julian Adams
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of NO914102D0 publication Critical patent/NO914102D0/no
Publication of NO914102L publication Critical patent/NO914102L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/73—Unsubstituted amino or imino radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C07D213/82—Amides; Imides in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
NO91914102A 1990-10-19 1991-10-18 Fremgangsmaate for fremstilling av 5,11-dihydro-6h-dipyrido(3,2-b:2',3'-e)(1,4)diazepiner NO914102L (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US60045190A 1990-10-19 1990-10-19

Publications (2)

Publication Number Publication Date
NO914102D0 true NO914102D0 (no) 1991-10-18
NO914102L NO914102L (no) 1992-04-21

Family

ID=24403650

Family Applications (1)

Application Number Title Priority Date Filing Date
NO91914102A NO914102L (no) 1990-10-19 1991-10-18 Fremgangsmaate for fremstilling av 5,11-dihydro-6h-dipyrido(3,2-b:2',3'-e)(1,4)diazepiner

Country Status (14)

Country Link
EP (1) EP0482481A1 (no)
JP (1) JPH05163272A (no)
KR (1) KR920008041A (no)
CA (1) CA2052946A1 (no)
CS (1) CS312691A3 (no)
FI (1) FI914923A (no)
HU (1) HU210678B (no)
IE (1) IE913662A1 (no)
NO (1) NO914102L (no)
NZ (1) NZ240279A (no)
PL (1) PL292097A1 (no)
PT (1) PT99273A (no)
YU (1) YU165891A (no)
ZA (1) ZA918335B (no)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5200522A (en) * 1991-06-11 1993-04-06 Boehringer Ingelheim Pharmaceuticals, Inc. Method for preparing 3-amino-2-chloro-4-alkylpyridines
HU213257B (en) * 1991-06-11 1997-04-28 Boehringer Ingelheim Pharma Process for producing 4-alkyl-3-amino-2-chloropyridines
DE4403311C1 (de) * 1994-02-03 1995-04-20 Boehringer Ingelheim Kg Verfahren zur Herstellung von Nevirapine (11-Cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3,2-b:2',3'-e][1,4-diazepin]-6-on)
CN113149896A (zh) * 2021-03-09 2021-07-23 利尔化学股份有限公司 一种3-氨基吡啶的制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2424811C3 (de) * 1974-05-22 1981-08-20 Dr. Karl Thomae Gmbh, 7950 Biberach Pyrido-benzodiazepinone, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel
IT1194766B (it) * 1981-03-10 1988-09-28 Crc Ricerca Chim Processo per la preparazione di 11-(2'-sostituito)-acetil-5,11-diidro-6h-pirido-(2,3-b)(1,4)-benzodiazepin-6-oni
DE3122670A1 (de) * 1981-06-06 1982-12-23 Dr. Karl Thomae Gmbh, 7950 Biberach "neue 1,4,9,10-tetrahydro-pyrazolo(4,3-e) pyrido(3,2-b)(1,4)diazepin-10-one, verfahren zu ihrer herstellung und ihre verwendung zur herstellung von pharmazeutischen wirkstoffen"
DE3222809A1 (de) * 1981-07-15 1983-02-03 Dr. Karl Thomae Gmbh, 7950 Biberach Verfahren zur herstellung von 5,11-dihydro-6h-pyrido(2,3-b)-(1,4) benzodiazepin-6-onen
EP0393529B1 (en) * 1989-04-20 1993-06-30 Boehringer Ingelheim Pharmaceuticals Inc. 5,11-dihydro-6H-dipyrido [3,2-b:2',3'-e][1,4]diazepin-6-ones and their use in the prevention or treatment of AIDS
ATE103918T1 (de) * 1989-06-28 1994-04-15 Boehringer Ingelheim Pharma 5,11-dihydro-6h-dipyrido(3,2-b:2',3'e>(1,4>diazepin-6-one und -thione und ihre verwendung bei der aids-vorbeugung oder behandlung.

Also Published As

Publication number Publication date
AU646096B2 (en) 1994-02-10
NZ240279A (en) 1993-12-23
JPH05163272A (ja) 1993-06-29
FI914923A0 (fi) 1991-10-18
EP0482481A1 (en) 1992-04-29
PT99273A (pt) 1992-08-31
HUT59408A (en) 1992-05-28
HU210678B (en) 1995-06-28
AU8592491A (en) 1992-04-30
CA2052946A1 (en) 1992-04-20
HU913296D0 (en) 1992-01-28
IE913662A1 (en) 1992-04-22
ZA918335B (en) 1992-09-30
KR920008041A (ko) 1992-05-27
YU165891A (sh) 1994-06-10
NO914102L (no) 1992-04-21
FI914923A (fi) 1992-04-20
PL292097A1 (en) 1992-07-13
CS312691A3 (en) 1992-05-13

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