NO20085252L - Imidazolidinon Kv1.5 kaliumkanalinhibitorer - Google Patents
Imidazolidinon Kv1.5 kaliumkanalinhibitorerInfo
- Publication number
- NO20085252L NO20085252L NO20085252A NO20085252A NO20085252L NO 20085252 L NO20085252 L NO 20085252L NO 20085252 A NO20085252 A NO 20085252A NO 20085252 A NO20085252 A NO 20085252A NO 20085252 L NO20085252 L NO 20085252L
- Authority
- NO
- Norway
- Prior art keywords
- potassium channel
- channel inhibitors
- imidazolidinone
- present
- relates
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/30—Oxygen or sulfur atoms
- C07D233/32—One oxygen atom
- C07D233/38—One oxygen atom with acyl radicals or hetero atoms directly attached to ring nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4166—1,3-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
Abstract
(I) Foreliggende oppfinnelse angår 1-N-amino-2-imidazolidinoner (I) og derivater derav som er effektive som Kv1.5 kaliumkanalinhibitorer som tilveiebringer atrial-selektive antiarytmiske midler. Foreliggende oppfinnelse angår videre preparater omfattende nevnte Kv1.5 kaliumkanalinhibitorer og metoder for behandling av hjertearytmi.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US81509106P | 2006-06-20 | 2006-06-20 | |
PCT/US2007/071587 WO2007149874A1 (en) | 2006-06-20 | 2007-06-19 | Imidazolidinone kv1.5 potassium channel inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20085252L true NO20085252L (no) | 2009-01-13 |
Family
ID=38582320
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20085252A NO20085252L (no) | 2006-06-20 | 2008-12-16 | Imidazolidinon Kv1.5 kaliumkanalinhibitorer |
Country Status (20)
Country | Link |
---|---|
US (2) | US7504517B2 (no) |
EP (1) | EP2035392A1 (no) |
JP (1) | JP2009541343A (no) |
KR (1) | KR20090021223A (no) |
CN (1) | CN101573341A (no) |
AR (1) | AR061523A1 (no) |
AU (1) | AU2007260985A1 (no) |
BR (1) | BRPI0713320A2 (no) |
CA (1) | CA2655574A1 (no) |
CL (1) | CL2007001794A1 (no) |
CO (1) | CO6150173A2 (no) |
CR (1) | CR10527A (no) |
EC (1) | ECSP088994A (no) |
MX (1) | MX2008016399A (no) |
NO (1) | NO20085252L (no) |
PE (1) | PE20080942A1 (no) |
RU (1) | RU2008150465A (no) |
TW (1) | TW200815363A (no) |
WO (1) | WO2007149874A1 (no) |
ZA (1) | ZA200810763B (no) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2035392A1 (en) * | 2006-06-20 | 2009-03-18 | Wyeth a Corporation of the State of Delaware | Imidazole kv1. 5 potassium channel inhibitors |
CN101544580B (zh) * | 2009-04-28 | 2019-03-15 | 大连凯飞精细化工有限公司 | R-alpha-氨基-4-甲氧基苯乙酰胺的合成方法 |
Family Cites Families (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4099009A (en) * | 1977-04-11 | 1978-07-04 | Morton-Norwick Products, Inc. | 1-(4-chlorophenyl)-3-(1-ureido)-2-imidazolidinone |
SK94393A3 (en) | 1992-09-11 | 1994-08-10 | Thomae Gmbh Dr K | Cyclic derivatives of urea, process for their production and their pharmaceutical agents with the content of those |
DE4332168A1 (de) | 1993-02-22 | 1995-03-23 | Thomae Gmbh Dr K | Cyclische Derivate, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung |
JP2000501111A (ja) | 1996-01-26 | 2000-02-02 | バーテックス ファーマシューティカルズ インコーポレイテッド | アスパルチルプロテアーゼインヒビター |
AU716153B2 (en) | 1996-04-03 | 2000-02-17 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
US7129359B2 (en) * | 2002-07-09 | 2006-10-31 | National Health Research Institutes | Imidazolidinone compounds |
BR0214437A (pt) | 2001-11-30 | 2004-10-13 | Lilly Co Eli | Composto, composição farmacêutica, métodos de modular um receptor ativado por proliferador de peroxissoma, de tratar e de prevenir a diabete melito, e de tratar a sìndrome x, e doenças cardiovasculares em um mamìfero, e, uso de um composto |
