NO20084278L - Bezothiazol derivatives as beta2 adrenoreceptor agonists - Google Patents
Bezothiazol derivatives as beta2 adrenoreceptor agonistsInfo
- Publication number
- NO20084278L NO20084278L NO20084278A NO20084278A NO20084278L NO 20084278 L NO20084278 L NO 20084278L NO 20084278 A NO20084278 A NO 20084278A NO 20084278 A NO20084278 A NO 20084278A NO 20084278 L NO20084278 L NO 20084278L
- Authority
- NO
- Norway
- Prior art keywords
- bezothiazole
- derivatives
- adrenoreceptor agonists
- beta2 adrenoreceptor
- beta2
- Prior art date
Links
Classifications
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- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/428—Thiazoles condensed with carbocyclic rings
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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Abstract
Foreliggende oppfinnelse angår forbindelser med formel (I): en fremgangsmåte for fremstilling av dem, intermediatforbindelser for fremgangsmåten og anvendelsen av forbindelsene for fremstilling av et medikament for anvendelse ved behandling av sykdommer slike som ARDS, lungeemfysem, bronkitt, bronkiekstasi, COPD, astma eller rhinitt. Forbindelsene er |32-adrenoreseptoragonister.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US78273306P | 2006-03-14 | 2006-03-14 | |
US86265106P | 2006-10-24 | 2006-10-24 | |
PCT/SE2007/000233 WO2007106016A1 (en) | 2006-03-14 | 2007-03-12 | Bezothiazol derivatives as beta2 adrenoreceptor agonists |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20084278L true NO20084278L (no) | 2008-10-30 |
Family
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Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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NO20084278A NO20084278L (no) | 2006-03-14 | 2008-10-13 | Bezothiazol derivatives as beta2 adrenoreceptor agonists |
Country Status (15)
Country | Link |
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US (1) | US7951954B2 (no) |
EP (1) | EP1996566A1 (no) |
JP (1) | JP2009530272A (no) |
KR (1) | KR20080103104A (no) |
AR (1) | AR059842A1 (no) |
AU (1) | AU2007225471A1 (no) |
BR (1) | BRPI0709589A2 (no) |
CA (1) | CA2644014A1 (no) |
EC (1) | ECSP088741A (no) |
IL (1) | IL193530A0 (no) |
NO (1) | NO20084278L (no) |
RU (1) | RU2008136553A (no) |
TW (1) | TW200745067A (no) |
UY (1) | UY30206A1 (no) |
WO (1) | WO2007106016A1 (no) |
Families Citing this family (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200738658A (en) | 2005-08-09 | 2007-10-16 | Astrazeneca Ab | Novel compounds |
TW200738659A (en) * | 2005-08-29 | 2007-10-16 | Astrazeneca Ab | Novel compounds |
TW200745067A (en) | 2006-03-14 | 2007-12-16 | Astrazeneca Ab | Novel compounds |
TW200833670A (en) * | 2006-12-20 | 2008-08-16 | Astrazeneca Ab | Novel compounds 569 |
GB0702458D0 (en) * | 2007-02-08 | 2007-03-21 | Astrazeneca Ab | Salts 668 |
WO2009037503A2 (en) * | 2007-09-18 | 2009-03-26 | Astrazeneca Ab | New combination - 012 for the treatment of respiratory diseases |
WO2009154557A1 (en) | 2008-06-18 | 2009-12-23 | Astrazeneca Ab | Benzoxazinone derivatives acting as beta2-adrenoreceptor agonist for the treatment of respiratory disorders |
EP2361242B1 (en) | 2008-10-17 | 2018-08-01 | Oryzon Genomics, S.A. | Oxidase inhibitors and their use |
WO2010084160A1 (en) | 2009-01-21 | 2010-07-29 | Oryzon Genomics S.A. | Phenylcyclopropylamine derivatives and their medical use |
US8859555B2 (en) | 2009-09-25 | 2014-10-14 | Oryzon Genomics S.A. | Lysine Specific Demethylase-1 inhibitors and their use |
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2007
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- 2007-03-12 WO PCT/SE2007/000233 patent/WO2007106016A1/en active Application Filing
- 2007-03-12 CA CA002644014A patent/CA2644014A1/en not_active Abandoned
- 2007-03-12 AU AU2007225471A patent/AU2007225471A1/en not_active Abandoned
- 2007-03-12 EP EP07716051A patent/EP1996566A1/en not_active Withdrawn
- 2007-03-12 RU RU2008136553/04A patent/RU2008136553A/ru not_active Application Discontinuation
- 2007-03-12 BR BRPI0709589-9A patent/BRPI0709589A2/pt not_active IP Right Cessation
- 2007-03-12 US US12/282,634 patent/US7951954B2/en not_active Expired - Fee Related
- 2007-03-12 KR KR1020087024962A patent/KR20080103104A/ko not_active Application Discontinuation
- 2007-03-12 JP JP2009500323A patent/JP2009530272A/ja not_active Withdrawn
- 2007-03-14 AR ARP070101043A patent/AR059842A1/es unknown
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- 2008-09-15 EC EC2008008741A patent/ECSP088741A/es unknown
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BRPI0709589A2 (pt) | 2011-07-19 |
CA2644014A1 (en) | 2007-09-20 |
US7951954B2 (en) | 2011-05-31 |
TW200745067A (en) | 2007-12-16 |
UY30206A1 (es) | 2007-10-31 |
JP2009530272A (ja) | 2009-08-27 |
RU2008136553A (ru) | 2010-04-20 |
KR20080103104A (ko) | 2008-11-26 |
IL193530A0 (en) | 2009-02-11 |
AU2007225471A1 (en) | 2007-09-20 |
AR059842A1 (es) | 2008-04-30 |
EP1996566A1 (en) | 2008-12-03 |
ECSP088741A (es) | 2008-10-31 |
US20090062259A1 (en) | 2009-03-05 |
WO2007106016A1 (en) | 2007-09-20 |
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