NO842529L - Fremgangsmaate for fremstilling av salter av metyllevallorfanium. - Google Patents

Fremgangsmaate for fremstilling av salter av metyllevallorfanium.

Info

Publication number
NO842529L
NO842529L NO842529A NO842529A NO842529L NO 842529 L NO842529 L NO 842529L NO 842529 A NO842529 A NO 842529A NO 842529 A NO842529 A NO 842529A NO 842529 L NO842529 L NO 842529L
Authority
NO
Norway
Prior art keywords
methyl
anion
levalorphanium
acid
active ingredient
Prior art date
Application number
NO842529A
Other languages
English (en)
Norwegian (no)
Inventor
Alberto Bianchetti
Dino Nisato
Luciano Manara
Roberto Sacilotto
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of NO842529L publication Critical patent/NO842529L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22Bridged ring systems
    • C07D221/28Morphinans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO842529A 1983-06-24 1984-06-22 Fremgangsmaate for fremstilling av salter av metyllevallorfanium. NO842529L (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8310526A FR2547820B1 (fr) 1983-06-24 1983-06-24 Antagonistes peripheriques des opiaces

Publications (1)

Publication Number Publication Date
NO842529L true NO842529L (no) 1984-12-27

Family

ID=9290167

Family Applications (1)

Application Number Title Priority Date Filing Date
NO842529A NO842529L (no) 1983-06-24 1984-06-22 Fremgangsmaate for fremstilling av salter av metyllevallorfanium.

Country Status (18)

Country Link
US (1) US4735947A (de)
EP (1) EP0135402B1 (de)
JP (1) JPS6019768A (de)
KR (1) KR850000403A (de)
AT (1) ATE30419T1 (de)
AU (1) AU576767B2 (de)
CA (1) CA1220199A (de)
DE (1) DE3466984D1 (de)
DK (1) DK160042C (de)
ES (1) ES8503336A1 (de)
FI (1) FI842531A7 (de)
FR (1) FR2547820B1 (de)
GR (1) GR79771B (de)
IL (1) IL72156A (de)
NO (1) NO842529L (de)
NZ (1) NZ208629A (de)
PT (1) PT78768B (de)
ZA (1) ZA844759B (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050191340A1 (en) * 2002-08-09 2005-09-01 Gruenenthal Gmbh Opioid-receptor antagonists in transdermal systems having buprenorphine

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1179915A (fr) * 1953-11-12 1959-05-29 Hoffmann La Roche Procédé pour la préparation de dérivés de morphinane
US3101339A (en) * 1958-10-30 1963-08-20 Boehringer Sohn Ingelheim Quaternary salts of normorphine and its acylated derivatives
US4176186A (en) * 1978-07-28 1979-11-27 Boehringer Ingelheim Gmbh Quaternary derivatives of noroxymorphone which relieve intestinal immobility
FR2514644A1 (fr) * 1981-10-19 1983-04-22 Sanofi Sa Composition pharmaceutique a action antagoniste peripherique des opiaces
FR2538805B1 (fr) * 1982-12-30 1985-10-25 Sanofi Sa Procede de preparation d'halomethylate de levallorphan et composition pharmaceutique antagoniste peripherique des opiaces en contenant

Also Published As

Publication number Publication date
FI842531L (fi) 1984-12-25
AU576767B2 (en) 1988-09-08
JPS6019768A (ja) 1985-01-31
FI842531A0 (fi) 1984-06-21
EP0135402A1 (de) 1985-03-27
IL72156A (en) 1987-08-31
GR79771B (de) 1984-10-31
PT78768A (fr) 1984-07-01
ZA844759B (en) 1985-02-27
DK160042C (da) 1991-06-17
PT78768B (fr) 1986-07-14
FR2547820A1 (fr) 1984-12-28
ATE30419T1 (de) 1987-11-15
NZ208629A (en) 1987-08-31
FR2547820B1 (fr) 1986-04-18
DE3466984D1 (en) 1987-12-03
ES533622A0 (es) 1985-02-16
AU2972584A (en) 1985-01-03
DK160042B (da) 1991-01-21
EP0135402B1 (de) 1987-10-28
ES8503336A1 (es) 1985-02-16
KR850000403A (ko) 1985-02-27
US4735947A (en) 1988-04-05
FI842531A7 (fi) 1984-12-25
CA1220199A (en) 1987-04-07
DK301584A (da) 1984-12-25
IL72156A0 (en) 1984-10-31
DK301584D0 (da) 1984-06-20

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