WO2003057214A1 (en) | 2001-12-28 | 2003-07-17 | Somatocor Pharmaceuticals, Inc. | Imidazolidin-2,4-dione derivatives as non-peptide somatostatin receptor ligands |
AU2003302027A1 (en) | 2002-11-21 | 2004-06-15 | Vicore Pharma Ab | New tricyclic angiotensin ii agonists |
JP2004262903A (ja) | 2003-03-04 | 2004-09-24 | Japan Science & Technology Agency | アジリジン類の製造方法 |
US7259174B2 (en) * | 2004-05-25 | 2007-08-21 | National Health Research Institutes | Imidazolidinone compounds |
TW200624429A (en) * | 2004-09-07 | 2006-07-16 | Glaxo Group Ltd | Novel cysteine protease inhibitors |
KR100677149B1 (ko) * | 2004-11-12 | 2007-02-02 | 삼성전자주식회사 | 잉크 조성물 |
EP2035392A1 (en) * | 2006-06-20 | 2009-03-18 | Wyeth a Corporation of the State of Delaware | Imidazole kv1. 5 potassium channel inhibitors |
-
2007
- 2007-06-19 EP EP07798773A patent/EP2035392A1/en not_active Withdrawn
- 2007-06-19 BR BRPI0713320-0A patent/BRPI0713320A2/pt not_active IP Right Cessation
- 2007-06-19 WO PCT/US2007/071587 patent/WO2007149874A1/en active Application Filing
- 2007-06-19 CA CA002655574A patent/CA2655574A1/en not_active Abandoned
- 2007-06-19 KR KR1020097000926A patent/KR20090021223A/ko not_active Application Discontinuation
- 2007-06-19 JP JP2009516686A patent/JP2009541343A/ja not_active Withdrawn
- 2007-06-19 MX MX2008016399A patent/MX2008016399A/es unknown
- 2007-06-19 CN CNA2007800285697A patent/CN101573341A/zh active Pending
- 2007-06-19 AU AU2007260985A patent/AU2007260985A1/en not_active Abandoned
- 2007-06-19 AR ARP070102688A patent/AR061523A1/es unknown
- 2007-06-19 CL CL2007001794A patent/CL2007001794A1/es unknown
- 2007-06-19 PE PE2007000779A patent/PE20080942A1/es not_active Application Discontinuation
- 2007-06-19 US US11/765,359 patent/US7504517B2/en not_active Expired - Fee Related
- 2007-06-19 RU RU2008150465/04A patent/RU2008150465A/ru not_active Application Discontinuation
- 2007-06-20 TW TW096122064A patent/TW200815363A/zh unknown
-
2008
- 2008-11-06 US US12/266,212 patent/US7803827B2/en not_active Expired - Fee Related
- 2008-12-16 NO NO20085252A patent/NO20085252L/no not_active Application Discontinuation
- 2008-12-18 CR CR10527A patent/CR10527A/es not_active Application Discontinuation
- 2008-12-19 EC EC2008008994A patent/ECSP088994A/es unknown
- 2008-12-19 ZA ZA200810763A patent/ZA200810763B/xx unknown
- 2008-12-19 CO CO08135447A patent/CO6150173A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
WO2007149874A8 (en) | 2008-03-20 |
AR061523A1 (es) | 2008-09-03 |
US20070299120A1 (en) | 2007-12-27 |
US7803827B2 (en) | 2010-09-28 |
CR10527A (es) | 2009-02-19 |
CA2655574A1 (en) | 2007-12-27 |
TW200815363A (en) | 2008-04-01 |
CN101573341A (zh) | 2009-11-04 |
JP2009541343A (ja) | 2009-11-26 |
ECSP088994A (es) | 2009-01-30 |
MX2008016399A (es) | 2009-02-03 |
WO2007149874A1 (en) | 2007-12-27 |
BRPI0713320A2 (pt) | 2012-02-07 |
ZA200810763B (en) | 2009-09-30 |
AU2007260985A1 (en) | 2007-12-27 |
US7504517B2 (en) | 2009-03-17 |
KR20090021223A (ko) | 2009-02-27 |
EP2035392A1 (en) | 2009-03-18 |
CL2007001794A1 (es) | 2008-01-18 |
US20090069342A1 (en) | 2009-03-12 |
CO6150173A2 (es) | 2010-04-20 |
RU2008150465A (ru) | 2010-07-27 |
PE20080942A1 (es) | 2008-09-03 |
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Legal Events
Date | Code | Title | Description |
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FC2A | Withdrawal, rejection or dismissal of laid open patent application |