NO346587B1 - Capsaicin derivatives in the treatment of idiopathic pulmonary fibrosis - Google Patents
Capsaicin derivatives in the treatment of idiopathic pulmonary fibrosis Download PDFInfo
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- NO346587B1 NO346587B1 NO20210693A NO20210693A NO346587B1 NO 346587 B1 NO346587 B1 NO 346587B1 NO 20210693 A NO20210693 A NO 20210693A NO 20210693 A NO20210693 A NO 20210693A NO 346587 B1 NO346587 B1 NO 346587B1
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/235—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Priority Applications (6)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| NO20210693A NO346587B1 (en) | 2021-06-02 | 2021-06-02 | Capsaicin derivatives in the treatment of idiopathic pulmonary fibrosis |
| US18/564,031 US20240277637A1 (en) | 2021-06-02 | 2022-06-01 | Capsaicin derivatives in the treatment of idiopathic pulmonary fibrosis |
| CN202280039778.6A CN117412742A (zh) | 2021-06-02 | 2022-06-01 | 治疗特发性肺纤维化的辣椒素衍生物 |
| JP2023574384A JP2024520650A (ja) | 2021-06-02 | 2022-06-01 | 特発性肺線維症の処置におけるカプサイシン誘導体 |
| EP22731584.3A EP4346789A1 (en) | 2021-06-02 | 2022-06-01 | Capsaicin derivatives in the treatment of idiopathic pulmonary fibrosis |
| PCT/EP2022/064876 WO2022253884A1 (en) | 2021-06-02 | 2022-06-01 | Capsaicin derivatives in the treatment of idiopathic pulmonary fibrosis |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| NO20210693A NO346587B1 (en) | 2021-06-02 | 2021-06-02 | Capsaicin derivatives in the treatment of idiopathic pulmonary fibrosis |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO346587B1 true NO346587B1 (en) | 2022-10-17 |
| NO20210693A1 NO20210693A1 (enExample) | 2022-10-17 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20210693A NO346587B1 (en) | 2021-06-02 | 2021-06-02 | Capsaicin derivatives in the treatment of idiopathic pulmonary fibrosis |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20240277637A1 (enExample) |
| EP (1) | EP4346789A1 (enExample) |
| JP (1) | JP2024520650A (enExample) |
| CN (1) | CN117412742A (enExample) |
| NO (1) | NO346587B1 (enExample) |
| WO (1) | WO2022253884A1 (enExample) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NO348880B1 (en) * | 2023-03-13 | 2025-06-30 | Axichem Ab | Physical performance aid |
Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1530466A2 (en) * | 2002-08-16 | 2005-05-18 | Boehringer Ingelheim Pharma KG | Use of lck inhibitor for treatment of immunologic diseases |
| WO2013006135A1 (en) * | 2011-07-07 | 2013-01-10 | Millqvist Eva | Cough reducing product |
| WO2015160842A1 (en) * | 2014-04-14 | 2015-10-22 | Flex Pharma, Inc. | Methods and formulatiions of capsaicinoids and capsinoids |
| WO2017160156A1 (en) * | 2016-03-18 | 2017-09-21 | Axichem Ab | Synthetic capasaicin analogs as trpv1 agonists |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NO20034069L (no) | 2003-09-12 | 2005-03-14 | Aximed As | Fremstilling og bruk av capsaicinderivater |
| JP7412424B2 (ja) * | 2018-09-18 | 2024-01-12 | ブリストル－マイヤーズ スクイブ カンパニー | Ｌｐａアンタゴニストとしてのオキサビシクロ酸 |
| WO2020160225A1 (en) * | 2019-01-30 | 2020-08-06 | Ohio State Innovation Foundation | ESTROGEN RECEPTOR BETA (ERβ) AGONISTS FOR THE TREATMENT OF FIBROTIC CONDITIONS |
| WO2020191501A1 (en) * | 2019-03-27 | 2020-10-01 | Algernon Pharmaceuticals Inc. | Methods and uses of bemithyl and derivatives for treating lung disease, fatty liver disease, and kidney disorders |
| WO2020227331A1 (en) * | 2019-05-06 | 2020-11-12 | Inspira, LLC | Chemical entities, pharmaceutical formulations, and methods for treating fibrosis |
| CN114026072A (zh) * | 2019-06-25 | 2022-02-08 | 北京泰德制药股份有限公司 | 治疗特发性肺纤维化的方法 |
| NO345530B1 (en) | 2020-03-20 | 2021-03-29 | Axichem As | Synthesis of capsaicin derivatives |
-
2021
- 2021-06-02 NO NO20210693A patent/NO346587B1/en unknown
-
2022
- 2022-06-01 WO PCT/EP2022/064876 patent/WO2022253884A1/en not_active Ceased
- 2022-06-01 US US18/564,031 patent/US20240277637A1/en active Pending
- 2022-06-01 JP JP2023574384A patent/JP2024520650A/ja active Pending
- 2022-06-01 EP EP22731584.3A patent/EP4346789A1/en active Pending
- 2022-06-01 CN CN202280039778.6A patent/CN117412742A/zh active Pending
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1530466A2 (en) * | 2002-08-16 | 2005-05-18 | Boehringer Ingelheim Pharma KG | Use of lck inhibitor for treatment of immunologic diseases |
| WO2013006135A1 (en) * | 2011-07-07 | 2013-01-10 | Millqvist Eva | Cough reducing product |
| WO2015160842A1 (en) * | 2014-04-14 | 2015-10-22 | Flex Pharma, Inc. | Methods and formulatiions of capsaicinoids and capsinoids |
| WO2017160156A1 (en) * | 2016-03-18 | 2017-09-21 | Axichem Ab | Synthetic capasaicin analogs as trpv1 agonists |
Non-Patent Citations (1)
| Title |
|---|
| LIN-MING, L. et al. Effect of small dose capsaicin for treatment of pulmonary fibrosis in mice and its mechanism, Chinese Journal of Applied Physiology, May 2020, vol.36, Nr. 3, (machine translated into English), page 216-222, Dated: 01.01.0001 * |
Also Published As
| Publication number | Publication date |
|---|---|
| NO20210693A1 (enExample) | 2022-10-17 |
| JP2024520650A (ja) | 2024-05-24 |
| US20240277637A1 (en) | 2024-08-22 |
| CN117412742A (zh) | 2024-01-16 |
| WO2022253884A1 (en) | 2022-12-08 |
| EP4346789A1 (en) | 2024-04-10 |
| WO2022253884A4 (en) | 2023-01-12 |
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